KR850000439A - 티아졸리딘 유도체의 제조방법 - Google Patents
티아졸리딘 유도체의 제조방법 Download PDFInfo
- Publication number
- KR850000439A KR850000439A KR1019840003520A KR840003520A KR850000439A KR 850000439 A KR850000439 A KR 850000439A KR 1019840003520 A KR1019840003520 A KR 1019840003520A KR 840003520 A KR840003520 A KR 840003520A KR 850000439 A KR850000439 A KR 850000439A
- Authority
- KR
- South Korea
- Prior art keywords
- benzopyran
- fluoro
- dihydro
- thiazolidine
- dioxospyro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 238000000034 method Methods 0.000 title claims 4
- 150000003548 thiazolidines Chemical class 0.000 title 1
- 150000001875 compounds Chemical class 0.000 claims 8
- 229910052739 hydrogen Inorganic materials 0.000 claims 5
- 239000001257 hydrogen Substances 0.000 claims 5
- 229910052736 halogen Inorganic materials 0.000 claims 4
- 150000002367 halogens Chemical class 0.000 claims 4
- 150000002431 hydrogen Chemical class 0.000 claims 4
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 claims 4
- -1 (±) -6-fluoro-8-acetamido-2,3-dihydrospiro [4H-1-benzopyran-4,5'-thiazolidine] Chemical compound 0.000 claims 3
- 125000000217 alkyl group Chemical group 0.000 claims 3
- 125000004093 cyano group Chemical group *C#N 0.000 claims 3
- FZXBGACPNKBGBJ-UHFFFAOYSA-N 6'-fluorospiro[1,3-thiazolidine-5,4'-2,3-dihydrochromene]-2,4-dione Chemical compound C12=CC(F)=CC=C2OCCC21SC(=O)NC2=O FZXBGACPNKBGBJ-UHFFFAOYSA-N 0.000 claims 2
- KXDAEFPNCMNJSK-UHFFFAOYSA-N Benzamide Chemical compound NC(=O)C1=CC=CC=C1 KXDAEFPNCMNJSK-UHFFFAOYSA-N 0.000 claims 2
- WSFSSNUMVMOOMR-UHFFFAOYSA-N Formaldehyde Chemical group O=C WSFSSNUMVMOOMR-UHFFFAOYSA-N 0.000 claims 2
- ZHNUHDYFZUAESO-UHFFFAOYSA-N Formamide Chemical compound NC=O ZHNUHDYFZUAESO-UHFFFAOYSA-N 0.000 claims 2
- NINIDFKCEFEMDL-UHFFFAOYSA-N Sulfur Chemical group [S] NINIDFKCEFEMDL-UHFFFAOYSA-N 0.000 claims 2
- 125000002252 acyl group Chemical group 0.000 claims 2
- 125000003277 amino group Chemical group 0.000 claims 2
- 150000001768 cations Chemical class 0.000 claims 2
- 239000007795 chemical reaction product Substances 0.000 claims 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 claims 2
- 238000004519 manufacturing process Methods 0.000 claims 2
- 150000003839 salts Chemical class 0.000 claims 2
- 229910052717 sulfur Chemical group 0.000 claims 2
- 239000011593 sulfur Chemical group 0.000 claims 2
- UWDNKLDNNGZHMQ-UHFFFAOYSA-N 6'-fluoro-2,4-dioxospiro[1,3-thiazolidine-5,4'-2,3-dihydrochromene]-8'-carbonitrile Chemical compound C12=CC(F)=CC(C#N)=C2OCCC21SC(=O)NC2=O UWDNKLDNNGZHMQ-UHFFFAOYSA-N 0.000 claims 1
- KILSWTGTFSIAIC-UHFFFAOYSA-N 6'-fluoro-8'-nitrospiro[1,3-thiazolidine-5,4'-2,3-dihydrochromene]-2,4-dione Chemical compound [O-][N+](=O)C1=CC(F)=CC2=C1OCCC21SC(=O)NC1=O KILSWTGTFSIAIC-UHFFFAOYSA-N 0.000 claims 1
- LWILNUCJTYZZQI-UHFFFAOYSA-N 8'-amino-6'-fluorospiro[1,3-thiazolidine-5,4'-2,3-dihydrochromene]-2,4-dione Chemical compound NC1=CC(F)=CC2=C1OCCC21SC(=O)NC1=O LWILNUCJTYZZQI-UHFFFAOYSA-N 0.000 claims 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 claims 1
- XBDQKXXYIPTUBI-UHFFFAOYSA-M Propionate Chemical compound CCC([O-])=O XBDQKXXYIPTUBI-UHFFFAOYSA-M 0.000 claims 1
- XSQUKJJJFZCRTK-UHFFFAOYSA-N Urea Chemical compound NC(N)=O XSQUKJJJFZCRTK-UHFFFAOYSA-N 0.000 claims 1
- UFIDINVHKAOTND-UHFFFAOYSA-N [6'-fluoro-3-(4-nitrophenyl)-2,4-dioxospiro[1,3-thiazolidine-5,4'-2,3-dihydrochromene]-8'-yl]carbamic acid Chemical compound C1COC2=C(C13C(=O)N(C(=O)S3)C4=CC=C(C=C4)[N+](=O)[O-])C=C(C=C2NC(=O)O)F UFIDINVHKAOTND-UHFFFAOYSA-N 0.000 claims 1
- KXKVLQRXCPHEJC-UHFFFAOYSA-N acetic acid trimethyl ester Natural products COC(C)=O KXKVLQRXCPHEJC-UHFFFAOYSA-N 0.000 claims 1
- 239000002253 acid Substances 0.000 claims 1
- 125000003710 aryl alkyl group Chemical group 0.000 claims 1
- 125000003118 aryl group Chemical group 0.000 claims 1
- QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical group [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 claims 1
- 239000004202 carbamide Substances 0.000 claims 1
- 125000003917 carbamoyl group Chemical group [H]N([H])C(*)=O 0.000 claims 1
- 125000001160 methoxycarbonyl group Chemical group [H]C([H])([H])OC(*)=O 0.000 claims 1
- 230000001546 nitrifying effect Effects 0.000 claims 1
- 229910052760 oxygen Inorganic materials 0.000 claims 1
- 239000001301 oxygen Substances 0.000 claims 1
- XIPFMBOWZXULIA-UHFFFAOYSA-N pivalamide Chemical compound CC(C)(C)C(N)=O XIPFMBOWZXULIA-UHFFFAOYSA-N 0.000 claims 1
- LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 claims 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Enzymes And Modification Thereof (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH343283 | 1983-06-23 | ||
| CH3432/83 | 1983-06-23 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR850000439A true KR850000439A (ko) | 1985-02-27 |
Family
ID=4255846
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1019840003520A Withdrawn KR850000439A (ko) | 1983-06-23 | 1984-06-22 | 티아졸리딘 유도체의 제조방법 |
Country Status (5)
| Country | Link |
|---|---|
| JP (1) | JPS6013774A (enrdf_load_stackoverflow) |
| KR (1) | KR850000439A (enrdf_load_stackoverflow) |
| ES (1) | ES541706A0 (enrdf_load_stackoverflow) |
| GR (1) | GR81637B (enrdf_load_stackoverflow) |
| ZA (1) | ZA844557B (enrdf_load_stackoverflow) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS56102431A (en) * | 1980-01-16 | 1981-08-15 | Inoue Japax Res Inc | Arc discharge work device |
| JPH06772B2 (ja) * | 1984-07-09 | 1994-01-05 | 鐘淵化学工業株式会社 | ３―（４―フルオロフエノキシ）プロピオニトリルを用いる６―フルオロ―４―クロマノンの製造法 |
| JPS61200991A (ja) * | 1985-03-04 | 1986-09-05 | Sanwa Kagaku Kenkyusho:Kk | スピロ―３―ヘテロアゾリジン化合物、その製法及びそれを有効成分とする糖尿病合併症の予防及び治療剤 |
| CA2568186C (en) * | 2004-05-24 | 2011-11-15 | Amgen Inc. | Inhibitors of 11-beta-hydroxy steroid dehydrogenase type 1 |
| US8686011B2 (en) | 2004-05-24 | 2014-04-01 | Amgen Inc. | Inhibitors of 11-β-hydroxy steroid dehydrogenase type 1 |
-
1984
- 1984-06-15 ZA ZA844557A patent/ZA844557B/xx unknown
- 1984-06-22 KR KR1019840003520A patent/KR850000439A/ko not_active Withdrawn
- 1984-06-22 GR GR75090A patent/GR81637B/el unknown
- 1984-06-22 JP JP59127641A patent/JPS6013774A/ja active Pending
-
1985
- 1985-03-29 ES ES541706A patent/ES541706A0/es active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| ES8602717A1 (es) | 1985-12-01 |
| JPS6013774A (ja) | 1985-01-24 |
| ZA844557B (en) | 1985-02-27 |
| GR81637B (enrdf_load_stackoverflow) | 1984-12-11 |
| ES541706A0 (es) | 1985-12-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PA0109 | Patent application |
Patent event code: PA01091R01D Comment text: Patent Application Patent event date: 19840622 |
|
| PG1501 | Laying open of application | ||
| PC1202 | Submission of document of withdrawal before decision of registration |
Comment text: [Withdrawal of Procedure relating to Patent, etc.] Withdrawal (Abandonment) Patent event code: PC12021R01D Patent event date: 19890622 |
|
| WITB | Written withdrawal of application |