KR20250151389A - 치환 피라졸로피리미딘 화합물 및 그의 의약 용도 - Google Patents

치환 피라졸로피리미딘 화합물 및 그의 의약 용도

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KR20250151389A
KR20250151389A KR1020257027024A KR20257027024A KR20250151389A KR 20250151389 A KR20250151389 A KR 20250151389A KR 1020257027024 A KR1020257027024 A KR 1020257027024A KR 20257027024 A KR20257027024 A KR 20257027024A KR 20250151389 A KR20250151389 A KR 20250151389A
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유스케 오바
가오루 아다치
겐타로 사쿠라이
심페이 사토
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니뽄 다바코 산교 가부시키가이샤
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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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    • A61P19/00Drugs for skeletal disorders
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    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
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    • C07DHETEROCYCLIC COMPOUNDS
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  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Rheumatology (AREA)
  • Cardiology (AREA)
  • Psychology (AREA)
  • Epidemiology (AREA)
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  • Immunology (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
KR1020257027024A 2023-02-24 2024-02-22 치환 피라졸로피리미딘 화합물 및 그의 의약 용도 Pending KR20250151389A (ko)

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JPJP-P-2023-027432 2023-02-24
JP2023027432 2023-02-24
PCT/JP2024/006433 WO2024177127A1 (ja) 2023-02-24 2024-02-22 置換ピラゾロピリミジン化合物及びその医薬用途

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KR20250151389A true KR20250151389A (ko) 2025-10-21

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EP (1) EP4671247A1 (enExample)
JP (2) JP7737490B2 (enExample)
KR (1) KR20250151389A (enExample)
CN (1) CN120752239A (enExample)
AR (1) AR131919A1 (enExample)
AU (1) AU2024226032A1 (enExample)
CO (1) CO2025011311A2 (enExample)
IL (1) IL322520A (enExample)
MX (1) MX2025009965A (enExample)
TW (1) TW202448887A (enExample)
WO (1) WO2024177127A1 (enExample)

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WO2025140708A1 (zh) * 2023-12-31 2025-07-03 杭州百新生物医药科技有限公司 吡唑并嘧啶类化合物及其医药用途
WO2025153532A1 (en) 2024-01-16 2025-07-24 NodThera Limited Nlrp3 inhibitors and glp-1 agonists combination therapies

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PL3064498T3 (pl) * 2013-10-30 2020-03-31 Shanghai Hengrui Pharmaceutical Co. Ltd. Pirazolopirymidon lub pochodne pirolotriazonu, sposób ich otrzymywania i ich zastosowania farmaceutyczne
WO2017205766A1 (en) * 2016-05-27 2017-11-30 Pharmacyclics Llc Inhibitors of interleukin-1 receptor-associated kinase
ES2930151T3 (es) * 2019-01-14 2022-12-07 Innate Tumor Immunity Inc Moduladores heterocíclicos de NLRP3, para su uso en el tratamiento del cáncer
KR102865929B1 (ko) * 2019-01-14 2025-09-29 인네이트 튜머 이뮤니티, 인코포레이티드 Nlrp3 조정제
WO2021132577A1 (ja) * 2019-12-27 2021-07-01 日本たばこ産業株式会社 アシルスルファミド化合物及びその医薬用途
US20240382488A1 (en) * 2021-03-29 2024-11-21 Halia Therapeutics, Inc. Nek7 inhibitors
JP2024513227A (ja) * 2021-04-05 2024-03-22 ハリア・セラピューティクス・インコーポレイテッド Nek7阻害剤
US20240287079A1 (en) * 2021-08-31 2024-08-29 Japan Tobacco Inc. 6-aminopyrazolopyrimidine compound and pharmaceutical use thereof
WO2024048519A1 (ja) * 2022-08-29 2024-03-07 日本たばこ産業株式会社 ピラゾロピリミジン化合物及びその医薬用途
AU2024255473A1 (en) * 2023-04-14 2025-10-16 Takeda Pharmaceutical Company Limited Pyrazolopyrimidine derivatives as inhibitors of nlrp3

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