KR20250004844A - 벤조트리아졸 화합물 - Google Patents

벤조트리아졸 화합물 Download PDF

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KR20250004844A
KR20250004844A KR1020247038642A KR20247038642A KR20250004844A KR 20250004844 A KR20250004844 A KR 20250004844A KR 1020247038642 A KR1020247038642 A KR 1020247038642A KR 20247038642 A KR20247038642 A KR 20247038642A KR 20250004844 A KR20250004844 A KR 20250004844A
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South Korea
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group
methyl
compound
ethyl
dihydro
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Korean (ko)
Inventor
요시히로 오구라
리에코 다카노
준야 가와이
뎃페이 후지모토
마사하루 이누이
마사후미 오후쿠
마사키 미야자키
마사야 후지이
겐 이시이
와카나 요코제키
가즈야 오타케
슌스케 다카시마
šœ스케 다카시마
마사후미 안도
Original Assignee
다이이찌 산쿄 가부시키가이샤
교토 야쿠힝 고교 가부시키가이샤
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Publication of KR20250004844A publication Critical patent/KR20250004844A/ko
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/554—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having at least one nitrogen and one sulfur as ring hetero atoms, e.g. clothiapine, diltiazem
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  • Diabetes (AREA)
  • Urology & Nephrology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Heart & Thoracic Surgery (AREA)
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  • Hospice & Palliative Care (AREA)
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  • Endocrinology (AREA)
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  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
KR1020247038642A 2022-04-28 2023-04-27 벤조트리아졸 화합물 Pending KR20250004844A (ko)

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JPJP-P-2022-075223 2022-04-28
JP2022075223 2022-04-28
PCT/JP2023/016629 WO2023210741A1 (ja) 2022-04-28 2023-04-27 ベンゾトリアゾール化合物

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US (3) US20250282724A1 (https=)
EP (1) EP4509504A4 (https=)
JP (1) JP7605446B2 (https=)
KR (1) KR20250004844A (https=)
CN (1) CN119173511A (https=)
AU (1) AU2023259936A1 (https=)
CA (1) CA3256688A1 (https=)
CO (1) CO2024014914A2 (https=)
IL (1) IL316449A (https=)
MX (1) MX2024013242A (https=)
TW (1) TW202404984A (https=)
WO (1) WO2023210741A1 (https=)
ZA (1) ZA202408061B (https=)

Citations (11)

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WO2015092713A1 (en) 2013-12-18 2015-06-25 Glaxosmithkline Intellectual Property Development Limited Nrf2 regulators
WO2016202253A1 (en) 2015-06-15 2016-12-22 Glaxosmithkline Intellectual Property Development Limited Nrf2 regulators
WO2016203401A1 (en) 2015-06-15 2016-12-22 Glaxosmithkline Intellectual Property Development Limited Nrf2 regulators
WO2016203400A1 (en) 2015-06-15 2016-12-22 Glaxosmithkline Intellectual Property Development Limited Nrf2 regulators
WO2018109648A1 (en) 2016-12-14 2018-06-21 Glaxosmithkline Intellectual Property Development Limited 3-oxo-1,4-diazepinyle compounds as nrf2 activators
WO2018109647A1 (en) 2016-12-14 2018-06-21 Glaxosmithkline Intellectual Property Development Limited Bisaryl amides as nrf2 regulators
WO2018109643A1 (en) 2016-12-14 2018-06-21 Glaxosmithkline Intellectual Property Development Limited Bisaryl heterocycles as nrf2 acti
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