KR20150123838A - 안정한 글루코키나제 활성화제 조성물 - Google Patents
안정한 글루코키나제 활성화제 조성물 Download PDFInfo
- Publication number
- KR20150123838A KR20150123838A KR1020157025036A KR20157025036A KR20150123838A KR 20150123838 A KR20150123838 A KR 20150123838A KR 1020157025036 A KR1020157025036 A KR 1020157025036A KR 20157025036 A KR20157025036 A KR 20157025036A KR 20150123838 A KR20150123838 A KR 20150123838A
- Authority
- KR
- South Korea
- Prior art keywords
- cyclohexyl
- ureido
- thiazol
- ylsulfanyl
- trans
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
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| NZ603614A (en) | 2010-05-26 | 2014-10-31 | Transtech Pharma Llc | Use of metformin in combination with a glucokinase activator and compositions comprising metformin and a glucokinase activator |
| CN118453592A (zh) | 2012-05-17 | 2024-08-09 | Vtv治疗有限责任公司 | 用于治疗糖尿病的葡萄糖激酶活化剂组合物 |
| CN109646404B (zh) * | 2016-12-15 | 2022-10-04 | 华领医药技术（上海）有限公司 | 葡萄糖激酶激活剂的口服制剂及其制备方法 |
| AU2019287437A1 (en) | 2018-06-12 | 2020-09-10 | Vtv Therapeutics Llc | Therapeutic uses of glucokinase activators in combination with insulin or insulin analogs |
| WO2021167840A1 (en) | 2020-02-18 | 2021-08-26 | Vtv Therapeutics Llc | Sulfoxide and sulfone glucokinase activators and methods of use thereof |
| AU2020451588A1 (en) * | 2020-06-04 | 2023-01-19 | Hua Medicine (Shanghai) Ltd. | Glucokinase activator for treating diabetes with renal impairment |
| US11857536B2 (en) | 2020-06-04 | 2024-01-02 | Hua Medicine (Shanghai) Ltd. | Glucokinase activator for treating diabetes with renal impairment |
| CN116194442A (zh) * | 2020-06-08 | 2023-05-30 | 维特卫治疗有限责任公司 | {2-[3-环己基-3-(反式-4-丙氧基-环己基)-脲基]-噻唑-5-基硫烷基}-乙酸的盐或共晶体及其用途 |
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| PT1723128E (pt) * | 2004-01-06 | 2013-02-27 | Novo Nordisk As | Heteroaril-ureias e o seu uso como activadores da glicoquinase |
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| JP2009500356A (ja) * | 2005-07-07 | 2009-01-08 | エラン ファーマ インターナショナル リミテッド | ナノ粒子クラリスロマイシン製剤 |
| US8367112B2 (en) * | 2006-02-28 | 2013-02-05 | Alkermes Pharma Ireland Limited | Nanoparticulate carverdilol formulations |
| CN101495096A (zh) * | 2006-05-30 | 2009-07-29 | 伊兰制药国际有限公司 | 纳米微粒泊沙康唑制剂 |
| WO2008066899A2 (en) * | 2006-11-28 | 2008-06-05 | Marinus Pharmaceuticals | Nanoparticulate formulations and methods for the making and use thereof |
| JP5419706B2 (ja) * | 2006-12-20 | 2014-02-19 | タケダ カリフォルニア インコーポレイテッド | グルコキナーゼアクチベーター |
| US20090028680A1 (en) * | 2007-07-27 | 2009-01-29 | Kling Troy L | Intermediate apparatus for towing utility vehicles |
| EA018988B1 (ru) * | 2008-05-16 | 2013-12-30 | Такеда Калифорния, Инк. | Активаторы глюкокиназы |
| US8054567B2 (en) * | 2008-07-23 | 2011-11-08 | Hitachi High-Technologies Corporation | Method for measuring write/read width of a composite magnetic head and a measuring device using the method |
| SG176929A1 (en) * | 2009-06-18 | 2012-01-30 | Abbott Lab | Stable nanoparticulate drug suspension |
| JP5778667B2 (ja) * | 2009-06-19 | 2015-09-16 | ナノフォーム ハンガリー リミテッド | ナノ粒子のテルミサルタン組成物及びその調製方法 |
| CN101829061A (zh) * | 2010-05-14 | 2010-09-15 | 无锡纳生生物科技有限公司 | 一种紫杉醇纳米颗粒组合物及其制备方法 |
| NZ603614A (en) * | 2010-05-26 | 2014-10-31 | Transtech Pharma Llc | Use of metformin in combination with a glucokinase activator and compositions comprising metformin and a glucokinase activator |
-
2014
- 2014-02-28 WO PCT/US2014/019349 patent/WO2014137797A2/en not_active Ceased
- 2014-02-28 JP JP2015561468A patent/JP6441828B2/ja not_active Expired - Fee Related
- 2014-02-28 HK HK16101756.4A patent/HK1213780A1/zh unknown
- 2014-02-28 AU AU2014226290A patent/AU2014226290B2/en not_active Expired - Fee Related
- 2014-02-28 CN CN201480011647.2A patent/CN105050585A/zh active Pending
- 2014-02-28 CA CA2903433A patent/CA2903433A1/en not_active Abandoned
- 2014-02-28 MX MX2015011109A patent/MX2015011109A/es unknown
- 2014-02-28 EP EP14714823.3A patent/EP2964198A2/en not_active Withdrawn
- 2014-02-28 KR KR1020157025036A patent/KR20150123838A/ko not_active Withdrawn
-
2015
- 2015-08-20 IL IL240735A patent/IL240735A0/en unknown
- 2015-08-31 US US14/840,682 patent/US20160015638A1/en not_active Abandoned
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2024123015A1 (ko) * | 2022-12-06 | 2024-06-13 | 유노비아 주식회사 | 안정성이 향상된 gpr40 효현제를 유효성분으로 포함하는 약제학적 조성물 |
Also Published As
| Publication number | Publication date |
|---|---|
| EP2964198A2 (en) | 2016-01-13 |
| WO2014137797A2 (en) | 2014-09-12 |
| CN105050585A (zh) | 2015-11-11 |
| WO2014137797A3 (en) | 2014-10-30 |
| CA2903433A1 (en) | 2014-09-12 |
| HK1213780A1 (zh) | 2016-07-15 |
| JP6441828B2 (ja) | 2018-12-19 |
| AU2014226290A1 (en) | 2015-10-08 |
| MX2015011109A (es) | 2015-11-16 |
| AU2014226290B2 (en) | 2018-11-15 |
| US20160015638A1 (en) | 2016-01-21 |
| IL240735A0 (en) | 2015-10-29 |
| JP2016513625A (ja) | 2016-05-16 |
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