KR20140023354A - 면역 장애의 치료를 위한 치환된 인돌 유도체 - Google Patents
면역 장애의 치료를 위한 치환된 인돌 유도체 Download PDFInfo
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- KR20140023354A KR20140023354A KR20137030038A KR20137030038A KR20140023354A KR 20140023354 A KR20140023354 A KR 20140023354A KR 20137030038 A KR20137030038 A KR 20137030038A KR 20137030038 A KR20137030038 A KR 20137030038A KR 20140023354 A KR20140023354 A KR 20140023354A
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| US4925860A (en) | 1987-08-05 | 1990-05-15 | E. I. Du Pont De Nemours And Company | Stable pharmaceutical composition of 3-(hydroxymethyl)-5,5-diphenylhydantoin disodium phosphate ester |
| DE4005970A1 (de) | 1990-02-26 | 1991-08-29 | Boehringer Mannheim Gmbh | Neue trisubstituierte maleinimide, verfahren zu ihrer herstellung sowie arzneimittel, die diese verbindungen enthalten |
| GB9721069D0 (en) | 1997-10-03 | 1997-12-03 | Pharmacia & Upjohn Spa | Polymeric derivatives of camptothecin |
| US6204257B1 (en) | 1998-08-07 | 2001-03-20 | Universtiy Of Kansas | Water soluble prodrugs of hindered alcohols |
| CA2385071A1 (en) | 1999-10-12 | 2001-04-19 | Norman Kong | Substituted pyrroles as antiproliferative agents for the treatment of cancer |
| EP2070921A1 (en) | 2000-11-07 | 2009-06-17 | Novartis Ag | Indolylmaleimide derivatives as protein kinase c inhibitors |
| JP4369237B2 (ja) | 2001-12-21 | 2009-11-18 | エーザイ コーポレーション オブ ノース アメリカ | アルコールおよびフェノールの水溶性ホスホノオキシメチル誘導体の調製法 |
| NZ533536A (en) | 2001-12-28 | 2006-11-30 | Mgi Gp Inc | Aqueous based pharmaceutical formulations of water-soluble prodrugs of propofol such as O-phosphonooxymethyl propofol |
| TW200918046A (en) | 2002-04-03 | 2009-05-01 | Novartis Ag | Indolylmaleimide derivatives |
| HUP0600241A2 (en) | 2002-04-08 | 2006-07-28 | Mgi Gp | Pharmaceutical compositions containing water-soluble prodrugs of propofol and methods of administering same |
| JP2007524596A (ja) | 2003-02-28 | 2007-08-30 | トランスフォーム・ファーマシューティカルズ・インコーポレイテッド | 共結晶医薬組成物 |
| AU2003223104A1 (en) | 2003-03-19 | 2004-10-11 | Suven Life Sciences Limited | A process for the preparation of indolymaleimides |
| AU2006206458B2 (en) | 2005-01-19 | 2012-10-25 | Rigel Pharmaceuticals, Inc. | Prodrugs of 2,4-pyrimidinediamine compounds and their uses |
| WO2007008514A2 (en) | 2005-07-07 | 2007-01-18 | Georgetown University | Inhibitors of glycogen synthase kinase 3 |
| US20070203236A1 (en) | 2006-01-11 | 2007-08-30 | Smith Jeffrey W | Novel antagonists of the human fatty acid synthase thioesterase |
| GB0605691D0 (en) | 2006-03-21 | 2006-05-03 | Novartis Ag | Organic Compounds |
| ATE540041T1 (de) | 2006-11-21 | 2012-01-15 | Rigel Pharmaceuticals Inc | Prodrug-salze von 2,4-pyrimidindiaminverbindungen und anwendungen davon |
| WO2011057204A2 (en) | 2009-11-06 | 2011-05-12 | The Johns Hopkins University | Lrrk2-mediated neuronal toxicity |
| CN101812097B (zh) | 2010-04-17 | 2012-04-25 | 中国海洋大学 | 吲哚咔唑和双吲哚马来酰亚胺生物碱及其制备方法和应用 |
| UY34072A (es) | 2011-05-17 | 2013-01-03 | Novartis Ag | Derivados sustituidos de indol |
-
2012
- 2012-05-14 UY UY34072A patent/UY34072A/es not_active Application Discontinuation
- 2012-05-15 US US13/471,512 patent/US8703782B2/en active Active
- 2012-05-16 MX MX2013013436A patent/MX2013013436A/es not_active Application Discontinuation
- 2012-05-16 TW TW101117465A patent/TW201249858A/zh unknown
- 2012-05-16 JP JP2014510933A patent/JP6043344B2/ja active Active
- 2012-05-16 EA EA201391710A patent/EA023238B1/ru not_active IP Right Cessation
- 2012-05-16 KR KR20137030038A patent/KR20140023354A/ko not_active Withdrawn
- 2012-05-16 CA CA2835169A patent/CA2835169C/en active Active
- 2012-05-16 CN CN201280023473.2A patent/CN103534250B/zh active Active
- 2012-05-16 ES ES12726226.9T patent/ES2565200T3/es active Active
- 2012-05-16 WO PCT/IB2012/052473 patent/WO2012156936A1/en not_active Ceased
- 2012-05-16 AU AU2012257345A patent/AU2012257345B2/en active Active
- 2012-05-16 EP EP12726226.9A patent/EP2709998B1/en active Active
- 2012-05-16 BR BR112013029416A patent/BR112013029416A2/pt not_active IP Right Cessation
- 2012-05-18 AR ARP120101769 patent/AR088414A1/es not_active Application Discontinuation
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2014
- 2014-03-03 US US14/194,879 patent/US9029396B2/en active Active
Also Published As
| Publication number | Publication date |
|---|---|
| WO2012156936A1 (en) | 2012-11-22 |
| TW201249858A (en) | 2012-12-16 |
| AR088414A1 (es) | 2014-06-11 |
| EA201391710A1 (ru) | 2014-03-31 |
| JP6043344B2 (ja) | 2016-12-14 |
| CN103534250A (zh) | 2014-01-22 |
| EP2709998B1 (en) | 2016-01-06 |
| CN103534250B (zh) | 2016-05-11 |
| MX2013013436A (es) | 2013-12-06 |
| EP2709998A1 (en) | 2014-03-26 |
| ES2565200T3 (es) | 2016-04-01 |
| UY34072A (es) | 2013-01-03 |
| JP2014518870A (ja) | 2014-08-07 |
| CA2835169C (en) | 2019-05-14 |
| US9029396B2 (en) | 2015-05-12 |
| AU2012257345B2 (en) | 2016-03-24 |
| BR112013029416A2 (pt) | 2017-01-31 |
| US20140179634A1 (en) | 2014-06-26 |
| US8703782B2 (en) | 2014-04-22 |
| EA023238B1 (ru) | 2016-05-31 |
| CA2835169A1 (en) | 2012-11-22 |
| US20130157980A1 (en) | 2013-06-20 |
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