KR20120104523A - 디펩티딜 펩티다제―４ 억제제와 피오글리타존의 조합물의 제약 조성물 - Google Patents
디펩티딜 펩티다제―４ 억제제와 피오글리타존의 조합물의 제약 조성물 Download PDFInfo
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Classifications
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- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
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- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
- A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
Landscapes
- Health & Medical Sciences (AREA)
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- Public Health (AREA)
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- Pharmacology & Pharmacy (AREA)
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- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Endocrinology (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Emergency Medicine (AREA)
- Inorganic Chemistry (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
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| US25429909P | 2009-10-23 | 2009-10-23 | |
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| KR20120104523A true KR20120104523A (ko) | 2012-09-21 |
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| EP (1) | EP2490534A4 (enExample) |
| JP (1) | JP2013508370A (enExample) |
| KR (1) | KR20120104523A (enExample) |
| CN (1) | CN102573476A (enExample) |
| AU (1) | AU2010308433A1 (enExample) |
| BR (1) | BR112012009496A2 (enExample) |
| CA (1) | CA2777231A1 (enExample) |
| IN (1) | IN2012DN03271A (enExample) |
| MX (1) | MX2012004673A (enExample) |
| RU (1) | RU2012121185A (enExample) |
| WO (1) | WO2011049773A1 (enExample) |
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| AR086675A1 (es) * | 2011-06-14 | 2014-01-15 | Merck Sharp & Dohme | Composiciones farmaceuticas de combinaciones de inhibidores de la dipeptidil peptidasa-4 con simvastatina |
| US20140248345A1 (en) * | 2011-10-24 | 2014-09-04 | Merck Sharp & Dohme Corp. | Pharmaceutical compositions of combinations of dipeptidyl peptidase-4 inhibitors with atorvastatin |
| UA114948C2 (uk) * | 2013-03-06 | 2017-08-28 | Новартіс Аг | Склади з органічними сполуками |
| US9937153B2 (en) * | 2013-08-30 | 2018-04-10 | Merck Sharp & Dohme Ltd. | Oral pharmaceutical formulation of omarigliptin |
| TR201402685A1 (tr) * | 2014-03-06 | 2015-09-21 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Vildagliptinin farmasotik formulasyonları. |
| CN105030724A (zh) * | 2015-08-20 | 2015-11-11 | 杭州成邦医药科技有限公司 | 一种抗糖尿病药物的组合物 |
| CN108096227A (zh) * | 2018-01-25 | 2018-06-01 | 河北科技大学 | 阿格列汀口腔溶膜制剂 |
| JP7109748B2 (ja) * | 2018-12-11 | 2022-08-01 | 日本ジェネリック株式会社 | アジルサルタンとアムロジピンベシル酸塩含有固形製剤及び固形製剤の製造方法 |
| JP7423264B2 (ja) * | 2019-10-17 | 2024-01-29 | 日本ジェネリック株式会社 | シタグリプチン含有錠剤 |
| WO2022074664A1 (en) * | 2020-10-05 | 2022-04-14 | V-Ensure Pharma Technologies Private Limited | An immediate release composition of sitagliptin hydrochloride |
| TR202022612A2 (tr) * | 2020-12-31 | 2022-07-21 | Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi | Alogli̇pti̇ni̇n farmasöti̇k kapsül kompozi̇syonlari |
| CN115227661B (zh) * | 2022-09-22 | 2022-12-13 | 北京惠之衡生物科技有限公司 | 一种利格列汀片及其制备方法 |
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| GB0014969D0 (en) * | 2000-06-19 | 2000-08-09 | Smithkline Beecham Plc | Novel method of treatment |
| EP1807066A1 (en) * | 2004-10-25 | 2007-07-18 | Novartis AG | Combination of dpp-iv inhibitor, ppar antidiabetic and metformin |
| CN101208085B (zh) * | 2005-06-10 | 2011-01-05 | 诺瓦提斯公司 | 1-[(3-羟基-金刚烷基-1-基氨基)-乙酰基]-吡咯烷基-2(s)-腈的调释制剂 |
| MY152185A (en) * | 2005-06-10 | 2014-08-29 | Novartis Ag | Modified release 1-[(3-hydroxy-adamant-1-ylamino)-acetyl]-pyrrolidine-2(s)-carbonitrile formulation |
| JOP20180109A1 (ar) * | 2005-09-29 | 2019-01-30 | Novartis Ag | تركيبة جديدة |
| PE20140960A1 (es) * | 2008-04-03 | 2014-08-15 | Boehringer Ingelheim Int | Formulaciones que comprenden un inhibidor de dpp4 |
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2010
- 2010-10-12 IN IN3271DEN2012 patent/IN2012DN03271A/en unknown
- 2010-10-12 BR BR112012009496A patent/BR112012009496A2/pt not_active IP Right Cessation
- 2010-10-12 WO PCT/US2010/052225 patent/WO2011049773A1/en not_active Ceased
- 2010-10-12 RU RU2012121185/13A patent/RU2012121185A/ru not_active Application Discontinuation
- 2010-10-12 EP EP10825413.7A patent/EP2490534A4/en not_active Withdrawn
- 2010-10-12 KR KR1020127010201A patent/KR20120104523A/ko not_active Withdrawn
- 2010-10-12 US US13/501,252 patent/US20120201885A1/en not_active Abandoned
- 2010-10-12 AU AU2010308433A patent/AU2010308433A1/en not_active Abandoned
- 2010-10-12 MX MX2012004673A patent/MX2012004673A/es unknown
- 2010-10-12 CA CA2777231A patent/CA2777231A1/en not_active Abandoned
- 2010-10-12 CN CN2010800477129A patent/CN102573476A/zh active Pending
- 2010-10-12 JP JP2012535230A patent/JP2013508370A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| WO2011049773A1 (en) | 2011-04-28 |
| AU2010308433A1 (en) | 2012-06-07 |
| IN2012DN03271A (enExample) | 2015-10-23 |
| BR112012009496A2 (pt) | 2015-09-29 |
| CA2777231A1 (en) | 2011-04-28 |
| US20120201885A1 (en) | 2012-08-09 |
| RU2012121185A (ru) | 2013-11-27 |
| EP2490534A4 (en) | 2013-06-12 |
| CN102573476A (zh) | 2012-07-11 |
| MX2012004673A (es) | 2012-06-14 |
| JP2013508370A (ja) | 2013-03-07 |
| EP2490534A1 (en) | 2012-08-29 |
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