KR20070100331A - 새로운 아데노신 에이3 수용체 조절제 - Google Patents

새로운 아데노신 에이3 수용체 조절제 Download PDF

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Publication number
KR20070100331A
KR20070100331A KR1020077017126A KR20077017126A KR20070100331A KR 20070100331 A KR20070100331 A KR 20070100331A KR 1020077017126 A KR1020077017126 A KR 1020077017126A KR 20077017126 A KR20077017126 A KR 20077017126A KR 20070100331 A KR20070100331 A KR 20070100331A
Authority
KR
South Korea
Prior art keywords
dione
compound
purine
substituted
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
KR1020077017126A
Other languages
English (en)
Korean (ko)
Inventor
피어 바랄디
피어 안드레아 보레아
델리아 프레티
모즈간 아가자데 타브리지
Original Assignee
킹 파머슈티칼스 리서치 앤드 디벨로프먼트 아이엔씨
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 킹 파머슈티칼스 리서치 앤드 디벨로프먼트 아이엔씨 filed Critical 킹 파머슈티칼스 리서치 앤드 디벨로프먼트 아이엔씨
Publication of KR20070100331A publication Critical patent/KR20070100331A/ko
Ceased legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/14Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Biomedical Technology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1020077017126A 2005-02-02 2006-02-01 새로운 아데노신 에이3 수용체 조절제 Ceased KR20070100331A (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US64972605P 2005-02-02 2005-02-02
US60/649,726 2005-02-02
US11/344,295 2006-01-31
US11/344,295 US7435740B2 (en) 2005-02-02 2006-01-31 Adenosine A3 receptor modulators

Publications (1)

Publication Number Publication Date
KR20070100331A true KR20070100331A (ko) 2007-10-10

Family

ID=36777854

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020077017126A Ceased KR20070100331A (ko) 2005-02-02 2006-02-01 새로운 아데노신 에이3 수용체 조절제

Country Status (11)

Country Link
US (1) US7435740B2 (enExample)
EP (1) EP1845993A4 (enExample)
JP (1) JP2008538099A (enExample)
KR (1) KR20070100331A (enExample)
AU (1) AU2006210817B2 (enExample)
BR (1) BRPI0606750A2 (enExample)
CA (1) CA2596612A1 (enExample)
IL (1) IL184532A0 (enExample)
MX (1) MX2007008501A (enExample)
NZ (1) NZ556649A (enExample)
WO (1) WO2006083916A2 (enExample)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20090088403A1 (en) * 2007-05-07 2009-04-02 Randy Blakely A3 adenosine receptors as targets for the modulation of central serotonergic signaling
WO2009092602A2 (en) * 2008-01-24 2009-07-30 Universität Zürich Anti-angiogenic compounds
US20110190324A1 (en) * 2008-07-16 2011-08-04 Edward Leung Methods of treating atherosclerosis
EP2456419B1 (en) 2009-07-21 2016-11-23 Oradin Pharmaceutical Ltd. A3 adenosine receptor ligands for modulation of pigmentation

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6586429B2 (en) * 2000-11-29 2003-07-01 Cell Therapeutics, Inc. Tricyclic fused xanthine compounds and their uses

Also Published As

Publication number Publication date
US7435740B2 (en) 2008-10-14
NZ556649A (en) 2010-03-26
AU2006210817A2 (en) 2006-08-10
IL184532A0 (en) 2007-10-31
WO2006083916A2 (en) 2006-08-10
AU2006210817A1 (en) 2006-08-10
AU2006210817B2 (en) 2010-12-23
JP2008538099A (ja) 2008-10-09
WO2006083916A3 (en) 2007-12-21
EP1845993A4 (en) 2009-03-11
BRPI0606750A2 (pt) 2009-07-14
CA2596612A1 (en) 2006-08-10
US20060178385A1 (en) 2006-08-10
EP1845993A2 (en) 2007-10-24
MX2007008501A (es) 2007-09-14

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Patent event date: 20070725

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Patent event code: PE06011S01I