KR20050100396A - 6-치환 이미다조피라진 - Google Patents

6-치환 이미다조피라진 Download PDF

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Publication number
KR20050100396A
KR20050100396A KR1020057014835A KR20057014835A KR20050100396A KR 20050100396 A KR20050100396 A KR 20050100396A KR 1020057014835 A KR1020057014835 A KR 1020057014835A KR 20057014835 A KR20057014835 A KR 20057014835A KR 20050100396 A KR20050100396 A KR 20050100396A
Authority
KR
South Korea
Prior art keywords
alkyl
alkoxy
hydrogen
hydroxy
compound
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Withdrawn
Application number
KR1020057014835A
Other languages
English (en)
Korean (ko)
Inventor
엠 비토리아 키사
안드레아스 팔머
크리스토프 브레엠
게르하르트 그룬틀러
외르크 젠-빌핑어
볼프강-알렉산더 시몬
슈테판 포스티우스
볼프강 크로메르
페터 얀 침머만
빌름 부어
Original Assignee
알타나 파마 아게
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by 알타나 파마 아게 filed Critical 알타나 파마 아게
Publication of KR20050100396A publication Critical patent/KR20050100396A/ko
Withdrawn legal-status Critical Current

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nutrition Science (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
KR1020057014835A 2003-02-18 2004-02-16 6-치환 이미다조피라진 Withdrawn KR20050100396A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP03003652.9 2003-02-18
EP03003652 2003-02-18

Publications (1)

Publication Number Publication Date
KR20050100396A true KR20050100396A (ko) 2005-10-18

Family

ID=32892854

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020057014835A Withdrawn KR20050100396A (ko) 2003-02-18 2004-02-16 6-치환 이미다조피라진

Country Status (19)

Country Link
US (1) US20060148796A1 (enExample)
EP (1) EP1599481A1 (enExample)
JP (1) JP2006517951A (enExample)
KR (1) KR20050100396A (enExample)
CN (1) CN1747956A (enExample)
AR (1) AR043002A1 (enExample)
AU (1) AU2004213177A1 (enExample)
BR (1) BRPI0407390A (enExample)
CA (1) CA2516021A1 (enExample)
EA (1) EA200501229A1 (enExample)
HR (1) HRP20050794A2 (enExample)
IS (1) IS8015A (enExample)
MX (1) MXPA05008582A (enExample)
NO (1) NO20054199L (enExample)
PL (1) PL376466A1 (enExample)
RS (1) RS20050619A (enExample)
TW (1) TW200504068A (enExample)
WO (1) WO2004074289A1 (enExample)
ZA (1) ZA200505670B (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2007028051A2 (en) 2005-09-02 2007-03-08 Abbott Laboratories Novel imidazo based heterocycles
CA2654202A1 (en) * 2006-06-06 2007-12-21 Schering Corporation Imidazopyrazines as protein kinase inhibitors
US20090175852A1 (en) 2006-06-06 2009-07-09 Schering Corporation Imidazopyrazines as protein kinase inhibitors
WO2008059373A1 (en) * 2006-11-17 2008-05-22 Raqualia Pharma Inc. Imidazo [1, 2-a] pyrazine derivatives and their use as acid pump antagonists
GB0716292D0 (en) 2007-08-21 2007-09-26 Biofocus Dpi Ltd Imidazopyrazine compounds
KR101743784B1 (ko) 2008-12-08 2017-06-05 질레드 코네티컷 인코포레이티드 이미다조피라진 syk 억제제
KR101745732B1 (ko) * 2008-12-08 2017-06-12 질레드 코네티컷 인코포레이티드 이미다조피라진 syk 억제제
ES2530449T3 (es) 2010-03-11 2015-03-02 Gilead Connecticut Inc Inhibidores de Syk de imidazopiridinas
CN116178295A (zh) * 2023-01-28 2023-05-30 山东亿盛实业股份有限公司 一种苯唑草酮代谢物t283的制备方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4725601A (en) * 1985-06-04 1988-02-16 Fujisawa Pharmaceutical Co., Ltd. Certain imidazo[1,2-a]pyridines useful in the treatment of ulcers
JPH07242666A (ja) * 1994-03-08 1995-09-19 Fujisawa Pharmaceut Co Ltd 複素環化合物
SE9704404D0 (sv) * 1997-11-28 1997-11-28 Astra Ab New compounds
SE9801526D0 (sv) * 1998-04-29 1998-04-29 Astra Ab New compounds
EP1363702A4 (en) * 2001-01-30 2007-08-22 Cytopia Pty Ltd PROCESS FOR INHIBITING KINASES

Also Published As

Publication number Publication date
BRPI0407390A (pt) 2006-02-07
CN1747956A (zh) 2006-03-15
TW200504068A (en) 2005-02-01
AR043002A1 (es) 2005-07-13
ZA200505670B (en) 2006-04-26
RS20050619A (sr) 2007-09-21
US20060148796A1 (en) 2006-07-06
NO20054199L (no) 2005-11-17
WO2004074289A1 (en) 2004-09-02
JP2006517951A (ja) 2006-08-03
AU2004213177A1 (en) 2004-09-02
MXPA05008582A (es) 2005-11-04
NO20054199D0 (no) 2005-09-09
CA2516021A1 (en) 2004-09-02
EA200501229A1 (ru) 2006-04-28
IS8015A (is) 2005-09-08
EP1599481A1 (en) 2005-11-30
PL376466A1 (en) 2005-12-27
HRP20050794A2 (hr) 2006-12-31

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Legal Events

Date Code Title Description
PA0105 International application

Patent event date: 20050811

Patent event code: PA01051R01D

Comment text: International Patent Application

PG1501 Laying open of application
PC1203 Withdrawal of no request for examination
WITN Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid