KR20010111580A - 개선된 용해도를 갖는 탁산 제형물 - Google Patents
개선된 용해도를 갖는 탁산 제형물 Download PDFInfo
- Publication number
- KR20010111580A KR20010111580A KR1020017012367A KR20017012367A KR20010111580A KR 20010111580 A KR20010111580 A KR 20010111580A KR 1020017012367 A KR1020017012367 A KR 1020017012367A KR 20017012367 A KR20017012367 A KR 20017012367A KR 20010111580 A KR20010111580 A KR 20010111580A
- Authority
- KR
- South Korea
- Prior art keywords
- pyridyl
- thienyl
- substituted
- furyl
- phenyl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
- C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Applications Claiming Priority (17)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US17968400P | 2000-02-02 | 2000-02-02 | |
| US17967000P | 2000-02-02 | 2000-02-02 | |
| US17966900P | 2000-02-02 | 2000-02-02 | |
| US17967200P | 2000-02-02 | 2000-02-02 | |
| US17967100P | 2000-02-02 | 2000-02-02 | |
| US17978200P | 2000-02-02 | 2000-02-02 | |
| US17979300P | 2000-02-02 | 2000-02-02 | |
| US17967400P | 2000-02-02 | 2000-02-02 | |
| US60/179,782 | 2000-02-02 | ||
| US60/179,684 | 2000-02-02 | ||
| US60/179,672 | 2000-02-02 | ||
| US60/179,671 | 2000-02-02 | ||
| US60/179,793 | 2000-02-02 | ||
| US60/179,674 | 2000-02-02 | ||
| US60/179,669 | 2000-02-02 | ||
| US60/179,670 | 2000-02-02 | ||
| PCT/US2001/003624 WO2001057013A1 (en) | 2000-02-02 | 2001-02-02 | Taxane formulations having improved solubility |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| KR20010111580A true KR20010111580A (ko) | 2001-12-19 |
Family
ID=27575082
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| KR1020017012367A KR20010111580A (ko) | 2000-02-02 | 2001-02-02 | 개선된 용해도를 갖는 탁산 제형물 |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP1175414A1 (hu) |
| KR (1) | KR20010111580A (hu) |
| AU (1) | AU3481001A (hu) |
| BR (1) | BR0104358A (hu) |
| HU (1) | HUP0200995A3 (hu) |
| IL (1) | IL145635A0 (hu) |
| NO (1) | NO20014752L (hu) |
| NZ (1) | NZ514073A (hu) |
| WO (1) | WO2001057013A1 (hu) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CO5280224A1 (es) | 2000-02-02 | 2003-05-30 | Univ Florida State Res Found | Taxanos sustituidos con ester en c7, utiles como agentes antitumorales y composiciones farmaceuticas que los contienen |
| AU782028B2 (en) | 2000-02-02 | 2005-06-30 | Florida State University Research Foundation, Inc. | C10 carbonate substituted taxanes as antitumor agents |
| JP2003521514A (ja) | 2000-02-02 | 2003-07-15 | フロリダ・ステイト・ユニバーシティ・リサーチ・ファウンデイション・インコーポレイテッド | 抗腫瘍剤としてのｃ１０ヘテロ置換アセテートタキサン |
| BR0104351A (pt) | 2000-02-02 | 2002-01-02 | Univ Florida State Res Found | Taxanos substituìdos com carbonato c7 como agentes antitumor |
| US6649632B2 (en) | 2000-02-02 | 2003-11-18 | Fsu Research Foundation, Inc. | C10 ester substituted taxanes |
| CA2368534A1 (en) | 2000-02-02 | 2001-08-09 | Florida State University Research Foundation, Inc. | C7 heterosubstituted acetate taxanes as antitumor agents |
| JP2003522173A (ja) | 2000-02-02 | 2003-07-22 | フロリダ・ステイト・ユニバーシティ・リサーチ・ファウンデイション・インコーポレイテッド | 抗腫瘍剤としてのｃ１０カルバモイルオキシ置換タキサン |
| CA2354486A1 (en) * | 2001-07-31 | 2003-01-31 | Florida State University Research Foundation, Inc. | C7 ester substituted taxanes |
| CA2354478A1 (en) * | 2001-07-31 | 2003-01-31 | Florida State University Research Foundation, Inc. | C10 carbonate substituted taxanes |
| CA2494074A1 (en) * | 2002-08-02 | 2004-02-12 | Immunogen, Inc. | Cytotoxic agents containing novel potent taxanes and their therapeutic use |
| US7390898B2 (en) | 2002-08-02 | 2008-06-24 | Immunogen Inc. | Cytotoxic agents containing novel potent taxanes and their therapeutic use |
| HN2005000054A (es) | 2004-02-13 | 2009-02-18 | Florida State University Foundation Inc | Taxanos sustituidos con esteres de ciclopentilo en c10 |
| TW200540164A (en) | 2004-03-05 | 2005-12-16 | Univ Florida State Res Found | C7 lactyloxy-substituted taxanes |
| US8242166B2 (en) | 2008-03-31 | 2012-08-14 | Florida State University Research Foundation, Inc. | C(10) ethyl ester and C(10) cyclopropyl ester substituted taxanes |
Family Cites Families (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5250683A (en) * | 1991-09-23 | 1993-10-05 | Florida State University | Certain substituted taxanes and pharmaceutical compositions containing them |
| US5243045A (en) * | 1991-09-23 | 1993-09-07 | Florida State University | Certain alkoxy substituted taxanes and pharmaceutical compositions containing them |
| IL107950A (en) * | 1992-12-15 | 2001-04-30 | Upjohn Co | b 7, b 8 - Matano - Taxols, their preparation and pharmaceutical preparations against malignant tumors containing them |
| CA2174350A1 (en) * | 1993-10-20 | 1995-04-27 | Richard B. Greenwald | 2'- and/or 7- substituted taxoids |
| US6100411A (en) * | 1994-10-28 | 2000-08-08 | The Research Foundation Of State University Of New York | Taxoid anti-tumor agents and pharmaceutical compositions thereof |
| JPH10508022A (ja) * | 1994-10-28 | 1998-08-04 | ザ リサーチ ファウンデーション オブ ステート ユニバーシティ オブ ニューヨーク | タキソイド誘導体、それらの製造、およびそれらの抗腫瘍薬としての使用 |
| US5801191A (en) * | 1995-06-01 | 1998-09-01 | Biophysica Foundation | Taxoids |
| AU710156B2 (en) * | 1996-07-15 | 1999-09-16 | Kabushiki Kaisha Yakult Honsha | Taxane derivatives and drugs containing the same |
| JPH1192468A (ja) * | 1997-09-17 | 1999-04-06 | Yakult Honsha Co Ltd | 新規なタキサン誘導体 |
| KR100551945B1 (ko) * | 1997-12-19 | 2006-02-20 | 가부시키가이샤 야쿠루트 혼샤 | 택산 유도체 |
| JP2003026673A (ja) * | 1999-03-05 | 2003-01-29 | Asahi Kasei Corp | 骨形成促進剤 |
-
2001
- 2001-02-02 KR KR1020017012367A patent/KR20010111580A/ko not_active Application Discontinuation
- 2001-02-02 IL IL14563501A patent/IL145635A0/xx unknown
- 2001-02-02 BR BR0104358-7A patent/BR0104358A/pt not_active IP Right Cessation
- 2001-02-02 NZ NZ514073A patent/NZ514073A/xx not_active Application Discontinuation
- 2001-02-02 AU AU34810/01A patent/AU3481001A/en not_active Abandoned
- 2001-02-02 EP EP01906972A patent/EP1175414A1/en not_active Withdrawn
- 2001-02-02 HU HU0200995A patent/HUP0200995A3/hu unknown
- 2001-02-02 WO PCT/US2001/003624 patent/WO2001057013A1/en not_active Application Discontinuation
- 2001-10-01 NO NO20014752A patent/NO20014752L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| AU3481001A (en) | 2001-08-14 |
| NO20014752D0 (no) | 2001-10-01 |
| NO20014752L (no) | 2001-11-27 |
| WO2001057013A1 (en) | 2001-08-09 |
| EP1175414A1 (en) | 2002-01-30 |
| BR0104358A (pt) | 2002-01-02 |
| HUP0200995A3 (en) | 2005-02-28 |
| NZ514073A (en) | 2004-02-27 |
| IL145635A0 (en) | 2002-06-30 |
| HUP0200995A2 (hu) | 2002-07-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| WITN | Application deemed withdrawn, e.g. because no request for examination was filed or no examination fee was paid |