KR20010101649A - 항균제로서 3,6-이치환된 페남 술폰 유도체 - Google Patents

항균제로서 3,6-이치환된 페남 술폰 유도체 Download PDF

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Publication number
KR20010101649A
KR20010101649A KR1020017009276A KR20017009276A KR20010101649A KR 20010101649 A KR20010101649 A KR 20010101649A KR 1020017009276 A KR1020017009276 A KR 1020017009276A KR 20017009276 A KR20017009276 A KR 20017009276A KR 20010101649 A KR20010101649 A KR 20010101649A
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KR
South Korea
Prior art keywords
formula
compound
methyl
hydrogen
pharmaceutically acceptable
Prior art date
Application number
KR1020017009276A
Other languages
English (en)
Korean (ko)
Inventor
린양-이
비타파나요타
리죵
프란시스코제라르도델라쿠르즈
Original Assignee
윌리암 에이취 캘넌, 에곤 이 버그
아메리칸사이아나미드컴파니
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by 윌리암 에이취 캘넌, 에곤 이 버그, 아메리칸사이아나미드컴파니 filed Critical 윌리암 에이취 캘넌, 에곤 이 버그
Publication of KR20010101649A publication Critical patent/KR20010101649A/ko

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Cephalosporin Compounds (AREA)
KR1020017009276A 1999-01-26 2000-01-26 항균제로서 3,6-이치환된 페남 술폰 유도체 KR20010101649A (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23772699A 1999-01-26 1999-01-26
US09/237,726 1999-01-26
PCT/US2000/001630 WO2000043399A1 (en) 1999-01-26 2000-01-26 3,6-disubstituted penam sulfone derivatives as antibacterials

Publications (1)

Publication Number Publication Date
KR20010101649A true KR20010101649A (ko) 2001-11-14

Family

ID=22894903

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1020017009276A KR20010101649A (ko) 1999-01-26 2000-01-26 항균제로서 3,6-이치환된 페남 술폰 유도체

Country Status (20)

Country Link
EP (1) EP1144418A1 (zh)
JP (1) JP2002535335A (zh)
KR (1) KR20010101649A (zh)
CN (1) CN1188417C (zh)
AU (1) AU2624600A (zh)
BG (1) BG105737A (zh)
BR (1) BR0007729A (zh)
CA (1) CA2355738A1 (zh)
CZ (1) CZ20012691A3 (zh)
EA (1) EA200100813A1 (zh)
HK (1) HK1038747A1 (zh)
HU (1) HUP0200013A3 (zh)
ID (1) ID29400A (zh)
IL (1) IL144116A0 (zh)
NO (1) NO20013640D0 (zh)
PL (1) PL349874A1 (zh)
SK (1) SK10142001A3 (zh)
TR (1) TR200102133T2 (zh)
WO (1) WO2000043399A1 (zh)
ZA (1) ZA200104323B (zh)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP2406267B1 (en) * 2009-03-10 2019-02-20 L'Air Liquide Société Anonyme pour l'Etude et l'Exploitation des Procédés Georges Claude Cyclic amino compounds for low-k silylation
CN109422765B (zh) * 2017-09-05 2020-08-28 香港理工大学深圳研究院 C类β-内酰胺酶抑制剂及其制备方法和应用

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2076812A (en) * 1980-05-22 1981-12-09 Ciba Geigy Ag Penam-dioxide compounds, processes for their manufacture, and their use
EP0083977A1 (en) * 1982-01-11 1983-07-20 Pfizer Inc. 6-Alpha-hydroxymethylpenicillanic acid sulfone as a beta-lactamase inhibitor
US4562073A (en) * 1982-12-24 1985-12-31 Taiho Pharmaceutical Company Limited Penicillin derivatives
US4503040A (en) * 1984-02-27 1985-03-05 Pfizer Inc. 6-(Aminoacyloxymethyl)penicillanic acid 1,1-dioxides as beta-lactamase inhibitors
US4591459A (en) * 1984-12-03 1986-05-27 Pfizer Inc. Intermediates for 6-(aminoacyloxymethyl) penicillanic acid 1,1-dioxides
TW383308B (en) * 1993-08-24 2000-03-01 Hoffmann La Roche 2-beta-alkenyl penam sulfones as beta-lactamase inhibitors

Also Published As

Publication number Publication date
HK1038747A1 (zh) 2002-03-28
BG105737A (en) 2002-05-31
CZ20012691A3 (cs) 2002-06-12
TR200102133T2 (tr) 2001-12-21
EA200100813A1 (ru) 2003-02-27
IL144116A0 (en) 2002-05-23
EP1144418A1 (en) 2001-10-17
AU2624600A (en) 2000-08-07
HUP0200013A2 (hu) 2002-05-29
BR0007729A (pt) 2001-10-30
NO20013640L (no) 2001-07-24
HUP0200013A3 (en) 2002-10-28
PL349874A1 (en) 2002-09-23
WO2000043399A1 (en) 2000-07-27
ID29400A (id) 2001-08-30
ZA200104323B (en) 2002-08-26
SK10142001A3 (sk) 2002-07-02
JP2002535335A (ja) 2002-10-22
CN1337965A (zh) 2002-02-27
NO20013640D0 (no) 2001-07-24
CN1188417C (zh) 2005-02-09
CA2355738A1 (en) 2000-07-27

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