KR102386952B1 - 항암 및 항-증식 활성을 나타내는 n-아실-n'-(피리딘-2-일) 우레아 및 유사체 - Google Patents

항암 및 항-증식 활성을 나타내는 n-아실-n'-(피리딘-2-일) 우레아 및 유사체 Download PDF

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KR102386952B1
KR102386952B1 KR1020217038874A KR20217038874A KR102386952B1 KR 102386952 B1 KR102386952 B1 KR 102386952B1 KR 1020217038874 A KR1020217038874 A KR 1020217038874A KR 20217038874 A KR20217038874 A KR 20217038874A KR 102386952 B1 KR102386952 B1 KR 102386952B1
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pyridin
methyl
oxy
carbamoyl
pyrazol
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KR20210149218A (ko
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마이클 디. 카우프만
티모시 말콤 콜드웰
다니엘 엘. 플린
윌리엄 씨. 패트
타이완카 사마라쿤
락슈미나라야나 보게티
카렌 엠. 예이츠
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데시페라 파마슈티칼스, 엘엘씨.
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    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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KR1020217038874A 2013-03-15 2014-03-14 항암 및 항-증식 활성을 나타내는 n-아실-n'-(피리딘-2-일) 우레아 및 유사체 Active KR102386952B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201361789971P 2013-03-15 2013-03-15
US61/789,971 2013-03-15
KR1020157029126A KR102333718B1 (ko) 2013-03-15 2014-03-14 항암 및 항-증식 활성을 나타내는 n-아실-n'-(피리딘-2-일) 우레아 및 유사체
PCT/US2014/029664 WO2014145028A2 (en) 2013-03-15 2014-03-14 N-acyl-n'-(pyridin-2-yl) ureas and analogs exhibiting anti-cancer and anti-proliferative activities

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KR1020157029126A Division KR102333718B1 (ko) 2013-03-15 2014-03-14 항암 및 항-증식 활성을 나타내는 n-아실-n'-(피리딘-2-일) 우레아 및 유사체

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KR20210149218A KR20210149218A (ko) 2021-12-08
KR102386952B1 true KR102386952B1 (ko) 2022-04-18

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KR1020157029126A Active KR102333718B1 (ko) 2013-03-15 2014-03-14 항암 및 항-증식 활성을 나타내는 n-아실-n'-(피리딘-2-일) 우레아 및 유사체

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US (1) US9382228B2 (https=)
EP (1) EP2968287B1 (https=)
JP (3) JP6364472B2 (https=)
KR (2) KR102386952B1 (https=)
CN (3) CN110563700A (https=)
AU (2) AU2014233414B2 (https=)
BR (1) BR112015022263B1 (https=)
CA (1) CA2903288C (https=)
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US8461179B1 (en) 2012-06-07 2013-06-11 Deciphera Pharmaceuticals, Llc Dihydronaphthyridines and related compounds useful as kinase inhibitors for the treatment of proliferative diseases
JP6364472B2 (ja) * 2013-03-15 2018-07-25 デシフェラ ファーマシューティカルズ，エルエルシー 抗がんおよび抗増殖活性を示すｎ−アシル−ｎ’−（ピリジン−２−イル）尿素および類似体
TWI747873B (zh) * 2016-02-01 2021-12-01 美商百歐克斯製藥公司 苯并吡唑化合物及其類似物
KR101691954B1 (ko) 2016-04-26 2017-01-02 고려대학교 산학협력단 신규 n-아실유레아 유도체 및 이를 함유하는 심혈관질환의 예방 또는 치료용 조성물
EP3632907B1 (en) * 2017-05-24 2024-02-28 Abbisko Therapeutics Co., Ltd. N-(azaaryl)cyclolactam-1-carboxamide derivative, preparation method therefor, and use thereof
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