KR101571400B1 - 자궁 섬유종의 치료를 위한 울리프리스탈 아세테이트의 용도 - Google Patents

자궁 섬유종의 치료를 위한 울리프리스탈 아세테이트의 용도 Download PDF

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Publication number
KR101571400B1
KR101571400B1 KR1020107019181A KR20107019181A KR101571400B1 KR 101571400 B1 KR101571400 B1 KR 101571400B1 KR 1020107019181 A KR1020107019181 A KR 1020107019181A KR 20107019181 A KR20107019181 A KR 20107019181A KR 101571400 B1 KR101571400 B1 KR 101571400B1
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South Korea
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medicament
uterine fibroids
acetate
patient
cdb
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KR1020107019181A
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English (en)
Korean (ko)
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KR20110021709A (ko
Inventor
에린 게이너
리네트 니먼
앙드레 울만
다이애너 블라이드
Original Assignee
라보라토이레 에이치알에이 파르마
더 유나이티드 스테이츠 오브 어메리카, 리프리젠티드 바이 더 세크러테리, 디파트먼트 오브 헬쓰 앤드 휴먼 서비씨즈
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40551565&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR101571400(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 라보라토이레 에이치알에이 파르마, 더 유나이티드 스테이츠 오브 어메리카, 리프리젠티드 바이 더 세크러테리, 디파트먼트 오브 헬쓰 앤드 휴먼 서비씨즈 filed Critical 라보라토이레 에이치알에이 파르마
Publication of KR20110021709A publication Critical patent/KR20110021709A/ko
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Publication of KR101571400B1 publication Critical patent/KR101571400B1/ko
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18—Feminine contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/36—Antigestagens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06—Antianaemics

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  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Endocrinology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Reproductive Health (AREA)
  • Oncology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Ultra Sonic Daignosis Equipment (AREA)
KR1020107019181A 2008-01-29 2009-01-28 자궁 섬유종의 치료를 위한 울리프리스탈 아세테이트의 용도 Expired - Fee Related KR101571400B1 (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US12/021,610 2008-01-29
US12/021,610 US8299050B2 (en) 2008-01-29 2008-01-29 Method for treating uterine fibroids

Related Child Applications (1)

Application Number Title Priority Date Filing Date
KR1020157011511A Division KR20150055626A (ko) 2008-01-29 2009-01-28 자궁 섬유종의 치료를 위한 울리프리스탈 아세테이트의 용도

Publications (2)

Publication Number Publication Date
KR20110021709A KR20110021709A (ko) 2011-03-04
KR101571400B1 true KR101571400B1 (ko) 2015-11-24

Family

ID=40551565

Family Applications (2)

Application Number Title Priority Date Filing Date
KR1020107019181A Expired - Fee Related KR101571400B1 (ko) 2008-01-29 2009-01-28 자궁 섬유종의 치료를 위한 울리프리스탈 아세테이트의 용도
KR1020157011511A Ceased KR20150055626A (ko) 2008-01-29 2009-01-28 자궁 섬유종의 치료를 위한 울리프리스탈 아세테이트의 용도

Family Applications After (1)

Application Number Title Priority Date Filing Date
KR1020157011511A Ceased KR20150055626A (ko) 2008-01-29 2009-01-28 자궁 섬유종의 치료를 위한 울리프리스탈 아세테이트의 용도

Country Status (20)

Country Link
US (5) US8299050B2 (https=)
EP (2) EP2252301B1 (https=)
JP (2) JP5906016B2 (https=)
KR (2) KR101571400B1 (https=)
AU (1) AU2009209652B2 (https=)
BR (1) BRPI0907028B8 (https=)
CA (2) CA2713254C (https=)
CY (1) CY1116485T1 (https=)
DK (1) DK2252301T3 (https=)
ES (1) ES2450592T3 (https=)
HR (1) HRP20140132T1 (https=)
IL (2) IL207182A (https=)
MX (1) MX2010008270A (https=)
NZ (1) NZ587439A (https=)
PL (1) PL2252301T3 (https=)
PT (1) PT2252301E (https=)
SI (1) SI2252301T1 (https=)
TW (1) TWI445537B (https=)
WO (1) WO2009095418A1 (https=)
ZA (1) ZA201006049B (https=)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8299050B2 (en) 2008-01-29 2012-10-30 Laboratoire Hra-Pharma Method for treating uterine fibroids
EP3865502A1 (en) * 2010-03-22 2021-08-18 Allergan Pharmaceuticals International Limited Compositions and methods for non-toxic delivery of cdb-2914
EP2471537A1 (en) * 2010-12-30 2012-07-04 PregLem S.A. Treatment of pain associated with dislocation of basal endometrium
EP2545922A1 (en) * 2011-07-12 2013-01-16 PregLem S.A. Treatment of excessive menstrual bleeding associated with uterine fibroids
EP2641602A1 (en) * 2012-03-23 2013-09-25 PregLem S.A. Method for treating gynecological diseases
WO2014050105A1 (en) * 2012-09-28 2014-04-03 Aska Pharmaceutical Co., Ltd. Amorphous ulipristal acetate
FR2997628B1 (fr) * 2012-11-08 2015-01-16 Hra Pharma Lab Produit de co-micronisation comprenant un modulateur selectif des recepteurs a la progesterone
FR2997627B1 (fr) * 2012-11-08 2015-01-16 Hra Pharma Lab Produit de co-micronisation comprenant de l'ulipristal acetate
HK1213487A1 (zh) * 2012-12-14 2016-07-08 The Population Council, Inc. 銅子宮環
CN103006595B (zh) * 2012-12-25 2018-04-06 江苏亚邦爱普森药业有限公司 制备醋酸优力司特片的方法
JP6255038B2 (ja) * 2013-02-26 2017-12-27 トリアクト セラピューティクス，インク． 癌治療
HK1221169A1 (zh) * 2013-04-10 2017-05-26 Preglem S.A. 孕酮受体调节剂在子宫肌瘤疗法中的用途
US10444958B2 (en) * 2013-09-23 2019-10-15 Adobe Systems Incorporated Visual example-based user interface for adjusting photos along two dimensions
US10238722B2 (en) 2014-11-24 2019-03-26 Ramot At Tel-Aviv University Ltd. Pigment epithelium derived factor (PEDF) for the treatment of uterine fibroids
WO2017216637A2 (en) 2017-08-04 2017-12-21 Alvogen Malta Operations (Row) Ltd Tablet form including ulipristal acetate and the methods for its preparation
KR102086827B1 (ko) * 2017-12-14 2020-03-10 경희대학교 산학협력단 자궁근육종 치료용 울리프리스탈 아세테이트
KR102043349B1 (ko) * 2018-01-10 2019-11-12 경희대학교 산학협력단 대장암 치료 용도의 울리프리스탈 아세테이트
AU2021225117A1 (en) 2020-02-19 2022-10-06 Vélfag ehf. Device and method for filleting and pin-bone removal

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US5468741A (en) * 1993-05-28 1995-11-21 The Regents Of The University Of California Use of low levels of mifepristone to treat leiomyomata
DE4426601A1 (de) * 1994-07-27 1996-02-01 Schering Ag Verwendung eines Kombinationsproduktes enthaltend einen kompetitiven Progesteronantagonisten und ein Gestagen zur Herstellung eines Arzneimittels zur Behandlung der Endometriose oder des Leiomyomata uteri
UA37259C2 (uk) * 1995-02-02 2001-05-15 Шерінг Актієнгезеллшафт Активна речовина для одержання лікарських засобів при лікуванні дисфункціональних маткових кровотеч
US5929262A (en) 1995-03-30 1999-07-27 The United States Of America As Represented By The Department Of Health And Human Services Method for preparing 17α-acetoxy-11β-(4-N, N-dimethylaminophyl)-19-Norpregna-4,9-diene-3, 20-dione, intermediates useful in the method, and methods for the preparation of such intermediates
WO1997041145A1 (en) 1996-05-01 1997-11-06 The Government Of The United States Of America, Represented By The Secretary, Department Of Health And Human Services 21-substituted progesterone derivatives as new antiprogestational agents
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US6262042B1 (en) * 1998-05-29 2001-07-17 Research Triangle Institute 17β-amino and hydroxylamino-11β-arylsteroids and their derivatives having agonist or antagonist hormonal properties
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SI2148681T1 (sl) 2007-04-20 2016-07-29 Preglem S.A. Selektivni modulatorji progesterona v zdravljenju maternične krvavitve
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UTERINE FIBROIDS, THE MERCK MANUAL 18TH EDITION*

Also Published As

Publication number Publication date
CA2857798A1 (en) 2009-09-06
US8299050B2 (en) 2012-10-30
IL207182A0 (en) 2010-12-30
EP2252301B1 (en) 2013-12-11
JP2015120711A (ja) 2015-07-02
WO2009095418A1 (en) 2009-08-06
US9682088B2 (en) 2017-06-20
JP6138838B2 (ja) 2017-05-31
US20170246189A1 (en) 2017-08-31
BRPI0907028B1 (pt) 2019-09-24
NZ587439A (en) 2012-06-29
EP2684565B1 (en) 2019-10-02
US20130023506A1 (en) 2013-01-24
MX2010008270A (es) 2011-01-14
IL207182A (en) 2015-06-30
ES2450592T3 (es) 2014-03-25
AU2009209652A1 (en) 2009-08-06
US9180133B2 (en) 2015-11-10
PL2252301T3 (pl) 2014-07-31
EP2252301A1 (en) 2010-11-24
IL234149A0 (en) 2014-09-30
JP2011510949A (ja) 2011-04-07
US20140187525A1 (en) 2014-07-03
US8722653B2 (en) 2014-05-13
AU2009209652B2 (en) 2013-03-21
US20090192130A1 (en) 2009-07-30
JP5906016B2 (ja) 2016-04-20
SI2252301T1 (sl) 2014-05-30
US20160022698A1 (en) 2016-01-28
DK2252301T3 (en) 2014-02-17
KR20110021709A (ko) 2011-03-04
CA2713254C (en) 2014-10-07
BRPI0907028A2 (pt) 2015-07-07
KR20150055626A (ko) 2015-05-21
PT2252301E (pt) 2014-02-24
EP2684565A1 (en) 2014-01-15
TW200944211A (en) 2009-11-01
ZA201006049B (en) 2011-05-25
TWI445537B (zh) 2014-07-21
BRPI0907028B8 (pt) 2021-05-25
CY1116485T1 (el) 2017-03-15
BRPI0907028A8 (pt) 2019-08-13
IL234149B (en) 2019-02-28
CA2713254A1 (en) 2009-09-06
HRP20140132T1 (hr) 2014-05-09

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