KR100982753B1 - 테트라사이클린 화합물 및 테트라사이클린 유도체의 전달조절 - Google Patents

테트라사이클린 화합물 및 테트라사이클린 유도체의 전달조절 Download PDF

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KR100982753B1
KR100982753B1 KR1020037012966A KR20037012966A KR100982753B1 KR 100982753 B1 KR100982753 B1 KR 100982753B1 KR 1020037012966 A KR1020037012966 A KR 1020037012966A KR 20037012966 A KR20037012966 A KR 20037012966A KR 100982753 B1 KR100982753 B1 KR 100982753B1
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tetracycline
release
tetracycline compound
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antibiotic
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KR20040002896A (ko
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로버트 에이. 애슐리
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콜라제넥스 파마슈티칼스, 인크
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/65—Tetracyclines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/166—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the carbon of a carboxamide group directly attached to the aromatic ring, e.g. procainamide, procarbazine, metoclopramide, labetalol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/06—Anabolic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurology (AREA)
  • Emergency Medicine (AREA)
  • Immunology (AREA)
  • Rheumatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
KR1020037012966A 2001-04-05 2002-04-05 테트라사이클린 화합물 및 테트라사이클린 유도체의 전달조절 Expired - Fee Related KR100982753B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US28185401P 2001-04-05 2001-04-05
US60/281,854 2001-04-05
PCT/US2002/010748 WO2002083106A1 (en) 2001-04-05 2002-04-05 Controlled delivery of tetracycline compounds and tetracycline derivatives

Publications (2)

Publication Number Publication Date
KR20040002896A KR20040002896A (ko) 2004-01-07
KR100982753B1 true KR100982753B1 (ko) 2010-09-16

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KR1020037012966A Expired - Fee Related KR100982753B1 (ko) 2001-04-05 2002-04-05 테트라사이클린 화합물 및 테트라사이클린 유도체의 전달조절

Country Status (8)

Country Link
US (2) US20040115261A1 (enExample)
EP (2) EP2311440A1 (enExample)
JP (3) JP2004525955A (enExample)
KR (1) KR100982753B1 (enExample)
AU (1) AU2002256092C1 (enExample)
CA (1) CA2447008A1 (enExample)
NZ (1) NZ529308A (enExample)
WO (1) WO2002083106A1 (enExample)

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JP2010047617A (ja) 2010-03-04
AU2002256092C1 (en) 2009-10-15
NZ529308A (en) 2005-03-24
AU2002256092B2 (en) 2007-05-31
EP1383483A4 (en) 2006-08-09
WO2002083106A1 (en) 2002-10-24
US20040115261A1 (en) 2004-06-17
JP2004525955A (ja) 2004-08-26
US20110262542A1 (en) 2011-10-27
EP1383483A1 (en) 2004-01-28
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EP2311440A1 (en) 2011-04-20
CA2447008A1 (en) 2002-10-24

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