KR100938136B1 - 안드로겐 수용체 조정자로서의 불화된 4-아자스테로이드 유도체 및 이를 포함하는 약제학적 조성물 - Google Patents

안드로겐 수용체 조정자로서의 불화된 4-아자스테로이드 유도체 및 이를 포함하는 약제학적 조성물 Download PDF

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KR100938136B1
KR100938136B1 KR1020047014281A KR20047014281A KR100938136B1 KR 100938136 B1 KR100938136 B1 KR 100938136B1 KR 1020047014281 A KR1020047014281 A KR 1020047014281A KR 20047014281 A KR20047014281 A KR 20047014281A KR 100938136 B1 KR100938136 B1 KR 100938136B1
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methyl
oxo
aza
fluoro
carboxamide
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KR20040097167A (ko
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메이스너로버트에스
퍼킨스제임스제이
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머크 앤드 캄파니 인코포레이티드
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom

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KR1020047014281A 2002-03-13 2003-03-07 안드로겐 수용체 조정자로서의 불화된 4-아자스테로이드 유도체 및 이를 포함하는 약제학적 조성물 Expired - Fee Related KR100938136B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US36382202P 2002-03-13 2002-03-13
US60/363,822 2002-03-13
PCT/US2003/008277 WO2003077919A1 (en) 2002-03-13 2003-03-07 Fluorinated 4-azasteroid derivatives as androgen receptor modulators

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KR20040097167A KR20040097167A (ko) 2004-11-17
KR100938136B1 true KR100938136B1 (ko) 2010-01-22

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US (1) US7186838B2 (enExample)
EP (1) EP1485095A4 (enExample)
JP (2) JP4516316B2 (enExample)
KR (1) KR100938136B1 (enExample)
CN (1) CN1652786A (enExample)
AU (1) AU2003218235B2 (enExample)
BR (1) BR0308355A (enExample)
CA (1) CA2478186C (enExample)
EC (1) ECSP045287A (enExample)
HR (1) HRP20040822A2 (enExample)
IL (2) IL163825A0 (enExample)
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MA (1) MA27112A1 (enExample)
MX (1) MXPA04008800A (enExample)
NO (1) NO20044312L (enExample)
NZ (1) NZ534946A (enExample)
PL (1) PL372920A1 (enExample)
RU (1) RU2320670C2 (enExample)
UA (1) UA78029C2 (enExample)
WO (1) WO2003077919A1 (enExample)
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