KR0169501B1 - 아닐리드 유도체 - Google Patents

아닐리드 유도체 Download PDF

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Publication number
KR0169501B1
KR0169501B1 KR1019930701531A KR930701531A KR0169501B1 KR 0169501 B1 KR0169501 B1 KR 0169501B1 KR 1019930701531 A KR1019930701531 A KR 1019930701531A KR 930701531 A KR930701531 A KR 930701531A KR 0169501 B1 KR0169501 B1 KR 0169501B1
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KR
South Korea
Prior art keywords
group
compound
carbon atoms
diisopropylphenyl
acetamide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
KR1019930701531A
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English (en)
Korean (ko)
Other versions
KR930702254A (ko
Inventor
마사카즈 사토
유타카 카와시마
카츠오 하타야마
Original Assignee
우에하라 아키라
다이쇼 세이야꾸 가부시끼가이샤
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Publication date
Application filed by 우에하라 아키라, 다이쇼 세이야꾸 가부시끼가이샤 filed Critical 우에하라 아키라
Publication of KR930702254A publication Critical patent/KR930702254A/ko
Application granted granted Critical
Publication of KR0169501B1 publication Critical patent/KR0169501B1/ko
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C327/00—Thiocarboxylic acids
    • C07C327/20—Esters of monothiocarboxylic acids
    • C07C327/32—Esters of monothiocarboxylic acids having sulfur atoms of esterified thiocarboxyl groups bound to carbon atoms of hydrocarbon radicals substituted by carboxyl groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Cosmetics (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
KR1019930701531A 1990-11-26 1991-11-21 아닐리드 유도체 Expired - Fee Related KR0169501B1 (ko)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP90-322136 1990-11-26
JP322136/1990 1990-11-26
JP32213690 1990-11-26
PCT/JP1991/001602 WO1992009572A1 (en) 1990-11-26 1991-11-21 Anilide derivative

Publications (2)

Publication Number Publication Date
KR930702254A KR930702254A (ko) 1993-09-08
KR0169501B1 true KR0169501B1 (ko) 1999-03-20

Family

ID=18140332

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019930701531A Expired - Fee Related KR0169501B1 (ko) 1990-11-26 1991-11-21 아닐리드 유도체

Country Status (11)

Country Link
US (1) US5475130A (enExample)
EP (1) EP0559898B1 (enExample)
JP (1) JP2650096B2 (enExample)
KR (1) KR0169501B1 (enExample)
AT (1) ATE137744T1 (enExample)
CA (1) CA2096970C (enExample)
DE (1) DE69119434T2 (enExample)
DK (1) DK0559898T3 (enExample)
ES (1) ES2088574T3 (enExample)
GR (1) GR3020257T3 (enExample)
WO (1) WO1992009572A1 (enExample)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5668136A (en) * 1990-09-25 1997-09-16 Eisai Co., Ltd. Trisubstituted benzene derivatives, composition and methods of treatment
WO1994002452A1 (fr) * 1992-07-20 1994-02-03 Eisai Co., Ltd. Derive du benzene
WO1995014463A1 (en) * 1993-11-25 1995-06-01 Taisho Pharmaceutical Co., Ltd. Composition of pharmaceutical preparation improved in peroral absorbability
FR2729665B1 (fr) * 1995-01-19 1997-04-18 Pf Medicament Nouveaux derives de glycylanilides, leur preparation et leur application en therapeutique
FR2741619B1 (fr) * 1995-11-28 1998-02-13 Pf Medicament Nouveaux derives de 2,3,5-trimethyl-4-hydroxy-anilides, leur preparation et leur application en therapeutique
CA2285374A1 (en) * 1997-04-01 1998-10-08 Taisho Pharmaceutical Co., Ltd. Preventives for reconstriction
KR20010005845A (ko) * 1997-04-01 2001-01-15 우에하라 아끼라 허혈성 심장 질환 예방제
WO2003020315A1 (fr) * 2001-08-28 2003-03-13 Sankyo Company, Limited Compositions medicinales contenant un antagoniste du recepteur d'angiotensine ii
US20050119314A1 (en) * 2002-04-05 2005-06-02 Sankyo Company, Limited Pharmaceutical composition comprising an ACAT inhibitor and an insulin resistance reducing agent
US7829552B2 (en) 2003-11-19 2010-11-09 Metabasis Therapeutics, Inc. Phosphorus-containing thyromimetics
MX2007005129A (es) * 2004-10-27 2007-09-11 Daiichi Sankyo Co Ltd Compuesto de benceno que tiene 2 o mas sustituyentes.
CA2657247A1 (en) * 2006-07-28 2008-01-31 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
WO2008039645A1 (en) * 2006-09-25 2008-04-03 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
CA2704684A1 (en) * 2007-11-07 2009-05-14 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
CA2730037A1 (en) * 2008-07-10 2010-01-14 Boehringer Ingelheim International Gmbh Sulfone compounds which modulate the cb2 receptor
KR20110063485A (ko) * 2008-09-25 2011-06-10 베링거 인겔하임 인터내셔날 게엠베하 Ｃｂ2 수용체를 선택적으로 조절하는 설포닐 화합물
US20120046364A1 (en) 2009-02-10 2012-02-23 Metabasis Therapeutics, Inc. Novel Sulfonic Acid-Containing Thyromimetics, and Methods for Their Use
US8299103B2 (en) 2009-06-15 2012-10-30 Boehringer Ingelheim International Gmbh Compounds which selectively modulate the CB2 receptor
JP5756800B2 (ja) 2009-06-16 2015-07-29 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｂ２受容体を調節するアゼチジン２−カルボキサミド誘導体
WO2011037795A1 (en) * 2009-09-22 2011-03-31 Boehringer Ingelheim International Gmbh Compounds which selectively modulate the cb2 receptor
WO2011088015A1 (en) 2010-01-15 2011-07-21 Boehringer Ingelheim International Gmbh Compounds which modulate the cb2 receptor
JP5746228B2 (ja) 2010-03-05 2015-07-08 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング Ｃｂ２受容体を選択的に調節するテトラゾール化合物
US8846936B2 (en) 2010-07-22 2014-09-30 Boehringer Ingelheim International Gmbh Sulfonyl compounds which modulate the CB2 receptor
EP2803668A1 (en) 2013-05-17 2014-11-19 Boehringer Ingelheim International Gmbh Novel (cyano-dimethyl-methyl)-isoxazoles and -[1,3,4]thiadiazoles

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3878248A (en) * 1971-05-03 1975-04-15 Monsanto Co Substituted alpha, alpha-dichloro-methane-sulfenyl chlorides
JPS5439028A (en) * 1977-08-31 1979-03-24 Hokko Chem Ind Co Ltd Acetanilide derivatives and bactericides containing the same for agricultural and horticultural, uses
US4329363A (en) * 1978-09-08 1982-05-11 Merck & Co., Inc. Substituted mercapto acid amides and their use
US4623662A (en) * 1985-05-23 1986-11-18 American Cyanamid Company Antiatherosclerotic ureas and thioureas
FR2540495B1 (fr) * 1983-02-07 1986-02-14 Roussel Uclaf Nouveaux derives de o-mercaptopropanamide et de ses homologues, leur procede de preparation, leur application comme medicaments, les compositions les renfermant et les nouveaux intermediaires obtenus
GB2149394B (en) * 1983-07-19 1986-09-24 American Cyanamid Co Ureas
US4859707A (en) * 1983-08-23 1989-08-22 Key Pharmaceuticals, Inc. Sulfur-substituted phenylacetamides
AU584669B2 (en) * 1985-02-04 1989-06-01 G.D. Searle & Co. Novel disubstituted 4-hydroxyphenylthio anilides
ZA871597B (en) * 1986-03-24 1988-10-26 Warner Lambert Co Substituted anilides of oleic,linoleic,or linolenic acid as inhibitors of acyl-coa:cholestrol acyltransferase
US4716175A (en) * 1987-02-24 1987-12-29 Warner-Lambert Company Saturated fatty acid amides as inhibitors of acyl-CoA:cholesterol acyltransferase
EP0361365A1 (en) * 1988-09-30 1990-04-04 E.R. SQUIBB & SONS, INC. Aminobenzoic and aminocyclohexane-carboylic acid compounds, compositions, and their method of use
WO1991004027A1 (en) * 1989-09-15 1991-04-04 Pfizer Inc. New n-aryl and n-heteroarylamide and urea derivatives as inhibitors of acyl coenzyme a: cholesterol acyl transferase (acat)

Also Published As

Publication number Publication date
DE69119434T2 (de) 1996-09-12
CA2096970A1 (en) 1992-05-27
DK0559898T3 (da) 1996-08-19
EP0559898A4 (enExample) 1994-01-12
JP2650096B2 (ja) 1997-09-03
KR930702254A (ko) 1993-09-08
US5475130A (en) 1995-12-12
ATE137744T1 (de) 1996-05-15
ES2088574T3 (es) 1996-08-16
WO1992009572A1 (en) 1992-06-11
DE69119434D1 (de) 1996-06-13
GR3020257T3 (en) 1996-09-30
EP0559898A1 (en) 1993-09-15
CA2096970C (en) 1998-07-14
EP0559898B1 (en) 1996-05-08

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