KE3155A - 4-amino-6,7-dimethoxy-2(4-(heterocyclocarbonyl)piperazin-1-yl)quinazolines - Google Patents

4-amino-6,7-dimethoxy-2(4-(heterocyclocarbonyl)piperazin-1-yl)quinazolines

Info

Publication number
KE3155A
KE3155A KE3155A KE315581A KE3155A KE 3155 A KE3155 A KE 3155A KE 3155 A KE3155 A KE 3155A KE 315581 A KE315581 A KE 315581A KE 3155 A KE3155 A KE 3155A
Authority
KE
Kenya
Prior art keywords
heterocyclocarbonyl
quinazolines
piperazin
dimethoxy
amino
Prior art date
Application number
KE3155A
Other languages
English (en)
Inventor
R A Partyka
R R Crenshaw
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/658,961 external-priority patent/US4001237A/en
Priority claimed from US05/658,979 external-priority patent/US4001238A/en
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of KE3155A publication Critical patent/KE3155A/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72Quinazolines; Hydrogenated quinazolines
    • C07D239/95Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Cardiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
KE3155A 1976-02-18 1981-08-25 4-amino-6,7-dimethoxy-2(4-(heterocyclocarbonyl)piperazin-1-yl)quinazolines KE3155A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US05/658,961 US4001237A (en) 1976-02-18 1976-02-18 Oxazole, isoxazole, thiazole and isothiazole amides
US05/658,979 US4001238A (en) 1976-02-18 1976-02-18 1,3,4-oxadiazole amides

Publications (1)

Publication Number Publication Date
KE3155A true KE3155A (en) 1981-09-18

Family

ID=27097727

Family Applications (1)

Application Number Title Priority Date Filing Date
KE3155A KE3155A (en) 1976-02-18 1981-08-25 4-amino-6,7-dimethoxy-2(4-(heterocyclocarbonyl)piperazin-1-yl)quinazolines

Country Status (16)

Country Link
JP (1) JPS584716B2 (US06589383-20030708-C00041.png)
CA (1) CA1081228A (US06589383-20030708-C00041.png)
CH (1) CH635838A5 (US06589383-20030708-C00041.png)
CY (1) CY1122A (US06589383-20030708-C00041.png)
DE (1) DE2707067A1 (US06589383-20030708-C00041.png)
DK (1) DK65177A (US06589383-20030708-C00041.png)
FI (1) FI770485A (US06589383-20030708-C00041.png)
FR (1) FR2348924A1 (US06589383-20030708-C00041.png)
GB (1) GB1533529A (US06589383-20030708-C00041.png)
IE (1) IE44614B1 (US06589383-20030708-C00041.png)
KE (1) KE3155A (US06589383-20030708-C00041.png)
LU (1) LU76802A1 (US06589383-20030708-C00041.png)
MY (1) MY8200110A (US06589383-20030708-C00041.png)
NL (1) NL7701753A (US06589383-20030708-C00041.png)
SE (1) SE7701732L (US06589383-20030708-C00041.png)
YU (4) YU45477A (US06589383-20030708-C00041.png)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5791987A (en) * 1980-11-26 1982-06-08 Sankyo Co Ltd Aminoquinazoline derivative and its preparation
US5994294A (en) * 1996-02-02 1999-11-30 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
US5932538A (en) * 1996-02-02 1999-08-03 Nitromed, Inc. Nitrosated and nitrosylated α-adrenergic receptor antagonist compounds, compositions and their uses
EP1517898A1 (de) * 2002-06-29 2005-03-30 Zentaris GmbH Aryl- und heteroarylcarbonylpiperazine und deren verwendung zur behandlung gutartiger und b sartiger tumorerkrankungen

Also Published As

Publication number Publication date
MY8200110A (en) 1982-12-31
DE2707067A1 (de) 1977-08-25
FI770485A (US06589383-20030708-C00041.png) 1977-08-19
FR2348924A1 (fr) 1977-11-18
YU267780A (en) 1983-06-30
IE44614B1 (en) 1982-01-27
CA1081228A (en) 1980-07-08
AU2242677A (en) 1978-07-06
SE7701732L (sv) 1977-08-19
LU76802A1 (US06589383-20030708-C00041.png) 1977-09-12
JPS52102286A (en) 1977-08-27
YU161282A (en) 1982-10-31
FR2348924B1 (US06589383-20030708-C00041.png) 1980-05-09
NL7701753A (nl) 1977-08-22
JPS584716B2 (ja) 1983-01-27
IE44614L (en) 1977-08-18
DK65177A (da) 1977-08-19
GB1533529A (en) 1978-11-29
YU161182A (en) 1982-10-31
YU45477A (en) 1982-10-31
CH635838A5 (en) 1983-04-29
CY1122A (en) 1981-12-04

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