JPWO2023076303A5 - - Google Patents

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Publication number
JPWO2023076303A5
JPWO2023076303A5 JP2024525065A JP2024525065A JPWO2023076303A5 JP WO2023076303 A5 JPWO2023076303 A5 JP WO2023076303A5 JP 2024525065 A JP2024525065 A JP 2024525065A JP 2024525065 A JP2024525065 A JP 2024525065A JP WO2023076303 A5 JPWO2023076303 A5 JP WO2023076303A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
compound
formula
tyrosine kinase
cancer
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024525065A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024542984A5 (https=
JP2024542984A (ja
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/047767 external-priority patent/WO2023076303A1/en
Publication of JP2024542984A publication Critical patent/JP2024542984A/ja
Publication of JP2024542984A5 publication Critical patent/JP2024542984A5/ja
Publication of JPWO2023076303A5 publication Critical patent/JPWO2023076303A5/ja
Pending legal-status Critical Current

Links

JP2024525065A 2021-10-26 2022-10-25 がんを治療および予防するためのピペリジニルピラジン-カルボキサミド化合物、およびbtkを分解するためのピペリジニルピラジン-カルボキサミド化合物 Pending JP2024542984A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202163263081P 2021-10-26 2021-10-26
US63/263,081 2021-10-26
US202263391671P 2022-07-22 2022-07-22
US63/391,671 2022-07-22
PCT/US2022/047767 WO2023076303A1 (en) 2021-10-26 2022-10-25 Piperidinylpyrazine-carboxamide compounds for treating and preventing cancer and for degrading btk

Publications (3)

Publication Number Publication Date
JP2024542984A JP2024542984A (ja) 2024-11-19
JP2024542984A5 JP2024542984A5 (https=) 2025-09-09
JPWO2023076303A5 true JPWO2023076303A5 (https=) 2025-09-09

Family

ID=84361163

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024525065A Pending JP2024542984A (ja) 2021-10-26 2022-10-25 がんを治療および予防するためのピペリジニルピラジン-カルボキサミド化合物、およびbtkを分解するためのピペリジニルピラジン-カルボキサミド化合物

Country Status (9)

Country Link
US (1) US12377106B2 (https=)
EP (1) EP4422630A1 (https=)
JP (1) JP2024542984A (https=)
KR (1) KR20240090898A (https=)
AU (1) AU2022379494A1 (https=)
CA (1) CA3236073A1 (https=)
IL (1) IL312357A (https=)
MX (1) MX2024004899A (https=)
WO (1) WO2023076303A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7600123B2 (ja) 2018-10-15 2024-12-16 ニューリックス セラピューティクス,インコーポレイテッド ユビキチンプロテオソーム経路を介してbtkを分解するための二官能性化合物
WO2020167518A1 (en) 2019-02-13 2020-08-20 Nurix Therapeutics, Inc. Bifunctional compounds for degrading btk via ubiquitin proteosome pathway
US11820781B2 (en) 2019-12-04 2023-11-21 Nurix Therapeutics, Inc. Bifunctional compounds for degrading BTK via ubiquitin proteosome pathway
AU2022379494A1 (en) 2021-10-26 2024-05-30 Nurix Therapeutics, Inc. Piperidinylpyrazine-carboxamide compounds for treating and preventing cancer and for degrading btk

Family Cites Families (38)

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