JP2024542984A5 - - Google Patents

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Publication number
JP2024542984A5
JP2024542984A5 JP2024525065A JP2024525065A JP2024542984A5 JP 2024542984 A5 JP2024542984 A5 JP 2024542984A5 JP 2024525065 A JP2024525065 A JP 2024525065A JP 2024525065 A JP2024525065 A JP 2024525065A JP 2024542984 A5 JP2024542984 A5 JP 2024542984A5
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JP
Japan
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JP2024525065A
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Japanese (ja)
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JPWO2023076303A5 (https=
JP2024542984A (ja
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Publication date
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Priority claimed from PCT/US2022/047767 external-priority patent/WO2023076303A1/en
Publication of JP2024542984A publication Critical patent/JP2024542984A/ja
Publication of JP2024542984A5 publication Critical patent/JP2024542984A5/ja
Publication of JPWO2023076303A5 publication Critical patent/JPWO2023076303A5/ja
Pending legal-status Critical Current

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JP2024525065A 2021-10-26 2022-10-25 がんを治療および予防するためのピペリジニルピラジン-カルボキサミド化合物、およびbtkを分解するためのピペリジニルピラジン-カルボキサミド化合物 Pending JP2024542984A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US202163263081P 2021-10-26 2021-10-26
US63/263,081 2021-10-26
US202263391671P 2022-07-22 2022-07-22
US63/391,671 2022-07-22
PCT/US2022/047767 WO2023076303A1 (en) 2021-10-26 2022-10-25 Piperidinylpyrazine-carboxamide compounds for treating and preventing cancer and for degrading btk

Publications (3)

Publication Number Publication Date
JP2024542984A JP2024542984A (ja) 2024-11-19
JP2024542984A5 true JP2024542984A5 (https=) 2025-09-09
JPWO2023076303A5 JPWO2023076303A5 (https=) 2025-09-09

Family

ID=84361163

Family Applications (1)

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JP2024525065A Pending JP2024542984A (ja) 2021-10-26 2022-10-25 がんを治療および予防するためのピペリジニルピラジン-カルボキサミド化合物、およびbtkを分解するためのピペリジニルピラジン-カルボキサミド化合物

Country Status (9)

Country Link
US (1) US12377106B2 (https=)
EP (1) EP4422630A1 (https=)
JP (1) JP2024542984A (https=)
KR (1) KR20240090898A (https=)
AU (1) AU2022379494A1 (https=)
CA (1) CA3236073A1 (https=)
IL (1) IL312357A (https=)
MX (1) MX2024004899A (https=)
WO (1) WO2023076303A1 (https=)

Families Citing this family (4)

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Publication number Priority date Publication date Assignee Title
JP7600123B2 (ja) 2018-10-15 2024-12-16 ニューリックス セラピューティクス,インコーポレイテッド ユビキチンプロテオソーム経路を介してbtkを分解するための二官能性化合物
WO2020167518A1 (en) 2019-02-13 2020-08-20 Nurix Therapeutics, Inc. Bifunctional compounds for degrading btk via ubiquitin proteosome pathway
US11820781B2 (en) 2019-12-04 2023-11-21 Nurix Therapeutics, Inc. Bifunctional compounds for degrading BTK via ubiquitin proteosome pathway
AU2022379494A1 (en) 2021-10-26 2024-05-30 Nurix Therapeutics, Inc. Piperidinylpyrazine-carboxamide compounds for treating and preventing cancer and for degrading btk

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