JPWO2022208113A5 - - Google Patents

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Publication number
JPWO2022208113A5
JPWO2022208113A5 JP2023560997A JP2023560997A JPWO2022208113A5 JP WO2022208113 A5 JPWO2022208113 A5 JP WO2022208113A5 JP 2023560997 A JP2023560997 A JP 2023560997A JP 2023560997 A JP2023560997 A JP 2023560997A JP WO2022208113 A5 JPWO2022208113 A5 JP WO2022208113A5
Authority
JP
Japan
Prior art keywords
dimethyl
cyclopropyl
azabicyclo
carboxamide
hexane
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023560997A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024511881A (ja
JP2024511881A5 (https=
Publication date
Priority claimed from GBGB2104742.8A external-priority patent/GB202104742D0/en
Priority claimed from GBGB2107026.3A external-priority patent/GB202107026D0/en
Application filed filed Critical
Priority claimed from PCT/GB2022/050836 external-priority patent/WO2022208113A1/en
Publication of JP2024511881A publication Critical patent/JP2024511881A/ja
Publication of JPWO2022208113A5 publication Critical patent/JPWO2022208113A5/ja
Publication of JP2024511881A5 publication Critical patent/JP2024511881A5/ja
Pending legal-status Critical Current

Links

JP2023560997A 2021-04-01 2022-04-01 SARS-COV-2 Mpro阻害剤化合物 Pending JP2024511881A (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB2104742.8 2021-04-01
GBGB2104742.8A GB202104742D0 (en) 2021-04-01 2021-04-01 Sars-Cov-2 MPRO inhibitor compounds
GBGB2107026.3A GB202107026D0 (en) 2021-05-17 2021-05-17 SARS-COV-2 MPRO inhibitor compounds
GB2107026.3 2021-05-17
PCT/GB2022/050836 WO2022208113A1 (en) 2021-04-01 2022-04-01 Sars-cov-2 mpro inhibitor compounds

Publications (3)

Publication Number Publication Date
JP2024511881A JP2024511881A (ja) 2024-03-15
JPWO2022208113A5 true JPWO2022208113A5 (https=) 2025-04-09
JP2024511881A5 JP2024511881A5 (https=) 2025-04-09

Family

ID=81307814

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023560997A Pending JP2024511881A (ja) 2021-04-01 2022-04-01 SARS-COV-2 Mpro阻害剤化合物

Country Status (7)

Country Link
US (1) US20240217930A1 (https=)
EP (1) EP4313305A1 (https=)
JP (1) JP2024511881A (https=)
KR (1) KR20240004275A (https=)
AU (1) AU2022247287A1 (https=)
CA (1) CA3213008A1 (https=)
WO (1) WO2022208113A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2024525589A (ja) 2021-07-09 2024-07-12 アリゴス セラピューティクス インコーポレイテッド 抗ウイルス化合物
WO2023043816A1 (en) 2021-09-17 2023-03-23 Aligos Therapeutics, Inc. Anti-viral compounds for treating coronavirus, picornavirus, and norovirus infections
GB202214644D0 (en) * 2022-10-05 2022-11-16 Heptares Therapeutics Ltd Sars-cov-2 mpro inhibitors and uses thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7244721B2 (en) * 2000-07-21 2007-07-17 Schering Corporation Peptides as NS3-serine protease inhibitors of hepatitis C virus
CN1498224A (zh) * 2000-07-21 2004-05-19 ���鹫˾ 用作丙型肝炎病毒ns3-丝氨酸蛋白酶抑制剂的新型肽
CA3180177A1 (en) * 2020-05-08 2021-11-11 The Board Of Trustees Of The Leland Stanford Junior University Protease inhibitors for treatment or prevention of coronavirus disease

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