JPWO2022107755A5 - - Google Patents

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Publication number
JPWO2022107755A5
JPWO2022107755A5 JP2022563761A JP2022563761A JPWO2022107755A5 JP WO2022107755 A5 JPWO2022107755 A5 JP WO2022107755A5 JP 2022563761 A JP2022563761 A JP 2022563761A JP 2022563761 A JP2022563761 A JP 2022563761A JP WO2022107755 A5 JPWO2022107755 A5 JP WO2022107755A5
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JP
Japan
Prior art keywords
alkyloxy
hydrogen atom
acridinium salt
formula
salt
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Application number
JP2022563761A
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English (en)
Japanese (ja)
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JPWO2022107755A1 (https=
JP7685522B2 (ja
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Priority claimed from PCT/JP2021/042049 external-priority patent/WO2022107755A1/ja
Publication of JPWO2022107755A1 publication Critical patent/JPWO2022107755A1/ja
Publication of JPWO2022107755A5 publication Critical patent/JPWO2022107755A5/ja
Application granted granted Critical
Publication of JP7685522B2 publication Critical patent/JP7685522B2/ja
Active legal-status Critical Current
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JP2022563761A 2020-11-17 2021-11-16 新規アクリジニウム塩およびその製造方法 Active JP7685522B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2020191118 2020-11-17
JP2020191118 2020-11-17
PCT/JP2021/042049 WO2022107755A1 (ja) 2020-11-17 2021-11-16 新規アクリジニウム塩およびその製造方法

Publications (3)

Publication Number Publication Date
JPWO2022107755A1 JPWO2022107755A1 (https=) 2022-05-27
JPWO2022107755A5 true JPWO2022107755A5 (https=) 2024-09-10
JP7685522B2 JP7685522B2 (ja) 2025-05-29

Family

ID=81707996

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022563761A Active JP7685522B2 (ja) 2020-11-17 2021-11-16 新規アクリジニウム塩およびその製造方法

Country Status (6)

Country Link
US (1) US20230278960A1 (https=)
EP (1) EP4249077A4 (https=)
JP (1) JP7685522B2 (https=)
CN (1) CN116783167A (https=)
AR (1) AR124071A1 (https=)
WO (1) WO2022107755A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20250129029A1 (en) * 2021-09-06 2025-04-24 Osaka University Acridine compound
CN116082361B (zh) * 2023-04-11 2023-06-13 和鼎(南京)医药技术有限公司 一种制备玛巴洛沙韦中间体和玛巴洛沙韦的方法

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI2320908T1 (sl) 2008-07-25 2014-05-30 Viiv Healthcare Company Predzdravila dolutegravirja
WO2010011819A1 (en) 2008-07-25 2010-01-28 Smithkline Beecham Corporation Chemical compounds
CA2744019C (en) 2008-12-11 2017-03-14 Shionogi & Co., Ltd. Synthesis of carbamoylpyridone hiv integrase inhibitors and intermediates
KR101682058B1 (ko) 2008-12-11 2016-12-02 비이브 헬쓰케어 컴퍼니 카르바모일피리돈 hiv 인테그라제 억제제를 위한 제조방법 및 중간체
TWI518084B (zh) 2009-03-26 2016-01-21 鹽野義製藥股份有限公司 哌喃酮與吡啶酮衍生物之製造方法
US20140011995A1 (en) 2010-08-05 2014-01-09 Yukihito Sumino Process for Preparing Compound Having HIV Integrase Inhibitory Activity
WO2014128545A2 (en) 2013-02-19 2014-08-28 Aurobindo Pharma Limited An improved process for the preparation of dolutegravir
EP3022209B1 (en) 2013-07-17 2018-03-07 ratiopharm GmbH Dolutegravir potassium salt
WO2015019310A1 (en) 2013-08-07 2015-02-12 Mylan Laboratories Ltd Process for the preparation of dolute-gravir and intermediates thereof
US9856271B2 (en) 2014-01-21 2018-01-02 Laurus Labs Limited Process for the preparation of dolutegravir and pharmaceutically acceptable salts thereof
ZA201503540B (en) 2014-05-20 2016-10-26 Cipla Ltd Process for preparing polycyclic carbamoyl pyridone derivatives
WO2016092527A1 (en) 2014-12-12 2016-06-16 Sun Pharmaceutical Industries Limited A process for the preparation of dolutegravir
US10730888B2 (en) 2015-02-06 2020-08-04 Mylan Laboratories Limited Process for the preparation of dolutegravir
BR112017022550B1 (pt) 2015-04-28 2021-02-23 Shionogi & Co., Ltd derivados policíclicos de piridona substituída
WO2016196816A1 (en) * 2015-06-03 2016-12-08 The University Of North Carolina At Chapel Hill Photoredox-catalyzed direct c-h functionalization of arenes
AU2016374416A1 (en) 2015-12-15 2018-06-14 Shionogi & Co., Ltd. Medicine for treating influenza characterized by comprising combination of cap-dependent endonuclease inhibitor with anti-influenza drug
JP6924839B2 (ja) * 2017-10-06 2021-08-25 塩野義製薬株式会社 置換された多環性ピリドン誘導体の立体選択的な製造方法
WO2020176804A1 (en) * 2019-02-28 2020-09-03 The University Of North Carolina At Chapel Hill Direct aromatic carbon-oxygen and carbon-hydrogen bond functionalization via organic photoredox catalyst

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