JPWO2022060094A5 - - Google Patents

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Publication number
JPWO2022060094A5
JPWO2022060094A5 JP2023515773A JP2023515773A JPWO2022060094A5 JP WO2022060094 A5 JPWO2022060094 A5 JP WO2022060094A5 JP 2023515773 A JP2023515773 A JP 2023515773A JP 2023515773 A JP2023515773 A JP 2023515773A JP WO2022060094 A5 JPWO2022060094 A5 JP WO2022060094A5
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JP
Japan
Prior art keywords
methyl
dihydropyrimido
pyrimidin
pyridin
oxo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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Application number
JP2023515773A
Other languages
English (en)
Japanese (ja)
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JP7824667B2 (ja
JP2023541052A5 (https=
JP2023541052A (ja
Publication date
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Priority claimed from PCT/KR2021/012616 external-priority patent/WO2022060094A1/ko
Publication of JP2023541052A publication Critical patent/JP2023541052A/ja
Publication of JP2023541052A5 publication Critical patent/JP2023541052A5/ja
Publication of JPWO2022060094A5 publication Critical patent/JPWO2022060094A5/ja
Application granted granted Critical
Publication of JP7824667B2 publication Critical patent/JP7824667B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2023515773A 2020-09-16 2021-09-15 ピリミドピリミジノン化合物及びそれを含む薬剤学的組成物 Active JP7824667B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
KR20200119100 2020-09-16
KR10-2020-0119100 2020-09-16
PCT/KR2021/012616 WO2022060094A1 (ko) 2020-09-16 2021-09-15 피리미도 피리미디논 화합물 및 그를 포함하는 약제학적 조성물

Publications (4)

Publication Number Publication Date
JP2023541052A JP2023541052A (ja) 2023-09-27
JP2023541052A5 JP2023541052A5 (https=) 2024-09-24
JPWO2022060094A5 true JPWO2022060094A5 (https=) 2024-09-24
JP7824667B2 JP7824667B2 (ja) 2026-03-05

Family

ID=80777269

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023515773A Active JP7824667B2 (ja) 2020-09-16 2021-09-15 ピリミドピリミジノン化合物及びそれを含む薬剤学的組成物

Country Status (11)

Country Link
US (1) US12590098B2 (https=)
EP (1) EP4215533B1 (https=)
JP (1) JP7824667B2 (https=)
KR (1) KR102673031B1 (https=)
CN (1) CN116137815B (https=)
AU (1) AU2021344164A1 (https=)
BR (1) BR112023004179A2 (https=)
CA (1) CA3190461A1 (https=)
IL (1) IL300920A (https=)
MX (1) MX2023003087A (https=)
WO (1) WO2022060094A1 (https=)

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MXPA06001098A (es) * 2003-07-29 2006-04-24 Irm Llc Compuestos y composiciones utiles como inhibidores de proteina cinasa.
BRPI0514738A (pt) 2004-08-31 2008-06-24 Hoffmann La Roche derivados de amida de 3-fenil-diidropirimido[4,5-d]pirimidinonas, sua fabricação e aplicação como agentes farmacêuticos
UY29439A1 (es) * 2005-03-25 2006-10-02 Glaxo Group Ltd Nuevos compuestos
RU2007147917A (ru) * 2005-06-10 2009-07-20 Айрм Ллк (Bm) Соединения, поддерживающие плюрипотентность эмбриональных стволовых клеток
EP2455382B1 (en) 2005-12-13 2016-10-26 Incyte Holdings Corporation Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors
GB201315072D0 (en) 2013-08-23 2013-10-02 Galapagos Nv Novel compounds and pharmaceutical compositions thereoffor the treatment of proliferative disorders
AU2017291812B2 (en) * 2016-07-05 2023-12-14 Dana-Farber Cancer Institute, Inc. Bicyclic urea kinase inhibitors and uses thereof
KR102591947B1 (ko) * 2018-04-19 2023-10-25 길리애드 사이언시즈, 인코포레이티드 Pd-1/pd-l1 억제제
KR102382613B1 (ko) * 2020-01-15 2022-04-06 한국과학기술연구원 단백질 키나아제 저해 활성을 갖는 7-아미노-3,4-디히드로피리미도피리미딘-2-온 유도체 및 이를 포함하는 치료용 약학 조성물

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