JPWO2021150673A5 - - Google Patents

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Publication number
JPWO2021150673A5
JPWO2021150673A5 JP2022544753A JP2022544753A JPWO2021150673A5 JP WO2021150673 A5 JPWO2021150673 A5 JP WO2021150673A5 JP 2022544753 A JP2022544753 A JP 2022544753A JP 2022544753 A JP2022544753 A JP 2022544753A JP WO2021150673 A5 JPWO2021150673 A5 JP WO2021150673A5
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JP
Japan
Prior art keywords
ethoxy
glu
amino
acetyl
carboxyphenoxy
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022544753A
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English (en)
Japanese (ja)
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JP2023511441A (ja
JP2023511441A5 (https=
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/014302 external-priority patent/WO2021150673A1/en
Publication of JP2023511441A publication Critical patent/JP2023511441A/ja
Publication of JP2023511441A5 publication Critical patent/JP2023511441A5/ja
Publication of JPWO2021150673A5 publication Critical patent/JPWO2021150673A5/ja
Pending legal-status Critical Current

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JP2022544753A 2020-01-23 2021-01-21 Gip/glp1共アゴニスト化合物 Pending JP2023511441A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202062964932P 2020-01-23 2020-01-23
US62/964,932 2020-01-23
PCT/US2021/014302 WO2021150673A1 (en) 2020-01-23 2021-01-21 Gip/glp1 co-agonist compounds

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2025195273A Division JP2026069790A (ja) 2020-01-23 2025-11-14 Gip/glp1共アゴニスト化合物

Publications (3)

Publication Number Publication Date
JP2023511441A JP2023511441A (ja) 2023-03-17
JP2023511441A5 JP2023511441A5 (https=) 2024-01-25
JPWO2021150673A5 true JPWO2021150673A5 (https=) 2024-01-25

Family

ID=74592824

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022544753A Pending JP2023511441A (ja) 2020-01-23 2021-01-21 Gip/glp1共アゴニスト化合物

Country Status (13)

Country Link
US (1) US20230265151A1 (https=)
EP (1) EP4093757A1 (https=)
JP (1) JP2023511441A (https=)
KR (1) KR20220131292A (https=)
CN (1) CN115298207A (https=)
AR (1) AR121093A1 (https=)
AU (1) AU2021211451B2 (https=)
BR (1) BR112022014397A2 (https=)
CA (1) CA3165430A1 (https=)
IL (1) IL294955A (https=)
MX (1) MX2022009149A (https=)
TW (1) TWI770781B (https=)
WO (1) WO2021150673A1 (https=)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI912614B (zh) * 2017-12-21 2026-01-21 美商美國禮來大藥廠 腸促胰島素(incretin)類似物及其用途
WO2022159395A1 (en) 2021-01-20 2022-07-28 Viking Therapeutics, Inc. Compositions and methods for the treatment of metabolic and liver disorders
JP2024508745A (ja) * 2021-02-17 2024-02-28 イーライ リリー アンド カンパニー Gip/glp1デュアルアゴニスト治療方法
IL310377A (en) 2021-08-30 2024-03-01 Mindrank Ai Ltd Novel aryl ether substituted heterocyclic compound as glp1r agonist
MX2024003236A (es) 2021-09-15 2024-06-19 Viking Therapeutics Inc Composiciones y metodos para el tratamiento de trastornos metabolicos y hepaticos.
CN117586373A (zh) * 2022-08-10 2024-02-23 成都奥达生物科技有限公司 一种长效双激动剂化合物
CN116023444B (zh) * 2022-08-12 2023-08-01 重庆宸安生物制药有限公司 一种gip和glp-1双受体激动剂多肽化合物及其应用
WO2024165571A2 (en) 2023-02-06 2024-08-15 E-Therapeutics Plc Inhibitors of expression and/or function
WO2025125576A2 (en) 2023-12-15 2025-06-19 E-Therapeutics Plc Inhibitors of expression and/or function
WO2025133348A1 (en) 2023-12-22 2025-06-26 E-Therapeutics Plc Inhibitors of expression and/or function
EP4686757A1 (en) 2024-07-31 2026-02-04 e-therapeutics PLC Inhibitors of expression and/or function
WO2025196502A1 (en) 2024-03-20 2025-09-25 North Carolina Agricultural & Technical State University Choline kinase inhibitors as a therapeutic treatment for obesity

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR080592A1 (es) * 2010-03-26 2012-04-18 Lilly Co Eli Peptido con actividad para el gip-r y glp-1-r, formulacion famaceutica que lo comprende, su uso para preparar un medicamento util para el tratamiento de diabetes mellitus y para inducir la perdida de peso
WO2012167744A1 (en) * 2011-06-10 2012-12-13 Beijing Hanmi Pharmaceutical Co., Ltd. Glucose dependent insulinotropic polypeptide analogs, pharmaceutical compositions and use thereof
JP6228187B2 (ja) * 2012-05-03 2017-11-08 ジーランド ファーマ アクティーゼルスカブ Gip−glp−1デュアルアゴニスト化合物及び方法
HK1211232A1 (en) * 2012-12-21 2016-05-20 Sanofi Exendin-4 derivatives as dual glp1/gip or trigonal glp1/gip/glucagon agonists
MX2016005556A (es) * 2013-11-06 2016-07-15 Zealand Pharma As Compuestos agonistas duales de gip-glp-1 y procedimientos.
JO3575B1 (ar) 2015-01-09 2020-07-05 Lilly Co Eli مركبات مساعد مشترك من gip وglp-1
TWI783244B (zh) * 2015-06-22 2022-11-11 美商美國禮來大藥廠 升糖素及glp-1共激動劑化合物
TWI767095B (zh) * 2017-12-21 2022-06-11 美商美國禮來大藥廠 腸促胰島素(incretin)類似物及其用途
CN112469731B (zh) * 2018-07-23 2024-11-29 伊莱利利公司 Gip/glp1共激动剂化合物

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