JPWO2021132472A1 - - Google Patents
Info
- Publication number
- JPWO2021132472A1 JPWO2021132472A1 JP2021567619A JP2021567619A JPWO2021132472A1 JP WO2021132472 A1 JPWO2021132472 A1 JP WO2021132472A1 JP 2021567619 A JP2021567619 A JP 2021567619A JP 2021567619 A JP2021567619 A JP 2021567619A JP WO2021132472 A1 JPWO2021132472 A1 JP WO2021132472A1
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/08—Drugs for disorders of the urinary system of the prostate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A61K31/343—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide condensed with a carbocyclic ring, e.g. coumaran, bufuralol, befunolol, clobenfurol, amiodarone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A61K31/416—1,2-Diazoles condensed with carbocyclic ring systems, e.g. indazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
- A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/423—Oxazoles condensed with carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Urology & Nephrology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicinal Preparation (AREA)
Priority Applications (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2024090606A JP7779953B2 (ja) | 2019-12-25 | 2024-06-04 | 慢性前立腺炎／慢性骨盤痛症候群の予防及び／又は治療剤 |
| JP2025199177A JP2026015542A (ja) | 2019-12-25 | 2025-11-19 | 慢性前立腺炎／慢性骨盤痛症候群の予防及び／又は治療剤 |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2019233865 | 2019-12-25 | ||
| JP2019233865 | 2019-12-25 | ||
| PCT/JP2020/048479 WO2021132472A1 (ja) | 2019-12-25 | 2020-12-24 | 慢性前立腺炎／慢性骨盤痛症候群の予防及び／又は治療剤 |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024090606A Division JP7779953B2 (ja) | 2019-12-25 | 2024-06-04 | 慢性前立腺炎／慢性骨盤痛症候群の予防及び／又は治療剤 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2021132472A1 true JPWO2021132472A1 (https=) | 2021-07-01 |
| JPWO2021132472A5 JPWO2021132472A5 (https=) | 2024-04-30 |
| JP7499789B2 JP7499789B2 (ja) | 2024-06-14 |
Family
ID=76575232
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021567619A Active JP7499789B2 (ja) | 2019-12-25 | 2020-12-24 | 慢性前立腺炎／慢性骨盤痛症候群の予防及び／又は治療剤 |
| JP2024090606A Active JP7779953B2 (ja) | 2019-12-25 | 2024-06-04 | 慢性前立腺炎／慢性骨盤痛症候群の予防及び／又は治療剤 |
| JP2025199177A Pending JP2026015542A (ja) | 2019-12-25 | 2025-11-19 | 慢性前立腺炎／慢性骨盤痛症候群の予防及び／又は治療剤 |
Family Applications After (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024090606A Active JP7779953B2 (ja) | 2019-12-25 | 2024-06-04 | 慢性前立腺炎／慢性骨盤痛症候群の予防及び／又は治療剤 |
| JP2025199177A Pending JP2026015542A (ja) | 2019-12-25 | 2025-11-19 | 慢性前立腺炎／慢性骨盤痛症候群の予防及び／又は治療剤 |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US12599589B2 (https=) |
| EP (1) | EP4082573A4 (https=) |
| JP (3) | JP7499789B2 (https=) |
| KR (1) | KR20220120646A (https=) |
| CN (2) | CN119303087A (https=) |
| AU (1) | AU2020413313B2 (https=) |
| BR (1) | BR112022012485A2 (https=) |
| CA (1) | CA3165891A1 (https=) |
| CO (1) | CO2022010343A2 (https=) |
| EC (1) | ECSP22058286A (https=) |
| IL (1) | IL294191A (https=) |
| MX (1) | MX2022007936A (https=) |
| PE (1) | PE20230164A1 (https=) |
| PH (1) | PH12022551578A1 (https=) |
| UA (1) | UA130283C2 (https=) |
| WO (1) | WO2021132472A1 (https=) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN116082247B (zh) * | 2023-01-19 | 2025-08-01 | 浙江工业大学 | 一种苯并咪唑类衍生物及其应用 |
| CN121401398A (zh) * | 2025-12-29 | 2026-01-27 | 汕头市中心医院 | 一种实验性自身免疫性前列腺炎大鼠模型的构建方法 |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2013024898A1 (ja) * | 2011-08-18 | 2013-02-21 | 日本新薬株式会社 | ヘテロ環誘導体及び医薬 |
| JP2013508325A (ja) * | 2009-10-23 | 2013-03-07 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ミクロソームプロスタグランジンｅ２シンターゼ−１のインヒビター |
| JP2015501784A (ja) * | 2011-11-04 | 2015-01-19 | グラクソスミスクライン、インテレクチュアル、プロパティー、ナンバー２、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｎｏ．２ Ｌｉｍｉｔｅｄ | 治療の方法 |
| WO2017073709A1 (ja) * | 2015-10-29 | 2017-05-04 | あすか製薬株式会社 | ピリミジン誘導体 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UY32470A (es) | 2009-03-05 | 2010-10-29 | Boehringer Ingelheim Int | Derivados de 2-{2-cloro-5-[(sustituido) metil]fenilamino} -1-metil]fenilamino}-1-metilbencimidazol-5-carboxamidas-n-(sustituidas) y sus sales fisiológicamente aceptables, composiciones conteniéndolos y aplicaciones |
| WO2011023812A1 (en) | 2009-08-27 | 2011-03-03 | Novasaid Ab | Microsomal prostaglandin e synthase-1 (mpges1) inhibitors |
| TW201206440A (en) * | 2010-04-28 | 2012-02-16 | Astellas Pharma Inc | Prophylactic or therapeutic agent for diseases associated with pains in urinary organs |
| US8759537B2 (en) | 2010-08-20 | 2014-06-24 | Boehringer Ingelheim International Gmbh | 3H-imidazo [4, 5-C] pyridine-6-carboxamides as anti-inflammatory agents |
| US8586604B2 (en) | 2010-08-20 | 2013-11-19 | Boehringer Ingelheim International Gmbh | Inhibitors of the microsomal prostaglandin E2 synthase-1 |
| UY33779A (es) | 2010-12-10 | 2012-07-31 | Boehringer Ingelheim Int | ?2-(fenilamino)-1H-bencimidazol-5-carboxamidas novedosas? |
| AR086254A1 (es) | 2011-05-26 | 2013-11-27 | Lilly Co Eli | Derivados de imidazol utiles para el tratamiento de artritis |
-
2020
- 2020-12-24 CN CN202411363159.XA patent/CN119303087A/zh active Pending
- 2020-12-24 KR KR1020227025732A patent/KR20220120646A/ko active Pending
- 2020-12-24 EP EP20905872.6A patent/EP4082573A4/en active Pending
- 2020-12-24 WO PCT/JP2020/048479 patent/WO2021132472A1/ja not_active Ceased
- 2020-12-24 AU AU2020413313A patent/AU2020413313B2/en active Active
- 2020-12-24 US US17/788,516 patent/US12599589B2/en active Active
- 2020-12-24 PH PH1/2022/551578A patent/PH12022551578A1/en unknown
- 2020-12-24 PE PE2022001326A patent/PE20230164A1/es unknown
- 2020-12-24 IL IL294191A patent/IL294191A/en unknown
- 2020-12-24 JP JP2021567619A patent/JP7499789B2/ja active Active
- 2020-12-24 MX MX2022007936A patent/MX2022007936A/es unknown
- 2020-12-24 UA UAA202202629A patent/UA130283C2/uk unknown
- 2020-12-24 CN CN202080090316.8A patent/CN114867495B/zh active Active
- 2020-12-24 CA CA3165891A patent/CA3165891A1/en active Pending
- 2020-12-24 BR BR112022012485A patent/BR112022012485A2/pt unknown
-
2022
- 2022-07-22 CO CONC2022/0010343A patent/CO2022010343A2/es unknown
- 2022-07-25 EC ECSENADI202258286A patent/ECSP22058286A/es unknown
-
2024
- 2024-06-04 JP JP2024090606A patent/JP7779953B2/ja active Active
-
2025
- 2025-11-19 JP JP2025199177A patent/JP2026015542A/ja active Pending
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2013508325A (ja) * | 2009-10-23 | 2013-03-07 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ミクロソームプロスタグランジンｅ２シンターゼ−１のインヒビター |
| WO2013024898A1 (ja) * | 2011-08-18 | 2013-02-21 | 日本新薬株式会社 | ヘテロ環誘導体及び医薬 |
| JP2015501784A (ja) * | 2011-11-04 | 2015-01-19 | グラクソスミスクライン、インテレクチュアル、プロパティー、ナンバー２、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｎｏ．２ Ｌｉｍｉｔｅｄ | 治療の方法 |
| WO2017073709A1 (ja) * | 2015-10-29 | 2017-05-04 | あすか製薬株式会社 | ピリミジン誘導体 |
Non-Patent Citations (1)
| Title |
|---|
| NAUSCH B. ET AL.: "Canephron(R) N reduces pain in experimental cystitis and prostatitis putatively by inhibition of PGE", EUROPEAN UROLOGY SUPPLEMENTS, vol. 15, no. 3, JPN6021006284, 2016, pages 262, ISSN: 0005316920 * |
Also Published As
| Publication number | Publication date |
|---|---|
| ECSP22058286A (es) | 2022-09-30 |
| JP2024103724A (ja) | 2024-08-01 |
| JP2026015542A (ja) | 2026-01-29 |
| MX2022007936A (es) | 2022-10-27 |
| PE20230164A1 (es) | 2023-02-01 |
| CA3165891A1 (en) | 2021-07-01 |
| BR112022012485A2 (pt) | 2022-09-06 |
| AU2020413313B2 (en) | 2025-11-27 |
| EP4082573A4 (en) | 2024-01-10 |
| NZ789736A (en) | 2025-10-31 |
| CO2022010343A2 (es) | 2022-10-31 |
| JP7779953B2 (ja) | 2025-12-03 |
| US12599589B2 (en) | 2026-04-14 |
| US20230094705A1 (en) | 2023-03-30 |
| CN114867495A (zh) | 2022-08-05 |
| AU2020413313A1 (en) | 2022-07-14 |
| JP7499789B2 (ja) | 2024-06-14 |
| PH12022551578A1 (en) | 2023-11-29 |
| WO2021132472A1 (ja) | 2021-07-01 |
| EP4082573A1 (en) | 2022-11-02 |
| CN119303087A (zh) | 2025-01-14 |
| KR20220120646A (ko) | 2022-08-30 |
| UA130283C2 (uk) | 2026-01-07 |
| CN114867495B (zh) | 2024-10-18 |
| IL294191A (en) | 2022-08-01 |
Similar Documents
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20220726 |
|
| RD03 | Notification of appointment of power of attorney |
Free format text: JAPANESE INTERMEDIATE CODE: A7423 Effective date: 20231031 |
|
| RD04 | Notification of resignation of power of attorney |
Free format text: JAPANESE INTERMEDIATE CODE: A7424 Effective date: 20231106 |
|
| A621 | Written request for application examination |
Free format text: JAPANESE INTERMEDIATE CODE: A621 Effective date: 20231222 |
|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20240417 |
|
| A871 | Explanation of circumstances concerning accelerated examination |
Free format text: JAPANESE INTERMEDIATE CODE: A871 Effective date: 20240417 |
|
| TRDD | Decision of grant or rejection written | ||
| A01 | Written decision to grant a patent or to grant a registration (utility model) |
Free format text: JAPANESE INTERMEDIATE CODE: A01 Effective date: 20240507 |
|
| A61 | First payment of annual fees (during grant procedure) |
Free format text: JAPANESE INTERMEDIATE CODE: A61 Effective date: 20240604 |
|
| R150 | Certificate of patent or registration of utility model |
Ref document number: 7499789 Country of ref document: JP Free format text: JAPANESE INTERMEDIATE CODE: R150 |