JPWO2021117861A1 - - Google Patents

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Publication number
JPWO2021117861A1
JPWO2021117861A1 JP2021564057A JP2021564057A JPWO2021117861A1 JP WO2021117861 A1 JPWO2021117861 A1 JP WO2021117861A1 JP 2021564057 A JP2021564057 A JP 2021564057A JP 2021564057 A JP2021564057 A JP 2021564057A JP WO2021117861 A1 JPWO2021117861 A1 JP WO2021117861A1
Authority
JP
Japan
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2021564057A
Other languages
Japanese (ja)
Other versions
JP7093473B2 (ja
JPWO2021117861A5 (ko
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of JPWO2021117861A1 publication Critical patent/JPWO2021117861A1/ja
Publication of JPWO2021117861A5 publication Critical patent/JPWO2021117861A5/ja
Priority to JP2022097803A priority Critical patent/JP2022123069A/ja
Application granted granted Critical
Publication of JP7093473B2 publication Critical patent/JP7093473B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/32—Macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. carbomers, poly(meth)acrylates, or polyvinyl pyrrolidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38—Cellulose; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Inorganic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2021564057A 2019-12-13 2020-12-11 製造性及び溶出性に優れた小型錠剤 Active JP7093473B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2022097803A JP2022123069A (ja) 2019-12-13 2022-06-17 製造性及び溶出性に優れた小型錠剤

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2019225718 2019-12-13
JP2019225718 2019-12-13
PCT/JP2020/046253 WO2021117861A1 (ja) 2019-12-13 2020-12-11 製造性及び溶出性に優れた小型錠剤

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2022097803A Division JP2022123069A (ja) 2019-12-13 2022-06-17 製造性及び溶出性に優れた小型錠剤

Publications (3)

Publication Number Publication Date
JPWO2021117861A1 true JPWO2021117861A1 (ko) 2021-06-17
JPWO2021117861A5 JPWO2021117861A5 (ko) 2022-06-02
JP7093473B2 JP7093473B2 (ja) 2022-06-29

Family

ID=76330003

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2021564057A Active JP7093473B2 (ja) 2019-12-13 2020-12-11 製造性及び溶出性に優れた小型錠剤
JP2022097803A Pending JP2022123069A (ja) 2019-12-13 2022-06-17 製造性及び溶出性に優れた小型錠剤

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2022097803A Pending JP2022123069A (ja) 2019-12-13 2022-06-17 製造性及び溶出性に優れた小型錠剤

Country Status (5)

Country Link
JP (2) JP7093473B2 (ko)
KR (1) KR20220113942A (ko)
CN (1) CN114945370A (ko)
TW (1) TW202135826A (ko)
WO (1) WO2021117861A1 (ko)

Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2009523139A (ja) * 2006-01-13 2009-06-18 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング トリアジン誘導体およびインスリン分泌促進剤の組合せ
JP2009523141A (ja) * 2006-01-13 2009-06-18 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング トリアジン誘導体およびＨＭＧ−ＣｏＡレダクターゼ阻害剤の組合せ
JP2012511521A (ja) * 2008-12-12 2012-05-24 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング インスリンとトリアジンの組合せ及び糖尿病を治療するためのその使用
WO2014038593A2 (ja) * 2012-09-05 2014-03-13 テイカ製薬株式会社 口腔内速崩壊性錠剤用造粒物
JP2017141289A (ja) * 2012-01-06 2017-08-17 エルセリクス セラピューティクス インコーポレイテッド ビグアナイド組成物および代謝障害を治療する方法
WO2017170858A1 (ja) * 2016-03-31 2017-10-05 大日本住友製薬株式会社 溶出性に優れた経口製剤
JP2018154586A (ja) * 2017-03-17 2018-10-04 ライオン株式会社 錠剤

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI436768B (zh) 2010-06-09 2014-05-11 Poxel 第２型糖尿病之治療
CN112218623A (zh) * 2018-06-14 2021-01-12 博希尔公司 用于治疗糖尿病的包含三嗪衍生物的薄膜包衣片剂

Patent Citations (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2009523139A (ja) * 2006-01-13 2009-06-18 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング トリアジン誘導体およびインスリン分泌促進剤の組合せ
JP2009523141A (ja) * 2006-01-13 2009-06-18 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング トリアジン誘導体およびＨＭＧ−ＣｏＡレダクターゼ阻害剤の組合せ
JP2012511521A (ja) * 2008-12-12 2012-05-24 メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツング インスリンとトリアジンの組合せ及び糖尿病を治療するためのその使用
JP2017141289A (ja) * 2012-01-06 2017-08-17 エルセリクス セラピューティクス インコーポレイテッド ビグアナイド組成物および代謝障害を治療する方法
WO2014038593A2 (ja) * 2012-09-05 2014-03-13 テイカ製薬株式会社 口腔内速崩壊性錠剤用造粒物
WO2017170858A1 (ja) * 2016-03-31 2017-10-05 大日本住友製薬株式会社 溶出性に優れた経口製剤
JP2018154586A (ja) * 2017-03-17 2018-10-04 ライオン株式会社 錠剤

Also Published As

Publication number Publication date
WO2021117861A1 (ja) 2021-06-17
TW202135826A (zh) 2021-10-01
JP7093473B2 (ja) 2022-06-29
CN114945370A (zh) 2022-08-26
KR20220113942A (ko) 2022-08-17
JP2022123069A (ja) 2022-08-23

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