JPWO2021085636A1 - - Google Patents
Info
- Publication number
- JPWO2021085636A1 JPWO2021085636A1 JP2021553744A JP2021553744A JPWO2021085636A1 JP WO2021085636 A1 JPWO2021085636 A1 JP WO2021085636A1 JP 2021553744 A JP2021553744 A JP 2021553744A JP 2021553744 A JP2021553744 A JP 2021553744A JP WO2021085636 A1 JPWO2021085636 A1 JP WO2021085636A1
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/025—Silicon compounds without C-silicon linkages
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- B—PERFORMING OPERATIONS; TRANSPORTING
- B01—PHYSICAL OR CHEMICAL PROCESSES OR APPARATUS IN GENERAL
- B01J—CHEMICAL OR PHYSICAL PROCESSES, e.g. CATALYSIS OR COLLOID CHEMISTRY; THEIR RELEVANT APPARATUS
- B01J31/00—Catalysts comprising hydrides, coordination complexes or organic compounds
- B01J31/02—Catalysts comprising hydrides, coordination complexes or organic compounds containing organic compounds or metal hydrides
- B01J31/0272—Catalysts comprising hydrides, coordination complexes or organic compounds containing organic compounds or metal hydrides containing elements other than those covered by B01J31/0201 - B01J31/0255
- B01J31/0275—Catalysts comprising hydrides, coordination complexes or organic compounds containing organic compounds or metal hydrides containing elements other than those covered by B01J31/0201 - B01J31/0255 also containing elements or functional groups covered by B01J31/0201 - B01J31/0269
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C231/00—Preparation of carboxylic acid amides
- C07C231/02—Preparation of carboxylic acid amides from carboxylic acids or from esters, anhydrides, or halides thereof by reaction with ammonia or amines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D223/00—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom
- C07D223/02—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D223/06—Heterocyclic compounds containing seven-membered rings having one nitrogen atom as the only ring hetero atom not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D223/12—Nitrogen atoms not forming part of a nitro radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/08—Compounds having one or more C—Si linkages
- C07F7/10—Compounds having one or more C—Si linkages containing nitrogen having a Si-N linkage
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K1/00—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
- C07K1/06—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
- C07K1/08—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using activating agents
- C07K1/088—General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using activating agents containing other elements, e.g. B, Si, As
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
- C07F7/02—Silicon compounds
- C07F7/04—Esters of silicic acids
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biochemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Biophysics (AREA)
- General Health & Medical Sciences (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Molecular Biology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Health & Medical Sciences (AREA)
- Analytical Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Materials Engineering (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2019197786 | 2019-10-30 | ||
| JP2019197776 | 2019-10-30 | ||
| JP2019197776 | 2019-10-30 | ||
| JP2019197786 | 2019-10-30 | ||
| JP2020059087 | 2020-03-27 | ||
| JP2020059087 | 2020-03-27 | ||
| PCT/JP2020/040960 WO2021085636A1 (ja) | 2019-10-30 | 2020-10-30 | アミド反応用反応剤及びそれを用いたアミド化合物の製造方法 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2021085636A1 true JPWO2021085636A1 (https=) | 2021-05-06 |
| JPWO2021085636A5 JPWO2021085636A5 (https=) | 2022-07-28 |
| JP7244134B2 JP7244134B2 (ja) | 2023-03-22 |
Family
ID=75715278
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021553744A Active JP7244134B2 (ja) | 2019-10-30 | 2020-10-30 | アミド反応用反応剤及びそれを用いたアミド化合物の製造方法 |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US20230002422A1 (https=) |
| EP (2) | EP4053132A4 (https=) |
| JP (1) | JP7244134B2 (https=) |
| WO (1) | WO2021085636A1 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20240368217A1 (en) | 2021-05-31 | 2024-11-07 | Chubu University Educational Foundation | Peptide compound production method and amidation agent |
| EP4357353A4 (en) * | 2021-06-17 | 2025-05-07 | Chubu University Educational Foundation | METHOD FOR PREPARING A PEPTIDE COMPOUND |
| WO2022265115A1 (ja) | 2021-06-17 | 2022-12-22 | 学校法人中部大学 | ペプチド化合物の製造方法 |
| EP4446332A4 (en) | 2022-01-17 | 2025-04-16 | Chubu University Educational Foundation | METHOD FOR PREPARING A PEPTIDE COMPOUND |
| JP7674770B2 (ja) | 2022-04-27 | 2025-05-12 | 学校法人中部大学 | ポリペプチド化合物の製造方法 |
| US11878958B2 (en) | 2022-05-25 | 2024-01-23 | Ikena Oncology, Inc. | MEK inhibitors and uses thereof |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN110662736A (zh) | 2017-04-25 | 2020-01-07 | 学校法人中部大学 | 酰胺化合物的制造方法 |
| CN112020492B (zh) * | 2018-04-25 | 2023-05-05 | 学校法人中部大学 | 酰胺化合物的制造方法 |
-
2020
- 2020-10-30 JP JP2021553744A patent/JP7244134B2/ja active Active
- 2020-10-30 WO PCT/JP2020/040960 patent/WO2021085636A1/ja not_active Ceased
- 2020-10-30 US US17/772,500 patent/US20230002422A1/en active Pending
- 2020-10-30 EP EP20882761.8A patent/EP4053132A4/en active Pending
- 2020-10-30 EP EP25160777.6A patent/EP4538279A3/en active Pending
Non-Patent Citations (6)
| Title |
|---|
| MURAMATSU, WATARU ET AL.: "Peptide bond-forming reaction via amino acid silyl esters: New catalytic reactivity of an aminosilan", ACS CATALYSIS, JPN6020050377, 2020, pages 10 - 16, ISSN: 0004984097 * |
| MURAMATSU, WATARU ET AL.: "Substrate-Directed Lewis-Acid Catalysis for Peptide Synthesis", JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, vol. 141, no. 31, JPN6020050375, 16 July 2019 (2019-07-16), pages 12288 - 12295, XP055930667, ISSN: 0004984096, DOI: 10.1021/jacs.9b03850 * |
| SCHMIDT, MICHAEL A. ET AL.: "Development of a Two-Step, Enantioselective Synthesis of an Amino Alcohol Drug Candidate", ORGANIC PROCESS RESEARCH & DEVELOPMENT, vol. 19, no. 9, JPN6020050370, 2015, pages 1317 - 1322, XP055930641, ISSN: 0004882636, DOI: 10.1021/acs.oprd.5b00192 * |
| TOZAWA, TAKASHI ET AL.: "A convenient method for preparations of 1-acylimidazoles and carboxamides by using novel imidazolyls", CHEMISTRY LETTERS, vol. 34, no. 5, JPN6020050372, 2005, pages 734 - 735, XP055930635, ISSN: 0004984099, DOI: 10.1246/cl.2005.734 * |
| TOZAWA, TAKASHI ET AL.: "An efficient method for the preparation of carboxamides by dehydration condensation using tetrakis(1", CHEMISTRY LETTERS, vol. 34, no. 12, JPN6020050368, 2005, pages 1586 - 1587, XP055930633, ISSN: 0004984098 * |
| 第５版 実験化学講座 １６, JPN6020050373, 2005, pages 259 - 260, ISSN: 0004882635 * |
Also Published As
| Publication number | Publication date |
|---|---|
| EP4538279A2 (en) | 2025-04-16 |
| EP4053132A1 (en) | 2022-09-07 |
| JP7244134B2 (ja) | 2023-03-22 |
| EP4053132A4 (en) | 2024-02-21 |
| WO2021085636A1 (ja) | 2021-05-06 |
| US20230002422A1 (en) | 2023-01-05 |
| EP4538279A3 (en) | 2025-07-16 |
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