JPWO2019169153A5 - - Google Patents

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Publication number
JPWO2019169153A5
JPWO2019169153A5 JP2020545526A JP2020545526A JPWO2019169153A5 JP WO2019169153 A5 JPWO2019169153 A5 JP WO2019169153A5 JP 2020545526 A JP2020545526 A JP 2020545526A JP 2020545526 A JP2020545526 A JP 2020545526A JP WO2019169153 A5 JPWO2019169153 A5 JP WO2019169153A5
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JP
Japan
Prior art keywords
oxy
propanamide
dimethyl
pyridin
trifluoromethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2020545526A
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English (en)
Japanese (ja)
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JP2021515004A (ja
JP2021515004A5 (https=
JP7297776B2 (ja
Publication date
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Priority claimed from PCT/US2019/020086 external-priority patent/WO2019169153A1/en
Publication of JP2021515004A publication Critical patent/JP2021515004A/ja
Publication of JP2021515004A5 publication Critical patent/JP2021515004A5/ja
Publication of JPWO2019169153A5 publication Critical patent/JPWO2019169153A5/ja
Priority to JP2023098091A priority Critical patent/JP2023134444A/ja
Application granted granted Critical
Publication of JP7297776B2 publication Critical patent/JP7297776B2/ja
Priority to JP2025016827A priority patent/JP2025084759A/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2020545526A 2018-03-01 2019-02-28 ピペリジニル-3-(アリールオキシ)プロパンアミド及びプロパノエート Active JP7297776B2 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2023098091A JP2023134444A (ja) 2018-03-01 2023-06-14 ピペリジニル-3-(アリールオキシ)プロパンアミド及びプロパノエート
JP2025016827A JP2025084759A (ja) 2018-03-01 2025-02-04 ピペリジニル-3-(アリールオキシ)プロパンアミド及びプロパノエート

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862637295P 2018-03-01 2018-03-01
US62/637,295 2018-03-01
PCT/US2019/020086 WO2019169153A1 (en) 2018-03-01 2019-02-28 Piperidinyl-3-(aryloxy)propanamides and propanoates

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023098091A Division JP2023134444A (ja) 2018-03-01 2023-06-14 ピペリジニル-3-(アリールオキシ)プロパンアミド及びプロパノエート

Publications (4)

Publication Number Publication Date
JP2021515004A JP2021515004A (ja) 2021-06-17
JP2021515004A5 JP2021515004A5 (https=) 2022-03-10
JPWO2019169153A5 true JPWO2019169153A5 (https=) 2022-03-10
JP7297776B2 JP7297776B2 (ja) 2023-06-26

Family

ID=65763866

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2020545526A Active JP7297776B2 (ja) 2018-03-01 2019-02-28 ピペリジニル-3-(アリールオキシ)プロパンアミド及びプロパノエート
JP2023098091A Pending JP2023134444A (ja) 2018-03-01 2023-06-14 ピペリジニル-3-(アリールオキシ)プロパンアミド及びプロパノエート
JP2025016827A Pending JP2025084759A (ja) 2018-03-01 2025-02-04 ピペリジニル-3-(アリールオキシ)プロパンアミド及びプロパノエート

Family Applications After (2)

Application Number Title Priority Date Filing Date
JP2023098091A Pending JP2023134444A (ja) 2018-03-01 2023-06-14 ピペリジニル-3-(アリールオキシ)プロパンアミド及びプロパノエート
JP2025016827A Pending JP2025084759A (ja) 2018-03-01 2025-02-04 ピペリジニル-3-(アリールオキシ)プロパンアミド及びプロパノエート

Country Status (22)

Country Link
US (3) US11045457B2 (https=)
EP (1) EP3759094A1 (https=)
JP (3) JP7297776B2 (https=)
KR (2) KR20250094741A (https=)
CN (1) CN112236423B (https=)
AR (1) AR114421A1 (https=)
AU (1) AU2019228568B2 (https=)
BR (1) BR112020017644A2 (https=)
CA (1) CA3092450A1 (https=)
CL (1) CL2020002257A1 (https=)
EA (1) EA202092054A1 (https=)
EC (1) ECSP20062464A (https=)
IL (1) IL276998B2 (https=)
MX (1) MX2020009062A (https=)
MY (1) MY206763A (https=)
PE (1) PE20211313A1 (https=)
PH (1) PH12020551359A1 (https=)
SG (1) SG11202008398XA (https=)
TW (1) TWI834637B (https=)
UA (1) UA126829C2 (https=)
WO (1) WO2019169153A1 (https=)
ZA (1) ZA202005438B (https=)

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TWI834637B (zh) * 2018-03-01 2024-03-11 日商武田藥品工業有限公司 六氫吡啶基-3-(芳氧基)丙醯胺及丙酸酯
GB201901559D0 (en) * 2019-02-05 2019-03-27 Syngenta Crop Protection Ag Herbicidal compositions
CN114867720B (zh) 2020-01-16 2024-10-22 浙江海正药业股份有限公司 杂芳基类衍生物及其制备方法和用途
AR121682A1 (es) * 2020-03-31 2022-06-29 Takeda Pharmaceuticals Co Derivados de n-(heterociclil y heterociclilalquil)-3-bencilpiridin-2-amina como agonistas de sstr4
AR121683A1 (es) * 2020-03-31 2022-06-29 Takeda Pharmaceuticals Co Derivados de n-heteroarilalquil-2-(heterociclil y heterociclilmetil)acetamida como agonistas de sstr4
CN113717161B (zh) * 2020-05-21 2023-06-09 广州费米子科技有限责任公司 含氮饱和杂环化合物及其制备方法、药物组合物和应用
US20240217913A2 (en) * 2020-08-24 2024-07-04 Hua Medicine (Shanghai) Ltd. Preparation of substituted acrylate compound
US20240208923A1 (en) 2021-03-10 2024-06-27 Jnana Therapeutics Inc. Small molecule inhibitors of mammalian slc6a19 function
CN115477640A (zh) * 2021-05-31 2022-12-16 由理生物医药(上海)有限公司 作为parp7抑制剂的哒嗪酮类化合物
IL315998A (en) * 2022-03-30 2024-11-01 Takeda Pharmaceuticals Co N-(pyrrolidin-3-yl or piperidin-4-yl)acetamide derivatives
WO2025247982A1 (en) 2024-05-29 2025-12-04 Grünenthal GmbH Piperazines which act as sstr4 modulators

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KR0166088B1 (ko) 1990-01-23 1999-01-15 . 수용해도가 증가된 시클로덱스트린 유도체 및 이의 용도
US5376645A (en) 1990-01-23 1994-12-27 University Of Kansas Derivatives of cyclodextrins exhibiting enhanced aqueous solubility and the use thereof
GB9518953D0 (en) 1995-09-15 1995-11-15 Pfizer Ltd Pharmaceutical formulations
GB9711643D0 (en) 1997-06-05 1997-07-30 Janssen Pharmaceutica Nv Glass thermoplastic systems
SE9902987D0 (sv) 1999-08-24 1999-08-24 Astra Pharma Prod Novel compounds
CN1960970A (zh) * 2004-05-28 2007-05-09 田边制药株式会社 作为cb1受体的拮抗剂的吡咯烷衍生物
TW200602314A (en) 2004-05-28 2006-01-16 Tanabe Seiyaku Co A novel pyrrolidine compound and a process for preparing the same
US8258305B2 (en) 2005-02-23 2012-09-04 Prexa Pharmaceuticals, Inc. Dopamine transporter inhibitors for use in treatment of movement disorders and other CNS indications
EP1893603B1 (en) 2005-06-02 2009-10-14 F. Hoffmann-La Roche AG Piperidin-4-yl-amide derivatives and their use as sst receptor subtype 5 antagonists
JP4943826B2 (ja) * 2005-11-25 2012-05-30 田辺三菱製薬株式会社 医薬組成物
JP5736098B2 (ja) 2007-08-21 2015-06-17 アッヴィ・インコーポレイテッド 中枢神経系障害を治療するための医薬組成物
CA2718038A1 (en) 2008-03-14 2009-09-17 Exelixis, Inc. Azabicyclo [3.2.1] octyl derivatives as 11 beta-hsd1 modulators
WO2010059922A1 (en) 2008-11-21 2010-05-27 Ligand Pharmaceuticals Incorporated Pyrrolidine carboxamide compounds
CA2771568A1 (en) 2009-09-04 2011-03-10 Novartis Ag Heteroaryl compounds as kinase inhibitors
US9371282B2 (en) 2013-05-17 2016-06-21 Centrexion Therapeutics Corporation Somatostatin receptor subtype 4 (SSTR4) agonists
EP3045448A4 (en) * 2013-09-12 2017-01-25 Sumitomo Chemical Company Limited Nitrogen-containing saturated heterocyclic compound
CA2965566A1 (en) 2014-11-14 2016-05-19 Boehringer Ingelheim International Gmbh Morpholine and 1,4-oxazepane amides as somatostatin receptor subtype 4 (sstr4) agonists
WO2017003723A1 (en) * 2015-07-01 2017-01-05 Crinetics Pharmaceuticals, Inc. Somatostatin modulators and uses thereof
TWI834637B (zh) * 2018-03-01 2024-03-11 日商武田藥品工業有限公司 六氫吡啶基-3-(芳氧基)丙醯胺及丙酸酯

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