JPS632279B2 - - Google Patents

Info

Publication number
JPS632279B2
JPS632279B2 JP55126776A JP12677680A JPS632279B2 JP S632279 B2 JPS632279 B2 JP S632279B2 JP 55126776 A JP55126776 A JP 55126776A JP 12677680 A JP12677680 A JP 12677680A JP S632279 B2 JPS632279 B2 JP S632279B2
Authority
JP
Japan
Prior art keywords
group
alkoxybenzoyldeoxyfluorouridine
fluorouridine
deoxy
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP55126776A
Other languages
English (en)
Japanese (ja)
Other versions
JPS5751000A (en
Inventor
Setsuo Fujii
Bonpei Yasui
Mitsuo Nakamura
Mitsuru Hirohashi
Tomohisa Myamoto
Kazuko Ando
Iwao Hashimoto
Naoki Umeda
Masahiro Kawasaki
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Funai Pharmaceutical Industries Ltd
Original Assignee
Funai Pharmaceutical Industries Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Funai Pharmaceutical Industries Ltd filed Critical Funai Pharmaceutical Industries Ltd
Priority to JP55126776A priority Critical patent/JPS5751000A/ja
Priority to DE19813105111 priority patent/DE3105111A1/de
Priority to GB8104375A priority patent/GB2072164B/en
Priority to ES499443A priority patent/ES8206550A1/es
Priority to AT0069181A priority patent/AT374203B/de
Priority to IT8119758A priority patent/IT1210989B/it
Priority to CH96481A priority patent/CH646715A5/de
Priority to FR8102922A priority patent/FR2476086A1/fr
Priority to US06/291,809 priority patent/US4425335A/en
Priority to CA000383619A priority patent/CA1173437A/en
Priority to PH26042A priority patent/PH17365A/en
Publication of JPS5751000A publication Critical patent/JPS5751000A/ja
Publication of JPS632279B2 publication Critical patent/JPS632279B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/06—Pyrimidine radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
JP55126776A 1980-02-15 1980-09-11 Ester derivative of alkoxybenzoyldeoxyfluorouridine Granted JPS5751000A (en)

Priority Applications (11)

Application Number Priority Date Filing Date Title
JP55126776A JPS5751000A (en) 1980-09-11 1980-09-11 Ester derivative of alkoxybenzoyldeoxyfluorouridine
DE19813105111 DE3105111A1 (de) 1980-02-15 1981-02-12 "2 -desoxy-3',5-di-o-alkylcarbonyl-5-fluoruridin-derivate, verfahren zu ihrer herstellung, ihre verwendung zur behandlung von tumoren und antitumormittel"
GB8104375A GB2072164B (en) 1980-02-15 1981-02-12 2'-deoxy-3',5'-di-o-alkylcarbonyl-5-fluorouridine derivatives a process for the preparation of the derivatives and antitumor agents containing the derivatives
ES499443A ES8206550A1 (es) 1980-02-15 1981-02-13 Un procedimiento para la preparacion de derivados de 2-desoxi-3-5-di-o-alquilcarbonil-5-fluorurina.
AT0069181A AT374203B (de) 1980-02-15 1981-02-13 Verfahren zur herstellung von neuen 2'-desoxy-3', 5'-di-o-alkylcarbonyl-5-fluoruridinderivaten
IT8119758A IT1210989B (it) 1980-02-15 1981-02-13 Derivati 2'-deossi-3',5'-di-o-alchilcarbonil-5-fluorouri dinici processo per la loro preparazione e agenti antitumorali che contengono i detti derivati.
CH96481A CH646715A5 (de) 1980-02-15 1981-02-13 2'-desoxy-3',5'-di-o-alkylcarbonyl-5-fluoruridin-derivate, verfahren zu ihrer herstellung und antitumormittel.
FR8102922A FR2476086A1 (fr) 1980-02-15 1981-02-13 2'-desoxy-3',5'-di-o-alkylcarbonyl-5-fluoro-uridines, leur preparation et leur utilisation therapeutique en tant qu'agents anti-tumeurs
US06/291,809 US4425335A (en) 1980-09-11 1981-08-10 Ester derivatives of alkoxybenzoyldeoxyfluorouridine
CA000383619A CA1173437A (en) 1980-09-11 1981-08-11 Ester derivatives of alkoxybenzoyldeoxyfluorouridine
PH26042A PH17365A (en) 1980-09-11 1981-08-12 Ester derivatives of alkoxybenzolyldeoxy-fluorouridine,their process of preparation and composition containing them

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP55126776A JPS5751000A (en) 1980-09-11 1980-09-11 Ester derivative of alkoxybenzoyldeoxyfluorouridine

Publications (2)

Publication Number Publication Date
JPS5751000A JPS5751000A (en) 1982-03-25
JPS632279B2 true JPS632279B2 (en, 2012) 1988-01-18

Family

ID=14943642

Family Applications (1)

Application Number Title Priority Date Filing Date
JP55126776A Granted JPS5751000A (en) 1980-02-15 1980-09-11 Ester derivative of alkoxybenzoyldeoxyfluorouridine

Country Status (4)

Country Link
US (1) US4425335A (en, 2012)
JP (1) JPS5751000A (en, 2012)
CA (1) CA1173437A (en, 2012)
PH (1) PH17365A (en, 2012)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4864021A (en) * 1984-10-30 1989-09-05 Otsuka Pharmaceutical Co., Ltd. 5-fluorouracil derivatives
JPS61189292A (ja) * 1985-02-15 1986-08-22 Funai Corp ５−フルオロデオキシウリジン誘導体の新規な固溶体及びこれを活性成分として含有する制癌剤
US20050131224A1 (en) * 2003-12-15 2005-06-16 Cti Pet Systems, Inc. Method for preparing radiolabeled thymidine
US7160537B2 (en) * 2003-12-15 2007-01-09 Siemens Medical Solutions Usa, Inc. Method for preparing radiolabeled thymidine having low chromophoric byproducts

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3853845A (en) 1971-08-18 1974-12-10 Icn Pharmaceuticals 5-n-aminoacyl-5-aminouridines
JPS5924999B2 (ja) * 1978-06-10 1984-06-13 富山化学工業株式会社 新規な５−フルオロ−２′−デオキシ−β−ウリジン誘導体の製造法
JPS56115799A (en) * 1980-02-15 1981-09-11 Funai Corp 2'-deoxy-3',5'-di-o-alkylcarbonyl-5-fluorouridine derivative, its preparation, and antitumor agnet containing the same

Also Published As

Publication number Publication date
PH17365A (en) 1984-08-01
CA1173437A (en) 1984-08-28
US4425335A (en) 1984-01-10
JPS5751000A (en) 1982-03-25

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