JPS6121239B2 - - Google Patents

Info

Publication number
JPS6121239B2
JPS6121239B2 JP52155753A JP15575377A JPS6121239B2 JP S6121239 B2 JPS6121239 B2 JP S6121239B2 JP 52155753 A JP52155753 A JP 52155753A JP 15575377 A JP15575377 A JP 15575377A JP S6121239 B2 JPS6121239 B2 JP S6121239B2
Authority
JP
Japan
Prior art keywords
tert
mmol
phe
boc
asp
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP52155753A
Other languages
English (en)
Japanese (ja)
Other versions
JPS53111060A (en
Inventor
Kisufuarudei Rayosu
Shoon Isutoaan
Uaruroo Uintsue
Uaruga Raasuroo
Naafuraadei Yoozefu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
RIHITAA GEDEON BEGIESUZECHI GIARU AARU TEII
Original Assignee
RIHITAA GEDEON BEGIESUZECHI GIARU AARU TEII
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by RIHITAA GEDEON BEGIESUZECHI GIARU AARU TEII filed Critical RIHITAA GEDEON BEGIESUZECHI GIARU AARU TEII
Publication of JPS53111060A publication Critical patent/JPS53111060A/ja
Publication of JPS6121239B2 publication Critical patent/JPS6121239B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/36—Oxygen or sulfur atoms
    • C07D207/40—2,5-Pyrrolidine-diones
    • C07D207/404—2,5-Pyrrolidine-diones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms, e.g. succinimide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C291/00—Compounds containing carbon and nitrogen and having functional groups not covered by groups C07C201/00 - C07C281/00
    • C07C291/02—Compounds containing carbon and nitrogen and having functional groups not covered by groups C07C201/00 - C07C281/00 containing nitrogen-oxide bonds
    • C07C291/04—Compounds containing carbon and nitrogen and having functional groups not covered by groups C07C201/00 - C07C281/00 containing nitrogen-oxide bonds containing amino-oxide bonds
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C53/00—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
    • C07C53/15—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen containing halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1024—Tetrapeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP15575377A 1976-12-30 1977-12-26 Alphaaaminoxyacyl grouppcontaining peptide Granted JPS53111060A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU76RI608A HU175152B (hu) 1976-12-30 1976-12-30 Sposob poluchenija peptidov s gastrin-aktivnost'ju, soderzhahhikh amino-oksi-kisloty

Publications (2)

Publication Number Publication Date
JPS53111060A JPS53111060A (en) 1978-09-28
JPS6121239B2 true JPS6121239B2 (oth) 1986-05-26

Family

ID=11001012

Family Applications (1)

Application Number Title Priority Date Filing Date
JP15575377A Granted JPS53111060A (en) 1976-12-30 1977-12-26 Alphaaaminoxyacyl grouppcontaining peptide

Country Status (10)

Country Link
US (1) US4172130A (oth)
JP (1) JPS53111060A (oth)
BE (1) BE862406A (oth)
DE (1) DE2759031A1 (oth)
FR (1) FR2376127A1 (oth)
GB (1) GB1541337A (oth)
HU (1) HU175152B (oth)
NL (1) NL7714582A (oth)
SE (1) SE441752B (oth)
SU (1) SU691082A3 (oth)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5815946A (ja) * 1981-07-21 1983-01-29 Eisai Co Ltd 新規ヘプタデカペプタイド
CH664560A5 (fr) * 1982-07-07 1988-03-15 Orgamol Sa Procede de preparation d'un ester dipeptide d'acide l-aspartique par deblocage reducteur.
FR2575164B1 (fr) * 1984-12-20 1987-03-20 Sanofi Sa Esters de tri- et tetrapeptides inhibiteurs de la secretion gastrique, procede d'obtention et compositions pharmaceutiques les contenant
CN101970015B (zh) * 2008-01-08 2014-05-07 兰休斯医疗成像公司 作为显像剂的n-烷氧基酰胺共轭物
CN113929737B (zh) * 2021-10-20 2024-07-23 中国科学院香港创新研究院再生医学与健康创新中心 一种多肽及其作为cck受体激动剂/拮抗剂的应用

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1042487A (en) * 1964-06-25 1966-09-14 Ici Ltd Polypeptide derivatives
HU167655B (oth) * 1972-08-18 1975-11-28

Also Published As

Publication number Publication date
FR2376127B1 (oth) 1980-04-04
SE7714524L (sv) 1978-07-01
SE441752B (sv) 1985-11-04
JPS53111060A (en) 1978-09-28
BE862406A (fr) 1978-04-14
US4172130A (en) 1979-10-23
SU691082A3 (ru) 1979-10-05
NL7714582A (nl) 1978-07-04
DE2759031C2 (oth) 1988-07-21
GB1541337A (en) 1979-02-28
FR2376127A1 (fr) 1978-07-28
HU175152B (hu) 1980-05-28
DE2759031A1 (de) 1978-07-13

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