JPS572277A - Quinoxalinone derivative, its preparation, and fungicide for agricultural and horticultural use - Google Patents
Quinoxalinone derivative, its preparation, and fungicide for agricultural and horticultural useInfo
- Publication number
- JPS572277A JPS572277A JP7683480A JP7683480A JPS572277A JP S572277 A JPS572277 A JP S572277A JP 7683480 A JP7683480 A JP 7683480A JP 7683480 A JP7683480 A JP 7683480A JP S572277 A JPS572277 A JP S572277A
- Authority
- JP
- Japan
- Prior art keywords
- compound
- formula
- fungicide
- agricultural
- horticultural use
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Abstract
NEW MATERIAL:A compound of formula I (X is halogen or lower alkyl; R is lower alkyl; n is an integer of 1W4).
EXAMPLE: 7-Bromo-1-methyl-2(1H)-quinoxalinone.
USE: Fungicide for agricultural and horticultural use, having remarkable effect to rice blast by the application to the water surface of the paddy rice field. It exhibits prolonged activity.
PROCESS: The compound of formula I is prepared by the lower-alkylation of the 1- position N-atom of the compound of formula II represented as a tautomer. The lower-alkylation can be carried out, e.g. by mixing the starting compound with an alkylating agent such as an alkylsulfuric acid ester, an alkyl halide, etc., in a solvent such as benzene, ether, etc., in the presence of a base (e.g. sodium ethoxide, sodium hydride, etc.) or in an alcohol in the presence of a base (e.g. sodium ethoxide, sodium hydroxide, etc.) at 0W150°C for 0.5W15hr.
COPYRIGHT: (C)1982,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP7683480A JPS572277A (en) | 1980-06-07 | 1980-06-07 | Quinoxalinone derivative, its preparation, and fungicide for agricultural and horticultural use |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP7683480A JPS572277A (en) | 1980-06-07 | 1980-06-07 | Quinoxalinone derivative, its preparation, and fungicide for agricultural and horticultural use |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS572277A true JPS572277A (en) | 1982-01-07 |
Family
ID=13616700
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP7683480A Pending JPS572277A (en) | 1980-06-07 | 1980-06-07 | Quinoxalinone derivative, its preparation, and fungicide for agricultural and horticultural use |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS572277A (en) |
Cited By (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5198441A (en) * | 1989-10-23 | 1993-03-30 | Pierre Fabre Medicament | Derivatives of 1,2-dihydro 2-oxo quinoxalines, their preparation and their use in therapy |
JP2002338552A (en) * | 2001-05-15 | 2002-11-27 | Takeda Chem Ind Ltd | Quinoxaline-based compound and industrial germicidal composition |
CN111423388A (en) * | 2020-04-29 | 2020-07-17 | 浙江工业大学 | 7-methoxy-3-phenylquinoxaline-2 (1H) -one derivative and preparation method and application thereof |
-
1980
- 1980-06-07 JP JP7683480A patent/JPS572277A/en active Pending
Cited By (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5198441A (en) * | 1989-10-23 | 1993-03-30 | Pierre Fabre Medicament | Derivatives of 1,2-dihydro 2-oxo quinoxalines, their preparation and their use in therapy |
JP2002338552A (en) * | 2001-05-15 | 2002-11-27 | Takeda Chem Ind Ltd | Quinoxaline-based compound and industrial germicidal composition |
JP4707261B2 (en) * | 2001-05-15 | 2011-06-22 | 日本エンバイロケミカルズ株式会社 | Quinoxaline compound and industrial bactericidal composition |
CN111423388A (en) * | 2020-04-29 | 2020-07-17 | 浙江工业大学 | 7-methoxy-3-phenylquinoxaline-2 (1H) -one derivative and preparation method and application thereof |
CN111423388B (en) * | 2020-04-29 | 2022-02-15 | 浙江工业大学 | 7-methoxy-3-phenylquinoxaline-2 (1H) -one derivative and preparation method and application thereof |
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