JPS5659781A - Penicillins - Google Patents

Penicillins

Info

Publication number
JPS5659781A
JPS5659781A JP13823280A JP13823280A JPS5659781A JP S5659781 A JPS5659781 A JP S5659781A JP 13823280 A JP13823280 A JP 13823280A JP 13823280 A JP13823280 A JP 13823280A JP S5659781 A JPS5659781 A JP S5659781A
Authority
JP
Japan
Prior art keywords
penicillins
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP13823280A
Other languages
English (en)
Inventor
Piitaa Kureiton Jiyon
Kooru Maachin
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Beecham Group PLC
Original Assignee
Beecham Group PLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Beecham Group PLC filed Critical Beecham Group PLC
Publication of JPS5659781A publication Critical patent/JPS5659781A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C07D499/72—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by carbon atoms having three bonds to hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/429—Thiazoles condensed with heterocyclic ring systems
    • A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/76—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with hetero rings directly attached to the carboxamido radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP13823280A 1979-10-02 1980-10-02 Penicillins Pending JPS5659781A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7934062 1979-10-02

Publications (1)

Publication Number Publication Date
JPS5659781A true JPS5659781A (en) 1981-05-23

Family

ID=10508217

Family Applications (1)

Application Number Title Priority Date Filing Date
JP13823280A Pending JPS5659781A (en) 1979-10-02 1980-10-02 Penicillins

Country Status (25)

Country Link
US (1) US4385060A (ja)
EP (1) EP0026644B1 (ja)
JP (1) JPS5659781A (ja)
KR (1) KR850000474B1 (ja)
AR (1) AR227953A1 (ja)
AU (1) AU534572B2 (ja)
CA (1) CA1148941A (ja)
DE (1) DE3061229D1 (ja)
DK (1) DK415780A (ja)
ES (1) ES495554A0 (ja)
FI (1) FI803015A (ja)
GR (1) GR70283B (ja)
HK (1) HK786A (ja)
HU (1) HU182676B (ja)
IE (1) IE50508B1 (ja)
IL (1) IL61031A0 (ja)
MY (1) MY8600395A (ja)
NO (1) NO802910L (ja)
NZ (1) NZ194912A (ja)
PH (1) PH17119A (ja)
PL (3) PL129141B1 (ja)
PT (1) PT71856B (ja)
SG (1) SG72685G (ja)
YU (2) YU249080A (ja)
ZA (1) ZA805665B (ja)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL67672A0 (en) * 1982-01-22 1983-05-15 Beecham Group Plc Penicillin derivatives,their preparation and pharmaceutical compositions containing them
WO2001066089A2 (en) 2000-03-09 2001-09-13 Gw Pharma Limited Pharmaceutical compositions comprising cannabis

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3853849A (en) * 1969-05-29 1974-12-10 Beecham Group Ltd Alpha(aryloxycarbonyl)-and alpha(alkoxy-carbonyl)-aralkyl penicillins
GB1229670A (ja) 1968-09-03 1971-04-28
BE759795A (fr) 1969-12-11 1971-06-03 Pfizer Synthese de penicillines par l'intermediaire d'anhydrides mixtes de l'acide sulfurique
US4171303A (en) * 1974-07-30 1979-10-16 Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. Process for the preparation of reactive penicillanic acid and cephalosporanic acid derivatives
GB1455529A (ja) 1975-02-27 1976-11-10
JO984B1 (en) 1977-10-11 1979-12-01 بيتشام غروب ليمتد A dry pharmaceutical compound with a suitable dosage unit for oral administration

Also Published As

Publication number Publication date
ZA805665B (en) 1981-09-30
IE50508B1 (en) 1986-04-30
HU182676B (en) 1984-02-28
PT71856A (en) 1980-10-01
PL129153B1 (en) 1984-04-30
ES8106733A1 (es) 1981-09-01
NZ194912A (en) 1983-05-31
PL227022A1 (ja) 1981-12-11
AU534572B2 (en) 1984-02-09
KR830003498A (ko) 1983-06-21
PL232294A1 (ja) 1982-03-29
PL232295A1 (ja) 1982-03-29
ES495554A0 (es) 1981-09-01
DK415780A (da) 1981-04-03
FI803015A (fi) 1981-04-03
PT71856B (en) 1981-07-09
YU249080A (en) 1983-06-30
PH17119A (en) 1984-06-01
SG72685G (en) 1986-05-02
US4385060A (en) 1983-05-24
PL129141B1 (en) 1984-04-30
YU45883A (en) 1983-12-31
KR850000474B1 (ko) 1985-04-08
HK786A (en) 1986-01-10
IL61031A0 (en) 1980-11-30
GR70283B (ja) 1982-09-03
EP0026644A1 (en) 1981-04-08
CA1148941A (en) 1983-06-28
IE802045L (en) 1981-04-02
AR227953A1 (es) 1982-12-30
EP0026644B1 (en) 1982-12-01
AU6283080A (en) 1981-04-09
DE3061229D1 (en) 1983-01-05
MY8600395A (en) 1986-12-31
NO802910L (no) 1981-04-03

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