HK786A - Ortho-tolyl ester of an alpha-carboxy penicillin,process for its preparation and pharmaceutical compositions comprising the penicillin - Google Patents
Ortho-tolyl ester of an alpha-carboxy penicillin,process for its preparation and pharmaceutical compositions comprising the penicillinInfo
- Publication number
- HK786A HK786A HK7/86A HK786A HK786A HK 786 A HK786 A HK 786A HK 7/86 A HK7/86 A HK 7/86A HK 786 A HK786 A HK 786A HK 786 A HK786 A HK 786A
- Authority
- HK
- Hong Kong
- Prior art keywords
- penicillin
- ortho
- alpha
- preparation
- pharmaceutical compositions
- Prior art date
Links
- 229930182555 Penicillin Natural products 0.000 title 2
- 229940049954 penicillin Drugs 0.000 title 2
- -1 Ortho-tolyl ester Chemical class 0.000 title 1
- JGSARLDLIJGVTE-MBNYWOFBSA-N Penicillin G Chemical compound N([C@H]1[C@H]2SC([C@@H](N2C1=O)C(O)=O)(C)C)C(=O)CC1=CC=CC=C1 JGSARLDLIJGVTE-MBNYWOFBSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
- C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
- C07D499/72—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by carbon atoms having three bonds to hetero atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/425—Thiazoles
- A61K31/429—Thiazoles condensed with heterocyclic ring systems
- A61K31/43—Compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula, e.g. penicillins, penems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
- C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/76—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with hetero rings directly attached to the carboxamido radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Oncology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB7934062 | 1979-10-02 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| HK786A true HK786A (en) | 1986-01-10 |
Family
ID=10508217
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HK7/86A HK786A (en) | 1979-10-02 | 1986-01-02 | Ortho-tolyl ester of an alpha-carboxy penicillin,process for its preparation and pharmaceutical compositions comprising the penicillin |
Country Status (25)
| Country | Link |
|---|---|
| US (1) | US4385060A (en) |
| EP (1) | EP0026644B1 (en) |
| JP (1) | JPS5659781A (en) |
| KR (1) | KR850000474B1 (en) |
| AR (1) | AR227953A1 (en) |
| AU (1) | AU534572B2 (en) |
| CA (1) | CA1148941A (en) |
| DE (1) | DE3061229D1 (en) |
| DK (1) | DK415780A (en) |
| ES (1) | ES495554A0 (en) |
| FI (1) | FI803015A (en) |
| GR (1) | GR70283B (en) |
| HK (1) | HK786A (en) |
| HU (1) | HU182676B (en) |
| IE (1) | IE50508B1 (en) |
| IL (1) | IL61031A0 (en) |
| MY (1) | MY8600395A (en) |
| NO (1) | NO802910L (en) |
| NZ (1) | NZ194912A (en) |
| PH (1) | PH17119A (en) |
| PL (3) | PL129141B1 (en) |
| PT (1) | PT71856B (en) |
| SG (1) | SG72685G (en) |
| YU (2) | YU249080A (en) |
| ZA (1) | ZA805665B (en) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL67672A0 (en) * | 1982-01-22 | 1983-05-15 | Beecham Group Plc | Penicillin derivatives,their preparation and pharmaceutical compositions containing them |
| WO2001066089A2 (en) | 2000-03-09 | 2001-09-13 | Gw Pharma Limited | Pharmaceutical compositions comprising cannabis |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3853849A (en) * | 1969-05-29 | 1974-12-10 | Beecham Group Ltd | Alpha(aryloxycarbonyl)-and alpha(alkoxy-carbonyl)-aralkyl penicillins |
| GB1229670A (en) | 1968-09-03 | 1971-04-28 | ||
| BE759795A (en) | 1969-12-11 | 1971-06-03 | Pfizer | SYNTHESIS OF PENICILLINS BY INTERMEDIATE OF MIXED ANHYDRIDES OF SULFURIC ACID |
| US4171303A (en) * | 1974-07-30 | 1979-10-16 | Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. | Process for the preparation of reactive penicillanic acid and cephalosporanic acid derivatives |
| GB1455529A (en) | 1975-02-27 | 1976-11-10 | ||
| JO984B1 (en) | 1977-10-11 | 1979-12-01 | بيتشام غروب ليمتد | K-clavulanate/tri hydrate formulations |
-
1980
- 1980-09-10 GR GR62854A patent/GR70283B/el unknown
- 1980-09-10 NZ NZ194912A patent/NZ194912A/en unknown
- 1980-09-12 ZA ZA00805665A patent/ZA805665B/en unknown
- 1980-09-14 IL IL61031A patent/IL61031A0/en unknown
- 1980-09-22 US US06/189,622 patent/US4385060A/en not_active Expired - Lifetime
- 1980-09-25 FI FI803015A patent/FI803015A/en not_active Application Discontinuation
- 1980-09-26 DE DE8080303378T patent/DE3061229D1/en not_active Expired
- 1980-09-26 EP EP80303378A patent/EP0026644B1/en not_active Expired
- 1980-09-30 YU YU02490/80A patent/YU249080A/en unknown
- 1980-09-30 KR KR1019800003787A patent/KR850000474B1/en active IP Right Grant
- 1980-09-30 PT PT71856A patent/PT71856B/en unknown
- 1980-09-30 AU AU62830/80A patent/AU534572B2/en not_active Ceased
- 1980-10-01 PL PL1980232295A patent/PL129141B1/en unknown
- 1980-10-01 DK DK415780A patent/DK415780A/en unknown
- 1980-10-01 PL PL1980227022A patent/PL129153B1/en unknown
- 1980-10-01 IE IE2045/80A patent/IE50508B1/en unknown
- 1980-10-01 ES ES495554A patent/ES495554A0/en active Granted
- 1980-10-01 PL PL23229480A patent/PL232294A1/xx unknown
- 1980-10-01 NO NO802910A patent/NO802910L/en unknown
- 1980-10-01 CA CA000361314A patent/CA1148941A/en not_active Expired
- 1980-10-01 HU HU802394A patent/HU182676B/en unknown
- 1980-10-02 JP JP13823280A patent/JPS5659781A/en active Pending
- 1980-10-02 PH PH24658A patent/PH17119A/en unknown
-
1981
- 1981-12-21 AR AR287880A patent/AR227953A1/en active
-
1983
- 1983-02-25 YU YU00458/83A patent/YU45883A/en unknown
-
1985
- 1985-10-05 SG SG726/85A patent/SG72685G/en unknown
-
1986
- 1986-01-02 HK HK7/86A patent/HK786A/en unknown
- 1986-12-30 MY MY395/86A patent/MY8600395A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA805665B (en) | 1981-09-30 |
| IE50508B1 (en) | 1986-04-30 |
| HU182676B (en) | 1984-02-28 |
| PT71856A (en) | 1980-10-01 |
| PL129153B1 (en) | 1984-04-30 |
| ES8106733A1 (en) | 1981-09-01 |
| NZ194912A (en) | 1983-05-31 |
| PL227022A1 (en) | 1981-12-11 |
| AU534572B2 (en) | 1984-02-09 |
| KR830003498A (en) | 1983-06-21 |
| PL232294A1 (en) | 1982-03-29 |
| PL232295A1 (en) | 1982-03-29 |
| ES495554A0 (en) | 1981-09-01 |
| DK415780A (en) | 1981-04-03 |
| FI803015A (en) | 1981-04-03 |
| PT71856B (en) | 1981-07-09 |
| YU249080A (en) | 1983-06-30 |
| PH17119A (en) | 1984-06-01 |
| SG72685G (en) | 1986-05-02 |
| US4385060A (en) | 1983-05-24 |
| PL129141B1 (en) | 1984-04-30 |
| YU45883A (en) | 1983-12-31 |
| KR850000474B1 (en) | 1985-04-08 |
| IL61031A0 (en) | 1980-11-30 |
| GR70283B (en) | 1982-09-03 |
| EP0026644A1 (en) | 1981-04-08 |
| CA1148941A (en) | 1983-06-28 |
| IE802045L (en) | 1981-04-02 |
| AR227953A1 (en) | 1982-12-30 |
| EP0026644B1 (en) | 1982-12-01 |
| AU6283080A (en) | 1981-04-09 |
| DE3061229D1 (en) | 1983-01-05 |
| MY8600395A (en) | 1986-12-31 |
| NO802910L (en) | 1981-04-03 |
| JPS5659781A (en) | 1981-05-23 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IL59914A (en) | Esters of acyl-carnitines,process for their preparation and pharmaceutical compositions containing them | |
| GB2050828B (en) | Process for the preparations of finely divided pharmaceutical compositions | |
| MY8500046A (en) | N-heterocyclyl-4-piperidinamines, methods for their preparation, pharmaceutical compositions comprising them, intermediates thereof, and methods for the preparation of the intermediates | |
| PT71676B (en) | Process for the preparation of new derivatives of 1h-indolhaving pharmaceutical properties | |
| GB2043644B (en) | 3-phosphonocephalosporanic acid derivatives process for preparation thereof and pharmaceutical composition comprising the same | |
| AU542902B2 (en) | Substituted carboxylic ceto-acids, process for the preparation thereof, use thereof and medicinal compositions containing them | |
| DE2861461D1 (en) | Derivatives of aminobenzoic acids, process for their preparation and pharmaceutical compositions containing them. | |
| DE3061438D1 (en) | Quinoline compounds, process for their preparation, and pharmaceutical compositions | |
| ZA792043B (en) | Esters of substituted 8-hydroxy-1-phenyl-2,3,4,5-tetrahydro-1h-3-benzazepines,process for the preparation thereof and pharmaceutical compositions containing them | |
| DE3061152D1 (en) | Pyrazoloindazole derivatives and process for preparing the same and pharmaceutical compositions | |
| GB2050833B (en) | Pharmaceutical compositions and process for the preparation thereof | |
| PT72066A (en) | Process for the preparation of novel halophenyl-pyridil-allylamine derivatives and pharmaceutical compositions thereof | |
| AU533471B2 (en) | Pharmaceutical composition comprising modified polyriboinosinic-polyribocytidylic acid | |
| IL60907A0 (en) | Substituted quinoline-alkanecarboxylic acids,process for their preparation and pharmaceutical compositions containing them | |
| PT72237B (en) | Process for the preparation of new pyrrolbenzotriazepines having pharmaceutical effect | |
| DE3061471D1 (en) | Process for the preparation of beta-alkoxy-acrylonitriles, 3-amino-acrylonitriles and 2-cyano-vinyl esters | |
| DE3061229D1 (en) | Ortho-tolyl ester of an alpha-carboxy penicillin, process for its preparation and pharmaceutical compositions comprising the penicillin | |
| DE2967215D1 (en) | Isoquinoline derivatives, process for their preparation, intermediates and pharmaceutical compositions containing them | |
| IL60604A (en) | 4-fluoro-3-bromo-benzoyl-fluoride,its preparation and its use for the preparation of the alpha-cyano-4-fluoro-3-phenoxybenzyl ester of permethric acid | |
| DE3062572D1 (en) | Penicillin derivatives, process for their preparation and pharmaceutical composition comprising them | |
| DE2861051D1 (en) | Oxaminic acids and esters, process for their preparation and pharmaceutical compositions containing them | |
| KE3568A (en) | Ortho-tolyl ester of an alpha-carboxy penicillin,process for its preparation and pharmaceutical compositions comprising the penicillin | |
| GB2004885B (en) | Indolopyrones process for the preparation thereof and pharmaceutical compositions containing them | |
| IL54585A (en) | 5-sulfamoyl-orthanilic acids,process for their preparation and pharmaceutical compositions containing them | |
| ZA794631B (en) | New 1-methyl-4-piperidinol esters,process for their preparation and pharmaceutical compositions containing them |