JPS56131575A - Locally available s-(-)-1-(tertiary-butylamino)- 3-((4-morpholino-1,2,5-thiadiazole-3-yl)-oxy)-2- propanolpamoate for treatment of intraocular pressure rise - Google Patents

Locally available s-(-)-1-(tertiary-butylamino)- 3-((4-morpholino-1,2,5-thiadiazole-3-yl)-oxy)-2- propanolpamoate for treatment of intraocular pressure rise

Info

Publication number
JPS56131575A
JPS56131575A JP2229981A JP2229981A JPS56131575A JP S56131575 A JPS56131575 A JP S56131575A JP 2229981 A JP2229981 A JP 2229981A JP 2229981 A JP2229981 A JP 2229981A JP S56131575 A JPS56131575 A JP S56131575A
Authority
JP
Japan
Prior art keywords
butylamino
morpholino
oxy
treatment
intraocular pressure
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2229981A
Other languages
English (en)
Japanese (ja)
Inventor
Daburiyu Henrii Maachin
Jiee Haautsudo Richiyaado
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck and Co Inc
Original Assignee
Merck and Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck and Co Inc filed Critical Merck and Co Inc
Publication of JPS56131575A publication Critical patent/JPS56131575A/ja
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/10—1,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Ophthalmology & Optometry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Cephalosporin Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
JP2229981A 1980-02-19 1981-02-19 Locally available s-(-)-1-(tertiary-butylamino)- 3-((4-morpholino-1,2,5-thiadiazole-3-yl)-oxy)-2- propanolpamoate for treatment of intraocular pressure rise Pending JPS56131575A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US12233880A 1980-02-19 1980-02-19

Publications (1)

Publication Number Publication Date
JPS56131575A true JPS56131575A (en) 1981-10-15

Family

ID=22402132

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2229981A Pending JPS56131575A (en) 1980-02-19 1981-02-19 Locally available s-(-)-1-(tertiary-butylamino)- 3-((4-morpholino-1,2,5-thiadiazole-3-yl)-oxy)-2- propanolpamoate for treatment of intraocular pressure rise

Country Status (11)

Country Link
EP (1) EP0034542B1 (enExample)
JP (1) JPS56131575A (enExample)
AT (1) ATE15193T1 (enExample)
AU (1) AU540656B2 (enExample)
DE (1) DE3171965D1 (enExample)
DK (1) DK70981A (enExample)
ES (1) ES499570A0 (enExample)
GR (1) GR74105B (enExample)
IE (1) IE50923B1 (enExample)
NZ (1) NZ196227A (enExample)
PT (1) PT72515B (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2106852T3 (es) * 1992-07-08 1997-11-16 Santen Oy Composicion oftalmica que contiene hemihidrato de timolol.

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3657237A (en) * 1968-05-22 1972-04-18 Frosst & Co Charles E Process for making 1 2 5-thiadiazoles in the sinister configuration
GB1253709A (en) * 1968-05-22 1971-11-17 Frosst & Co Charles E Thiadiazole derivatives
US3833727A (en) * 1972-03-06 1974-09-03 Merck & Co Inc Hydralazine and beta-adrenergic blocking agent compositions for treating hypertension
GB1429420A (en) * 1974-06-05 1976-03-24 Merck Sharp & Dohme Thiadiazole derivatives
DE2428030A1 (de) * 1974-06-11 1976-01-02 Merck Sharp & Dohme Substituierte thiadiazole und verfahren zu ihrer herstellung
CH597209A5 (en) * 1974-06-18 1978-03-31 Merck Sharp & Dohme 4-(3-Amino-2-acyloxypropoxyl)-1,2,5-thiadiazoles
FR2277581A1 (fr) * 1974-07-09 1976-02-06 Merck Sharp & Dohme Thiadiazoles substitues et procede pour leur preparation

Also Published As

Publication number Publication date
AU6713181A (en) 1981-08-27
ES8205795A1 (es) 1982-07-01
EP0034542A2 (en) 1981-08-26
AU540656B2 (en) 1984-11-29
EP0034542B1 (en) 1985-08-28
ES499570A0 (es) 1982-07-01
EP0034542A3 (en) 1981-10-21
GR74105B (enExample) 1984-06-06
NZ196227A (en) 1984-09-28
PT72515B (en) 1982-12-20
IE50923B1 (en) 1986-08-20
DE3171965D1 (en) 1985-10-03
DK70981A (da) 1981-08-20
PT72515A (en) 1981-03-01
ATE15193T1 (de) 1985-09-15
IE810310L (en) 1981-08-19

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