FR2277581A1 - Thiadiazoles substitues et procede pour leur preparation - Google Patents

Thiadiazoles substitues et procede pour leur preparation

Info

Publication number
FR2277581A1
FR2277581A1 FR7423783A FR7423783A FR2277581A1 FR 2277581 A1 FR2277581 A1 FR 2277581A1 FR 7423783 A FR7423783 A FR 7423783A FR 7423783 A FR7423783 A FR 7423783A FR 2277581 A1 FR2277581 A1 FR 2277581A1
Authority
FR
France
Prior art keywords
useful
morpholino
beta
adrenergic blocking
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7423783A
Other languages
English (en)
Other versions
FR2277581B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Merck Sharp and Dohme IA Corp
Merck Sharp and Dohme Corp
Original Assignee
Merck Sharp and Dohme IA Corp
Merck Sharp and Dohme Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp and Dohme IA Corp, Merck Sharp and Dohme Corp filed Critical Merck Sharp and Dohme IA Corp
Priority to FR7423783A priority Critical patent/FR2277581A1/fr
Publication of FR2277581A1 publication Critical patent/FR2277581A1/fr
Application granted granted Critical
Publication of FR2277581B1 publication Critical patent/FR2277581B1/fr
Granted legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D285/00Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01Five-membered rings
    • C07D285/02Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/101,2,5-Thiadiazoles; Hydrogenated 1,2,5-thiadiazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
FR7423783A 1974-07-09 1974-07-09 Thiadiazoles substitues et procede pour leur preparation Granted FR2277581A1 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
FR7423783A FR2277581A1 (fr) 1974-07-09 1974-07-09 Thiadiazoles substitues et procede pour leur preparation

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7423783A FR2277581A1 (fr) 1974-07-09 1974-07-09 Thiadiazoles substitues et procede pour leur preparation

Publications (2)

Publication Number Publication Date
FR2277581A1 true FR2277581A1 (fr) 1976-02-06
FR2277581B1 FR2277581B1 (fr) 1978-07-21

Family

ID=9141052

Family Applications (1)

Application Number Title Priority Date Filing Date
FR7423783A Granted FR2277581A1 (fr) 1974-07-09 1974-07-09 Thiadiazoles substitues et procede pour leur preparation

Country Status (1)

Country Link
FR (1) FR2277581A1 (fr)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0034542A2 (fr) * 1980-02-19 1981-08-26 Merck & Co. Inc. Pamoate de S-(-)-1-(tert-butylamino)-3-((4-morpholino-1,2,5-thiadiazol-3-yl)-oxy)-2-propanol pour application locale dans le traitement de pression intraoculaire élevée

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0034542A2 (fr) * 1980-02-19 1981-08-26 Merck & Co. Inc. Pamoate de S-(-)-1-(tert-butylamino)-3-((4-morpholino-1,2,5-thiadiazol-3-yl)-oxy)-2-propanol pour application locale dans le traitement de pression intraoculaire élevée
EP0034542A3 (en) * 1980-02-19 1981-10-21 Merck & Co. Inc. S-(-)-1-(tert-butylamino)-3-((4-morpholino-1,2,5-thiadiazol-3-yl)-oxy)-2-propanol pamoate for topical application in the treatment of elevated intraocular pressure

Also Published As

Publication number Publication date
FR2277581B1 (fr) 1978-07-21

Similar Documents

Publication Publication Date Title
DK0652001T3 (da) Fremgangsmåder til behandling af det perimenopausale syndrom
FI923494A (fi) Peptidylderivat.
BG105271A (en) 1h-imidazopyridine derivatives
ES2183439T3 (es) Mezclas fungicidas a base de piridinamidas y clorotalonil.
ES2070151T3 (es) Agentes cardiotonicos.
TW375615B (en) Galanthamine derivatives and their use as medicaments
ZA915366B (en) Diphenylmethyl piperazine derivatives
ATE37869T1 (de) Benzoylharnstoffderivate und diese verbindungen enthaltende pestizide kompositionen.
ES438931A1 (es) Procedimiento para la preparacion de nuevos derivados de amino-3 hidroxi-2 fenoxi-1 propano.
GB1236735A (en) Fungicidal agents and methods
FR2277581A1 (fr) Thiadiazoles substitues et procede pour leur preparation
NL7407218A (en) 4-(3-Amino-2-acyloxypropoxyl)-1,2,5-thiadiazoles - useful as beta-adrenergic blocking agents
DK1044968T3 (da) 6-amino-2-oxo-pyrimidin-4-on-derivater, deres fremstilling og deres anvendelse som stabilisatorer for halogenholdige polymerer
IE33929L (en) Adamantanyl alkylamines
ES2191763T3 (es) Inhibidor del desarrollo de dependencia/tolerancia a un agente analgesico narcotico.
IT1155358B (it) Derivati chinazolinonici attivi contro la coccidiosi
EA199800366A1 (ru) Способы ингибирования ингибитора 1 активатора плазминогена
FR2630110B1 (fr) Nouveaux derives heteroarotinoides, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
ES8406431A1 (es) Procedimiento para preparar derivados de pleuromutilina
NO158019C (no) Analogifremgangsmaate for fremstilling av terapeutisk aktive imidazolinderivater.
ES2111768T3 (es) Derivados de carboestirilo utilizados como agentes antiarritmicos.
ES2080175T3 (es) Estabilizador para una preparacion que contiene 4-etil-2-hidroxiimino-5-nitro-3-hexenamida y metodo de estabilizacion correspondiente.
GB1440163A (en) Stabilizing polyolefins by means of amidothiophosphate diesters and amidothiophosphate diesters useful for such stabilization
AR035613A1 (es) Compuesto derivado de 2-piperidilimidazol, composicion farmaceutica que lo comprende y su uso en la fabricacion de un medicamento
ES2094132T3 (es) Uso de derivados de xantina contra la ulcera peptica.

Legal Events

Date Code Title Description
ST Notification of lapse