JPS5610179A - Synthesis of benzoxazole - Google Patents
Synthesis of benzoxazoleInfo
- Publication number
- JPS5610179A JPS5610179A JP8566179A JP8566179A JPS5610179A JP S5610179 A JPS5610179 A JP S5610179A JP 8566179 A JP8566179 A JP 8566179A JP 8566179 A JP8566179 A JP 8566179A JP S5610179 A JPS5610179 A JP S5610179A
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- oxime
- formula
- amide
- reacting
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
PURPOSE: To prepare the titled compound useful as an intermediate of medicines, etc., easily, in high yield, by reacting an oxime such as 2,4-dihydroxy-acetophenone oxime with phosphorus oxychloride in the presence of an amide such as N,N-dimethylacetamide under mild conditions.
CONSTITUTION: A benzoxazole of formula III (e.g. 2-methyl-6-hydroxybenzoxazole) is prepared by reacting an oxime of formula I (R1 is alkyl; R2 is halogen, OH, acyloxy, alkyl, alkyloxy, alkylthio, nitro, cyano, phenyl, etc., n is 0W4) with phosphorus oxychloride in the presence of an amide of formula II (R3 is H or alkyl; R4, R5 are alkyl; R3 and R4 or R4 and R5 may together form a ring).
EFFECT: A 2,5-dihydroxyacetophenone oxime derivative which is easily hydrolyzed at high temperature, can be used as a raw material.
USE: Intermediate of organic compounds for photographic use.
COPYRIGHT: (C)1981,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP8566179A JPS5610179A (en) | 1979-07-06 | 1979-07-06 | Synthesis of benzoxazole |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP8566179A JPS5610179A (en) | 1979-07-06 | 1979-07-06 | Synthesis of benzoxazole |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5610179A true JPS5610179A (en) | 1981-02-02 |
JPS613339B2 JPS613339B2 (en) | 1986-01-31 |
Family
ID=13865003
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP8566179A Granted JPS5610179A (en) | 1979-07-06 | 1979-07-06 | Synthesis of benzoxazole |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5610179A (en) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4594426A (en) * | 1980-01-17 | 1986-06-10 | Fuji Photo Film Co., Ltd. | Benzoxazole derivative intermediates for synthesis of dye releasing redox compounds |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS61296549A (en) * | 1985-06-24 | 1986-12-27 | Sharp Corp | Production of optical memory element |
-
1979
- 1979-07-06 JP JP8566179A patent/JPS5610179A/en active Granted
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4594426A (en) * | 1980-01-17 | 1986-06-10 | Fuji Photo Film Co., Ltd. | Benzoxazole derivative intermediates for synthesis of dye releasing redox compounds |
Also Published As
Publication number | Publication date |
---|---|
JPS613339B2 (en) | 1986-01-31 |
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