JPS5535045A - Imidazoline riboside derivative and its preparation - Google Patents
Imidazoline riboside derivative and its preparationInfo
- Publication number
- JPS5535045A JPS5535045A JP10851678A JP10851678A JPS5535045A JP S5535045 A JPS5535045 A JP S5535045A JP 10851678 A JP10851678 A JP 10851678A JP 10851678 A JP10851678 A JP 10851678A JP S5535045 A JPS5535045 A JP S5535045A
- Authority
- JP
- Japan
- Prior art keywords
- imidazoline
- aralkyl
- compound
- preparation
- ester
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Classifications
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Abstract
NEW MATERIAL:An imidazoline riboside derivative of formula I (R1 is alkyl or aralkyl; Y, Z are H or protecting group).
EXAMPLE: 1-(2, 3- O -Isopropylidene-5- O -acetyl-β- D -ribofuranosyl)2-oxo-5-cyanomethyl-4-imidazoline-4-carboxylic acid methyl ester.
USE: Intermediate of an intiviral substnace 3-deazaguanosine.
PROCESS: An alkyl ester or an aralkyl ester of 1-β-D-ribofuranosyl-2-oxo-5-acyloxymethyl-4-imidazoline-4-corboxylic acid of formula II (R2 is acyl) is reacted with a cyanide anion to afford the compound III. The compound II is novel compound which can be prepared from a compound III (R' is alkoxy or aralkyl).
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP10851678A JPS5535045A (en) | 1978-09-06 | 1978-09-06 | Imidazoline riboside derivative and its preparation |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP10851678A JPS5535045A (en) | 1978-09-06 | 1978-09-06 | Imidazoline riboside derivative and its preparation |
Publications (1)
Publication Number | Publication Date |
---|---|
JPS5535045A true JPS5535045A (en) | 1980-03-11 |
Family
ID=14486764
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP10851678A Pending JPS5535045A (en) | 1978-09-06 | 1978-09-06 | Imidazoline riboside derivative and its preparation |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5535045A (en) |
-
1978
- 1978-09-06 JP JP10851678A patent/JPS5535045A/en active Pending
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