JPS5511504A - Condensed heterocyclic-s-oxide - Google Patents

Condensed heterocyclic-s-oxide

Info

Publication number
JPS5511504A
JPS5511504A JP6736978A JP6736978A JPS5511504A JP S5511504 A JPS5511504 A JP S5511504A JP 6736978 A JP6736978 A JP 6736978A JP 6736978 A JP6736978 A JP 6736978A JP S5511504 A JPS5511504 A JP S5511504A
Authority
JP
Japan
Prior art keywords
formula
oxide
compound
condensed heterocyclic
lower alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP6736978A
Other languages
Japanese (ja)
Other versions
JPS6145609B2 (en
Inventor
Hironobu Sato
Kuniyuki Tomita
Shinsaku Kobayashi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Sankyo Co Ltd
Original Assignee
Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co Ltd filed Critical Sankyo Co Ltd
Priority to JP6736978A priority Critical patent/JPS5511504A/en
Priority to IT68217/79A priority patent/IT1119096B/en
Priority to CH524179A priority patent/CH644602A5/en
Priority to DE19792922756 priority patent/DE2922756A1/en
Priority to ES481298A priority patent/ES481298A1/en
Priority to GB7919498A priority patent/GB2022093B/en
Priority to FR7914314A priority patent/FR2428035A1/en
Priority to FR7927643A priority patent/FR2433521A1/en
Publication of JPS5511504A publication Critical patent/JPS5511504A/en
Priority to US06/184,096 priority patent/US4328238A/en
Publication of JPS6145609B2 publication Critical patent/JPS6145609B2/ja
Granted legal-status Critical Current

Links

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)

Abstract

NEW MATERIAL:A condensed heterocyclic-S-oxide of formula I (R1W3 are H, lower alkyl; X1,2 are H, lower alkyl, lower alkoxy, lower alkanesulphinyl, lower alkanesulphonyl, halogen, trifluoromethyl, nitro, cyano, lower alkoxy-carbonyl; n is 1, 2) and its acid addition salt.
EXAMPLE: 1,3,4,6-Tetrahydro-2H-5,1-benzothiazocin-S-oxide.
USE: Antiulcers having remarkable inhibiting activity of gastric secretion.
PROCESS: The oxidation of a compound of formula II gives the compound of formula I. The compound of formula II can be obtained by the ring-closure of a compound of formula IV, obtained by (1) oxidizing a novel derivative of an ω-substituted thioalkylaniline of formula III with a halide, etc., (2) alkylating or acylating the oxide if necessary, and (3) reducing the product.
COPYRIGHT: (C)1980,JPO&Japio
JP6736978A 1978-06-05 1978-06-05 Condensed heterocyclic-s-oxide Granted JPS5511504A (en)

Priority Applications (9)

Application Number Priority Date Filing Date Title
JP6736978A JPS5511504A (en) 1978-06-05 1978-06-05 Condensed heterocyclic-s-oxide
GB7919498A GB2022093B (en) 1978-06-05 1979-06-05 Benzothalzocines and benzothiazonines
CH524179A CH644602A5 (en) 1978-06-05 1979-06-05 DERIVATIVES OF BENZOTHIAZOCINE AND BENZOTHIAZONE, THEIR PRODUCTION AND PHARMACEUTICAL PREPARATIONS CONTAINING THESE DERIVATIVES.
DE19792922756 DE2922756A1 (en) 1978-06-05 1979-06-05 BENZOTHIAZOCINE, BENZOTHIAZOCINE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION
ES481298A ES481298A1 (en) 1978-06-05 1979-06-05 Benzothiazocine and benzothiazonine derivatives and use
IT68217/79A IT1119096B (en) 1978-06-05 1979-06-05 DERIVATIVES OF BENZOTHIAZOCIN AND BENZOTHIAZONIN PARTICULARLY USEFUL AS MEDICATIONS AND PROCEDURE FOR THEIR PREPARATION
FR7914314A FR2428035A1 (en) 1978-06-05 1979-06-05 BENZOTHIAZOCINE AND BENZOTHIAZONINE DERIVATIVES AND THEIR THERAPEUTIC APPLICATION
FR7927643A FR2433521A1 (en) 1978-06-05 1979-11-09 PROCESS FOR THE PREPARATION OF BENZOTHIAZOCIN AND BENZOTHIAZONINE DERIVATIVES
US06/184,096 US4328238A (en) 1978-06-05 1980-09-04 Benzothiazocine and benzothiazonine derivatives and use

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP6736978A JPS5511504A (en) 1978-06-05 1978-06-05 Condensed heterocyclic-s-oxide

Publications (2)

Publication Number Publication Date
JPS5511504A true JPS5511504A (en) 1980-01-26
JPS6145609B2 JPS6145609B2 (en) 1986-10-08

Family

ID=13343021

Family Applications (1)

Application Number Title Priority Date Filing Date
JP6736978A Granted JPS5511504A (en) 1978-06-05 1978-06-05 Condensed heterocyclic-s-oxide

Country Status (1)

Country Link
JP (1) JPS5511504A (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0543967U (en) * 1991-11-20 1993-06-15 積水化成品工業株式会社 A cup made of expanded polypropylene

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH0543967U (en) * 1991-11-20 1993-06-15 積水化成品工業株式会社 A cup made of expanded polypropylene

Also Published As

Publication number Publication date
JPS6145609B2 (en) 1986-10-08

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