JPS55104286A - Preparation of thienoimidazoline compound - Google Patents
Preparation of thienoimidazoline compoundInfo
- Publication number
- JPS55104286A JPS55104286A JP1175879A JP1175879A JPS55104286A JP S55104286 A JPS55104286 A JP S55104286A JP 1175879 A JP1175879 A JP 1175879A JP 1175879 A JP1175879 A JP 1175879A JP S55104286 A JPS55104286 A JP S55104286A
- Authority
- JP
- Japan
- Prior art keywords
- acid
- benzyl
- compound
- thienoimidazoline
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
PURPOSE: To prepare the title compound known as vitamin H, and useful as a growth-promoting agent and remdey for skin disease, in high yield and purity, at a low cost, by heating a benzyl biotin derivative in the presence of an alkanesulfonic acid such as methanesulfonic acid.
CONSTITUTION: Cis-tetrahydro-2-oxothieno[3,4-d]-imidazoline-4-valeric acid (biotin) is prepared by reacting 100 pts. wt. of a compound of formula (R1,2 are H or benzyl, provided that at least one of R1,2 is benzyl; R3 is H or carboxyl) with pref. 300W5000 parts of an alkanesulfonic acid (e.g. methanesulfonic acid and ethanesulfonic acid) at 110W150°C for 0.5W10hr. Crude crystals of the objective compound obtained by cooling the reaction mixture, is recrystallized with water.
COPYRIGHT: (C)1980,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP1175879A JPS55104286A (en) | 1979-02-02 | 1979-02-02 | Preparation of thienoimidazoline compound |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP1175879A JPS55104286A (en) | 1979-02-02 | 1979-02-02 | Preparation of thienoimidazoline compound |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS55104286A true JPS55104286A (en) | 1980-08-09 |
JPS638954B2 JPS638954B2 (en) | 1988-02-25 |
Family
ID=11786875
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP1175879A Granted JPS55104286A (en) | 1979-02-02 | 1979-02-02 | Preparation of thienoimidazoline compound |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS55104286A (en) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH02136996U (en) * | 1989-04-18 | 1990-11-15 | ||
JPH037824A (en) * | 1989-06-02 | 1991-01-16 | Sanyo Electric Co Ltd | Heat exchanging unit |
JPH09227564A (en) | 1995-12-20 | 1997-09-02 | Sumitomo Chem Co Ltd | Production of imidazole derivative |
CA2193774C (en) | 1995-12-26 | 2005-02-01 | Norihiko Hirata | Process for producing 1-hydroxythienoimidazole carboxylic acid and thienoimidazole carboxylic acid |
CH693745A5 (en) | 1998-12-24 | 2004-01-15 | Sumitomo Chemical Co | Process for the preparation of hexahydro-2-oxo-1H-thieno (3,4-d) imidazol-4-pentansaeure. |
-
1979
- 1979-02-02 JP JP1175879A patent/JPS55104286A/en active Granted
Also Published As
Publication number | Publication date |
---|---|
JPS638954B2 (en) | 1988-02-25 |
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