JPS5459293A - Novel cyclopeptide - Google Patents
Novel cyclopeptideInfo
- Publication number
- JPS5459293A JPS5459293A JP11983978A JP11983978A JPS5459293A JP S5459293 A JPS5459293 A JP S5459293A JP 11983978 A JP11983978 A JP 11983978A JP 11983978 A JP11983978 A JP 11983978A JP S5459293 A JPS5459293 A JP S5459293A
- Authority
- JP
- Japan
- Prior art keywords
- cyclopeptide
- novel
- novel cyclopeptide
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/08—Tripeptides
- C07K5/0821—Tripeptides with the first amino acid being heterocyclic, e.g. His, Pro, Trp
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/02—Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- C07K14/575—Hormones
- C07K14/655—Somatostatins
- C07K14/6555—Somatostatins at least 1 amino acid in D-form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
- Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y10S930/00—Peptide or protein sequence
- Y10S930/01—Peptide or protein sequence
- Y10S930/16—Somatostatin; related peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Endocrinology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Biochemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Gastroenterology & Hepatology (AREA)
- Zoology (AREA)
- Toxicology (AREA)
- Diabetes (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
LU78191A LU78191A1 (de) | 1977-09-28 | 1977-09-28 | Verfahren zur herstellung von neuen cyclopeptiden |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5459293A true JPS5459293A (en) | 1979-05-12 |
JPS6218560B2 JPS6218560B2 (ja) | 1987-04-23 |
Family
ID=19728716
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP11983978A Granted JPS5459293A (en) | 1977-09-28 | 1978-09-28 | Novel cyclopeptide |
Country Status (18)
Country | Link |
---|---|
US (1) | US4238481A (ja) |
EP (1) | EP0001295B1 (ja) |
JP (1) | JPS5459293A (ja) |
AT (1) | AT370090B (ja) |
AU (1) | AU523050B2 (ja) |
CA (1) | CA1111841A (ja) |
DD (1) | DD140142A5 (ja) |
DE (1) | DE2861672D1 (ja) |
DK (1) | DK151034C (ja) |
ES (1) | ES473677A1 (ja) |
FI (1) | FI68246C (ja) |
HU (1) | HU184612B (ja) |
IE (1) | IE47380B1 (ja) |
IL (1) | IL55643A (ja) |
LU (1) | LU78191A1 (ja) |
NO (1) | NO148957C (ja) |
NZ (1) | NZ188517A (ja) |
ZA (1) | ZA785488B (ja) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH0748272A (ja) * | 1987-07-10 | 1995-02-21 | Sandoz Ag | ソマトスタチン類に関する改良 |
Families Citing this family (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4328214A (en) * | 1979-07-04 | 1982-05-04 | Ciba-Geigy Corporation | Cyclopeptides and pharmaceutical preparations thereof and also processes for their manufacture |
NZ195303A (en) * | 1979-10-31 | 1984-10-19 | Merck & Co Inc | Cyclic hexapeptide somatostatin analogues,and pharmaceutical compositions |
US4369179A (en) * | 1979-12-14 | 1983-01-18 | Ciba-Geigy Corporation | Acylpeptides |
DD155985A5 (de) * | 1979-12-21 | 1982-07-21 | Ciba Geigy Ag | Verfahren zur herstellung cyclischr octapeptide |
US4360516A (en) * | 1981-04-13 | 1982-11-23 | Merck & Co., Inc. | Modified D-retro cyclic hexapeptide somatostatin analogs |
ATE14226T1 (de) * | 1981-12-24 | 1985-07-15 | Ciba Geigy Ag | Cyclische octapeptide und pharmazeutische praeparate davon, sowie verfahren zur herstellung derselben und ihre anwendung. |
HUT42101A (en) * | 1985-01-07 | 1987-06-29 | Sandoz Ag | Process for preparing stomatostatine derivatives and pharmaceutical compositions containing such compounds |
US4798821A (en) * | 1987-03-02 | 1989-01-17 | Merck & Co., Inc. | Antihypertensive therapy for diabetics |
CA2053250A1 (en) * | 1989-04-26 | 1990-10-27 | David H. Coy | Linear somatostatin analogs |
US5633263A (en) * | 1989-04-26 | 1997-05-27 | The Administrators Of The Tulane Educational Fund | Linear somatostatin analogs |
US5504069A (en) * | 1993-02-11 | 1996-04-02 | Biomeasure, Inc. | Inhibition of trauma-induced tumor growth |
US5597894A (en) * | 1995-06-05 | 1997-01-28 | The Louisiana State University Medical Center Foundation | Multi-tyrosinated somatostatin analogs |
ES2202864T3 (es) | 1997-05-13 | 2004-04-01 | Societe De Conseils De Recherches Et D'applications Scientifiques S.A.S. | Agonistas de la somatostatina para disminuir el peso corporal. |
US6004928A (en) * | 1997-05-13 | 1999-12-21 | Biomeasure, Incorporated | Method of treating hyperlipidemia |
ES2216290T3 (es) * | 1997-05-13 | 2004-10-16 | Societe De Conseils De Recherches Et D'applications Scientifiques S.A.S. | Somatostatina y agonistas de la somatostatina para el tratamiento de insensibilidad a la insulina y de sindrome x. |
EP0981364B1 (en) * | 1997-05-13 | 2006-03-01 | Societe De Conseils De Recherches Et D'applications Scientifiques S.A.S. | Method and compositions for treating hyperlipidemia |
US5968903A (en) * | 1998-05-07 | 1999-10-19 | Biomeasure, Incorporated | Inhibition of H. pylori proliferation |
ES2325880T3 (es) | 2001-06-08 | 2009-09-23 | Ipsen Pharma | Analogos quimericos de somatostatina-dopamina. |
WO2004092202A1 (en) * | 2003-04-07 | 2004-10-28 | Novetide, Ltd. | Process for production of cyclic peptides |
AU2004232314B2 (en) | 2003-04-22 | 2007-11-22 | Ipsen Pharma S.A.S. | Peptide vectors |
US20110171191A1 (en) | 2008-06-12 | 2011-07-14 | Syntaxin Limited | Suppression of neuroendocrine diseases |
JP5799397B2 (ja) | 2008-06-12 | 2015-10-28 | イプセン・バイオイノベーション・リミテッドIpsen Bioinnovation Limited | 癌の抑制 |
GB0820970D0 (en) | 2008-11-17 | 2008-12-24 | Syntaxin Ltd | Suppression of cancer |
EP2654772B1 (en) | 2010-12-22 | 2018-09-26 | The Salk Institute for Biological Studies | Cyclic crf antagonist peptides |
DK3007704T3 (da) | 2013-06-13 | 2021-03-29 | Antisense Therapeutics Ltd | Kombinationsterapi til akromegali |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS543085A (en) * | 1977-06-08 | 1979-01-11 | Merck & Co Inc | Somatostatin homologues*compositions and preparations |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4011182A (en) * | 1975-03-21 | 1977-03-08 | American Home Products Corporation | Cyclic undecapeptide analogs of somatostatin and intermediates |
US4000259A (en) * | 1975-06-16 | 1976-12-28 | American Home Products Corporation | Cyclic dodecapeptide analogs of somatostatin and intermediates |
NL7607987A (nl) * | 1975-08-08 | 1977-02-10 | Merck & Co Inc | Werkwijze voor het bereiden van peptiden. |
US3988304A (en) * | 1975-08-25 | 1976-10-26 | American Home Products Corporation | Cyclic dodecapeptide derivatives of somatostatin and intermediates thereof |
US4133805A (en) * | 1975-12-16 | 1979-01-09 | American Home Products Corporation | Cyclic undecapeptides related to somatostatin and intermediates therefor |
US4054558A (en) * | 1976-05-24 | 1977-10-18 | American Home Products Corporation | Cyclic dodecapeptide and intermediates therefor |
US4115554A (en) * | 1977-08-29 | 1978-09-19 | Merck & Co., Inc. | Somatostatin analogs |
-
1977
- 1977-09-28 LU LU78191A patent/LU78191A1/de unknown
-
1978
- 1978-09-15 US US05/942,565 patent/US4238481A/en not_active Expired - Lifetime
- 1978-09-25 DD DD78208064A patent/DD140142A5/de unknown
- 1978-09-25 FI FI782907A patent/FI68246C/fi not_active IP Right Cessation
- 1978-09-26 EP EP78100994A patent/EP0001295B1/de not_active Expired
- 1978-09-26 IL IL55643A patent/IL55643A/xx unknown
- 1978-09-26 DE DE7878100994T patent/DE2861672D1/de not_active Expired
- 1978-09-26 CA CA312,129A patent/CA1111841A/en not_active Expired
- 1978-09-26 ES ES473677A patent/ES473677A1/es not_active Expired
- 1978-09-27 DK DK428478A patent/DK151034C/da not_active IP Right Cessation
- 1978-09-27 AU AU40229/78A patent/AU523050B2/en not_active Expired
- 1978-09-27 NZ NZ188517A patent/NZ188517A/xx unknown
- 1978-09-27 AT AT0698278A patent/AT370090B/de not_active IP Right Cessation
- 1978-09-27 ZA ZA00785488A patent/ZA785488B/xx unknown
- 1978-09-27 HU HU78CI1860A patent/HU184612B/hu unknown
- 1978-09-27 IE IE1931/78A patent/IE47380B1/en unknown
- 1978-09-27 NO NO783268A patent/NO148957C/no unknown
- 1978-09-28 JP JP11983978A patent/JPS5459293A/ja active Granted
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS543085A (en) * | 1977-06-08 | 1979-01-11 | Merck & Co Inc | Somatostatin homologues*compositions and preparations |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPH0748272A (ja) * | 1987-07-10 | 1995-02-21 | Sandoz Ag | ソマトスタチン類に関する改良 |
Also Published As
Publication number | Publication date |
---|---|
FI782907A (fi) | 1979-03-29 |
ATA698278A (de) | 1982-07-15 |
IE47380B1 (en) | 1984-03-07 |
IE781931L (en) | 1979-03-28 |
FI68246C (fi) | 1985-08-12 |
FI68246B (fi) | 1985-04-30 |
DE2861672D1 (en) | 1982-04-15 |
US4238481A (en) | 1980-12-09 |
AU523050B2 (en) | 1982-07-08 |
CA1111841A (en) | 1981-11-03 |
HU184612B (en) | 1984-09-28 |
AT370090B (de) | 1983-02-25 |
NO783268L (no) | 1979-03-29 |
LU78191A1 (de) | 1979-05-25 |
DD140142A5 (de) | 1980-02-13 |
DK428478A (da) | 1979-03-29 |
NO148957B (no) | 1983-10-10 |
EP0001295A3 (en) | 1979-06-13 |
ES473677A1 (es) | 1980-05-16 |
IL55643A (en) | 1981-12-31 |
IL55643A0 (en) | 1978-12-17 |
EP0001295A2 (de) | 1979-04-04 |
JPS6218560B2 (ja) | 1987-04-23 |
DK151034B (da) | 1987-10-12 |
EP0001295B1 (de) | 1982-03-17 |
DK151034C (da) | 1988-02-22 |
AU4022978A (en) | 1980-04-03 |
NZ188517A (en) | 1981-04-24 |
NO148957C (no) | 1984-01-18 |
ZA785488B (en) | 1979-09-26 |
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