JPS5441871A - Novel 55hydroxymethyloxazolidinons and its manufacture - Google Patents

Novel 55hydroxymethyloxazolidinons and its manufacture

Info

Publication number
JPS5441871A
JPS5441871A JP10082478A JP10082478A JPS5441871A JP S5441871 A JPS5441871 A JP S5441871A JP 10082478 A JP10082478 A JP 10082478A JP 10082478 A JP10082478 A JP 10082478A JP S5441871 A JPS5441871 A JP S5441871A
Authority
JP
Japan
Prior art keywords
novel
manufacture
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP10082478A
Other languages
English (en)
Other versions
JPS6354710B2 (ja
Inventor
Dosuteru Fuiritsupu
Douzon Koretsuto
Buurugerii Gii
Guure Kuroodo
Motsukiyuu Gizeeru
Kosuton Jiyannaran
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Delalande SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR7726105A external-priority patent/FR2381037A2/fr
Priority claimed from FR7815342A external-priority patent/FR2426684A2/fr
Application filed by Delalande SA filed Critical Delalande SA
Publication of JPS5441871A publication Critical patent/JPS5441871A/ja
Publication of JPS6354710B2 publication Critical patent/JPS6354710B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2
    • C07D263/24—Oxygen atoms attached in position 2 with hydrocarbon radicals, substituted by oxygen atoms, attached to other ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine
JP10082478A 1977-08-26 1978-08-18 Novel 55hydroxymethyloxazolidinons and its manufacture Granted JPS5441871A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR7726105A FR2381037A2 (fr) 1977-02-22 1977-08-26 Nouvelles hydroxymethyl-5 oxazolidinones-2, leur procede de preparation et leur application therapeutique
FR7815342A FR2426684A2 (fr) 1978-05-23 1978-05-23 Nouvelles hydroxymethyl-5 oxazolidinones-2, leur procede de preparation et leur application en therapeutique

Publications (2)

Publication Number Publication Date
JPS5441871A true JPS5441871A (en) 1979-04-03
JPS6354710B2 JPS6354710B2 (ja) 1988-10-28

Family

ID=26220188

Family Applications (1)

Application Number Title Priority Date Filing Date
JP10082478A Granted JPS5441871A (en) 1977-08-26 1978-08-18 Novel 55hydroxymethyloxazolidinons and its manufacture

Country Status (13)

Country Link
US (2) US4250318A (ja)
JP (1) JPS5441871A (ja)
AU (1) AU526714B2 (ja)
CA (1) CA1113093A (ja)
CH (1) CH634836A5 (ja)
DE (1) DE2836305A1 (ja)
ES (1) ES472825A1 (ja)
GB (1) GB2003151B (ja)
GR (1) GR64146B (ja)
IT (1) IT1118099B (ja)
LU (1) LU80081A1 (ja)
NL (1) NL7808817A (ja)
SE (1) SE444813B (ja)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS53108278A (en) * 1977-11-14 1978-09-20 Nec Corp Manufacture of semiconductor device
JPS57128058A (en) * 1980-12-15 1982-08-09 Seiko Epson Corp Manufacture of semiconductor device
JPS5980668A (ja) * 1982-06-08 1984-05-10 デラランデ・エス・ア− Ｎ−アリル化オキサゾリジン−２−オンの光学活性な誘導体、該誘導体の製法及び該誘導体による薬剤
US5169803A (en) * 1990-11-28 1992-12-08 Nec Corporation Method of filling contact holes of a semiconductor device

Families Citing this family (58)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4348393A (en) 1978-06-09 1982-09-07 Delalande S.A. N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones
FR2460940A2 (fr) * 1979-07-10 1981-01-30 Delalande Sa Nouvelles hydroxymethyl-5 oxazolidinones-2, leur procede de preparation et leur application en therapeutique
CA1171865A (en) * 1980-06-04 1984-07-31 Alain Lacour N-aryl azolone derivatives, the process for preparing the same and their application in therapeutics
US4340606A (en) 1980-10-23 1982-07-20 E. I. Du Pont De Nemours And Company 3-(p-Alkylsulfonylphenyl)oxazolidinone derivatives as antibacterial agents
FR2500450A1 (fr) * 1981-02-25 1982-08-27 Delalande Sa Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique
ES517852A0 (es) * 1981-12-04 1984-01-16 Du Pont Un procedimiento para la preparacion de derivados de bencenosulfonamidas.
US4405794A (en) * 1981-12-18 1983-09-20 The Dow Chemical Company Preparation of 2-oxazolidinone and ethyleneurea
US4461773A (en) * 1982-09-15 1984-07-24 E. I. Dupont De Nemours And Company P-Oxooxazolidinylbenzene compounds as antibacterial agents
US4500717A (en) * 1983-03-28 1985-02-19 The Dow Chemical Company Process for preparation of 2-oxazolidinones
US4705799A (en) * 1983-06-07 1987-11-10 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl benzenes useful as antibacterial agents
US4732956A (en) * 1984-06-18 1988-03-22 Loctite (Ireland) Ltd. Styryloxy resins and compositions thereof
CA1260948A (en) 1984-12-05 1989-09-26 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl benzene derivatives useful as antibacterial agents
US4965268A (en) * 1987-10-09 1990-10-23 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US4985429A (en) * 1987-10-09 1991-01-15 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5036093A (en) * 1987-10-09 1991-07-30 Du Pont Merck Pharmaceutical Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents
US4801600A (en) * 1987-10-09 1989-01-31 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5032605A (en) * 1987-10-09 1991-07-16 Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US5039690A (en) * 1987-10-09 1991-08-13 Du Pont Merck Pharmaceutical Company Aminomethyl oxooxazolidinyl oxa or thia cycloalkylbenzene derivatives useful as antibacterial agents
US4921869A (en) * 1987-10-09 1990-05-01 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl cycloalkylbenzene derivatives useful as antibacterial agents
US5036092A (en) * 1987-10-09 1991-07-30 Du Pont Merck Pharmaceutical Aminomethyl oxooxazolidinyl azacycloalkylbenzene derivatives useful as antibacterial agents
US4942183A (en) * 1987-10-16 1990-07-17 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl aroylbenzene derivatives useful as antibacterial agents
US4977173A (en) * 1987-10-21 1990-12-11 E. I. Du Pont De Nemours And Company Aminomethyl oxooxazolidinyl ethenylbenzene derivatives useful as antibacterial agents
US5254577A (en) * 1988-07-29 1993-10-19 The Du Pont Merck Pharmaceutical Company Aminomethyloxooxazolidinyl arylbenzene derivatives useful as antibacterial agents
US5182403A (en) * 1988-09-15 1993-01-26 The Upjohn Company Substituted 3(5'indazolyl) oxazolidin-2-ones
US5225565A (en) * 1988-09-15 1993-07-06 The Upjohn Company Antibacterial 3-(fused-ring substituted)phenyl-5β-amidomethyloxazolidin-2-ones
US5235063A (en) * 1989-10-17 1993-08-10 Delalande S.A. Process of preparing by condensation certain
US5196543A (en) * 1989-10-17 1993-03-23 Delalande S.A. 3-aryloxazolidinone derivatives, process for their preparation and their use in therapy
FR2653017B1 (fr) * 1989-10-17 1995-05-05 Delalande Sa Derives d'aryl-3 oxazolidinone-2, leur procede de preparation et leur application en therapeutique.
US5231188A (en) * 1989-11-17 1993-07-27 The Upjohn Company Tricyclic [6.5.51]-fused oxazolidinone antibacterial agents
AU667198B2 (en) * 1991-11-01 1996-03-14 Pharmacia & Upjohn Company Substituted aryl- and heteroarylphenyloxazolidinones useful as antibacterial agents
KR100276382B1 (ko) * 1992-12-08 2000-12-15 로렌스 티. 마이젠헬더 트로폰-치환된 페닐옥사졸리디논 항균제
TW286317B (ja) * 1993-12-13 1996-09-21 Hoffmann La Roche
MX9703040A (es) * 1995-09-12 1997-07-31 Upjohn Co Antimicrobianos de feniloxazolidinona.
FR2741071B1 (fr) * 1995-11-09 1997-12-12 Synthelabo Derives de 3-(benzofuran-5-yl)oxazolidin-2-one, leur preparation et leur application en therapeutique
US5795985A (en) * 1996-03-05 1998-08-18 Ciba Specialty Chemicals Corporation Phenyl alkyl ketone substituted by cyclic amine and a process for the preparation thereof
KR100530297B1 (ko) * 1996-04-11 2005-11-22 파마시아 앤드 업존 캄파니 엘엘씨 옥사졸리디논의 제조 방법
US6037354A (en) 1997-06-18 2000-03-14 Merck & Co., Inc. Alpha 1a adrenergic receptor antagonists
EP1028940B1 (en) 1997-11-07 2007-04-18 Pharmacia & Upjohn Company LLC Process to produce oxazolidinones
DE19962924A1 (de) * 1999-12-24 2001-07-05 Bayer Ag Substituierte Oxazolidinone und ihre Verwendung
CA2423599A1 (en) 2000-10-17 2002-04-25 Pharmacia & Upjohn Company Methods of producing oxazolidinone compounds
DE10129725A1 (de) * 2001-06-20 2003-01-02 Bayer Ag Kombinationstherapie substituierter Oxazolidinone
TW200302095A (en) * 2002-01-25 2003-08-01 Upjohn Co Oxazolidinone cotherapy
DE10300111A1 (de) * 2003-01-07 2004-07-15 Bayer Healthcare Ag Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid
DE10355461A1 (de) 2003-11-27 2005-06-23 Bayer Healthcare Ag Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung
KR100854211B1 (ko) 2003-12-18 2008-08-26 동아제약주식회사 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물
DE102004062475A1 (de) * 2004-12-24 2006-07-06 Bayer Healthcare Ag Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung
EP1685841A1 (en) * 2005-01-31 2006-08-02 Bayer Health Care Aktiengesellschaft Prevention and treatment of thromboembolic disorders
DE102005045518A1 (de) * 2005-09-23 2007-03-29 Bayer Healthcare Ag 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung
DE102005047561A1 (de) 2005-10-04 2007-04-05 Bayer Healthcare Ag Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung
EP1934208B1 (de) 2005-10-04 2011-03-23 Bayer Schering Pharma Aktiengesellschaft Neue polymorphe form von 5-chlor-n-({ ( 5s )-2-0x0-3-[4-( 3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl} -methyl)-2-thiophencarboxamid
DE102005047558A1 (de) * 2005-10-04 2008-02-07 Bayer Healthcare Ag Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen
DE102005048824A1 (de) * 2005-10-10 2007-04-12 Bayer Healthcare Ag Behandlung und Prophylaxe von Mikroangiopathien
DE102006051625A1 (de) * 2006-11-02 2008-05-08 Bayer Materialscience Ag Kombinationstherapie substituierter Oxazolidinone
KR101674146B1 (ko) * 2008-10-10 2016-11-08 머크 샤프 앤드 돔 코포레이션 옥사졸리디논 및 이를 포함하는 조성물을 제조하는 방법
CN102439006A (zh) 2009-02-03 2012-05-02 特留斯治疗学公司 (r)-3-(4-(2-(2-甲基四唑-5-基)吡啶-5-基)-3-氟苯基)-5-羟甲基噁唑烷-2-酮二氢磷酸酯的晶型
US8580767B2 (en) * 2009-05-28 2013-11-12 Trius Therapeutics, Inc. Oxazolidinone containing dimer compounds, compositions and methods to make and use
CN103601724B (zh) * 2013-11-14 2016-05-25 暨南大学 一种新型噁唑烷酮类化合物及其制备方法和应用
CN103965085B (zh) * 2014-04-17 2016-02-24 上海恒晟药业有限公司 一种取代1,2-氨基醇药物的制备方法

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6040428A (ja) * 1983-08-12 1985-03-02 Wakachiku Kensetsu Kk ケ−ソンの据付工法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1180089A (en) * 1967-10-20 1970-02-04 Delalande Sa Acetylenic Derivatives of 2-Oxazolidinones and processes of preparation
GB1224995A (en) * 1968-09-20 1971-03-10 Delalande Sa New 5-propargyloxymethyl-2-substituted oxazolidinones and their process of preparation
GB1222708A (en) * 1968-10-22 1971-02-17 Delalande Sa Novel 5-(n-substituted aminomethyl)-2-oxazolidinones and their process of preparation
GB1252101A (ja) * 1969-03-18 1971-11-03
DE2538424C2 (de) * 1975-08-29 1983-01-05 Nordmark-Werke Gmbh, 2000 Hamburg 4-substituierte 5-Phenyl-oxazolidon-(2)- Verbindungen und ein diese enthaltendes pharmazeutisches Präparat
FR2356422A1 (fr) * 1976-03-01 1978-01-27 Delalande Sa Nouveaux hydroxymethyl-5 oxazolidinone-2, leur procede de preparation et leur application en therapeutique

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6040428A (ja) * 1983-08-12 1985-03-02 Wakachiku Kensetsu Kk ケ−ソンの据付工法

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS53108278A (en) * 1977-11-14 1978-09-20 Nec Corp Manufacture of semiconductor device
JPS5442585B2 (ja) * 1977-11-14 1979-12-14
JPS57128058A (en) * 1980-12-15 1982-08-09 Seiko Epson Corp Manufacture of semiconductor device
JPS6334619B2 (ja) * 1980-12-15 1988-07-11 Seiko Epson Corp
JPS5980668A (ja) * 1982-06-08 1984-05-10 デラランデ・エス・ア− Ｎ−アリル化オキサゾリジン−２−オンの光学活性な誘導体、該誘導体の製法及び該誘導体による薬剤
US5169803A (en) * 1990-11-28 1992-12-08 Nec Corporation Method of filling contact holes of a semiconductor device
US5278449A (en) * 1990-11-28 1994-01-11 Nec Corporation Semiconductor memory device

Also Published As

Publication number Publication date
ES472825A1 (es) 1979-02-16
US4338451A (en) 1982-07-06
GB2003151B (en) 1982-10-06
JPS6354710B2 (ja) 1988-10-28
NL7808817A (nl) 1979-02-28
DE2836305A1 (de) 1979-03-01
SE444813B (sv) 1986-05-12
GB2003151A (en) 1979-03-07
GR64146B (en) 1980-01-31
CA1113093A (fr) 1981-11-24
US4250318A (en) 1981-02-10
AU3924978A (en) 1980-02-28
LU80081A1 (fr) 1979-05-15
CH634836A5 (fr) 1983-02-28
AU526714B2 (en) 1983-01-27
IT7868979A0 (it) 1978-08-25
SE7808804L (sv) 1979-02-27
IT1118099B (it) 1986-02-24

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