JPS5112630B2 - - Google Patents
Info
- Publication number
- JPS5112630B2 JPS5112630B2 JP48022273A JP2227373A JPS5112630B2 JP S5112630 B2 JPS5112630 B2 JP S5112630B2 JP 48022273 A JP48022273 A JP 48022273A JP 2227373 A JP2227373 A JP 2227373A JP S5112630 B2 JPS5112630 B2 JP S5112630B2
- Authority
- JP
- Japan
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/48—Acylated amino or imino radicals by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof, e.g. carbonylguanidines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT2108672 | 1972-02-25 | ||
| IT2023173 | 1973-02-09 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPS4897868A JPS4897868A (enExample) | 1973-12-13 |
| JPS5112630B2 true JPS5112630B2 (enExample) | 1976-04-21 |
Family
ID=26327456
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP48022273A Expired JPS5112630B2 (enExample) | 1972-02-25 | 1973-02-26 |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US3933838A (enExample) |
| JP (1) | JPS5112630B2 (enExample) |
| BE (1) | BE795907A (enExample) |
| CA (1) | CA1006525A (enExample) |
| DE (2) | DE2309251A1 (enExample) |
| ES (1) | ES412052A1 (enExample) |
| FR (1) | FR2181764B1 (enExample) |
| GB (1) | GB1425505A (enExample) |
| NL (1) | NL7302528A (enExample) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4025528A (en) * | 1973-10-24 | 1977-05-24 | Shionogi & Co., Ltd. | Thiazole derivatives of benzoic and phenylalkanoic acids |
| DE2828091A1 (de) * | 1978-06-27 | 1980-01-10 | Boehringer Sohn Ingelheim | 4-substituierte thiazoloxamsaeuren sowie ihre salze und ester |
| US4225719A (en) * | 1978-12-29 | 1980-09-30 | Eastman Kodak Company | Process for preparing 2-amino-5-formylthiazole and its hydrobromide salt |
| US4336388A (en) * | 1980-06-23 | 1982-06-22 | Hoffmann-La Roche Inc. | Thiazolyl benzophenone compounds |
| FR2581063B1 (fr) * | 1985-04-30 | 1987-07-17 | Chauvin Blache Lab | Amino-2 thiazoles n-substitues, leur procede de preparation et leur application en therapeutique |
| US5000775A (en) * | 1985-12-31 | 1991-03-19 | Monsanto Company | 2-amino-4,5-disubstituted-oxazole/thiazole compounds as herbicide antidotes |
| US4761422A (en) * | 1986-11-20 | 1988-08-02 | Lusofarmaco Istituto Lusofarmaco D'italia Spa | (2-amino-4-aryl-thiazole-5-yl)ethanols and their derivatives having diuretic activity and methods for preparing the same |
| AU644281B2 (en) * | 1991-04-24 | 1993-12-02 | Sumitomo Pharmaceuticals Company, Limited | Novel thiazole derivatives |
| WO2000035455A1 (en) * | 1998-12-15 | 2000-06-22 | Telik, Inc. | Heteroaryl-aryl ureas as igf-1 receptor antagonists |
| EP1418909B1 (en) * | 2001-08-13 | 2013-02-20 | Janssen Pharmaceutica NV | 2-AMINO-4, 5-TRISUBSTITUTED THIAzOLYL DERIVATIVES AND THEIR USE AGAINST AUTOIMMUNE DISEASES |
| US7138403B2 (en) * | 2001-08-13 | 2006-11-21 | Janssen Pharmaceutica N.V. | 2,4,5-trisubstituted thiazolyl derivatives and their antiinflammatory activity |
| US7183276B2 (en) | 2002-02-28 | 2007-02-27 | Takeda Pharmaceutical Company Limited | Azole compounds |
| KR20080019213A (ko) * | 2005-05-09 | 2008-03-03 | 아칠리온 파르마세우티칼스 인코포레이티드 | 티아졸 화합물 및 그 사용방법 |
| JP5341516B2 (ja) * | 2005-09-13 | 2013-11-13 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | ２−アニリン−４−アリール置換チアゾール誘導体 |
| EP2460800A1 (en) * | 2006-03-08 | 2012-06-06 | Achillion Pharmaceuticals, Inc. | Substituted aminothiazole derivatives with anti-HCV activity |
| MX2009012613A (es) * | 2007-05-22 | 2010-04-21 | Achillion Pharmaceuticals Inc | Tiazoles substituidos por heteroarilo y su uso como agentes antivirales. |
| JO2784B1 (en) * | 2007-10-18 | 2014-03-15 | شركة جانسين فارماسوتيكا ان. في | 5,3,1 - Triazole substitute derivative |
| JP2011500625A (ja) * | 2007-10-18 | 2011-01-06 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | トリ置換された１，２，４−トリアゾール |
| NZ587669A (en) * | 2008-03-19 | 2011-07-29 | Janssen Pharmaceutica Nv | Trisubstituted 1, 2, 4 -triazoles as nicotinic acetylcholine receptor modulators |
| EP2280945B1 (en) * | 2008-05-09 | 2014-09-03 | Janssen Pharmaceutica, N.V. | Trisubstituted pyrazoles as acetylcholine receptor modulators |
| US9453002B2 (en) | 2013-08-16 | 2016-09-27 | Janssen Pharmaceutica Nv | Substituted imidazoles as N-type calcium channel blockers |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US2423709A (en) * | 1947-07-08 | X-aryl thiazole | ||
| US3575991A (en) * | 1969-03-11 | 1971-04-20 | American Home Prod | 1-(4-aryl - 5 - carboxymethyl-2-thiazolyl)-1,6-dihydro -6 - oxonicotinic acids and esters thereof |
-
0
- BE BE795907D patent/BE795907A/xx unknown
-
1973
- 1973-02-23 NL NL7302528A patent/NL7302528A/xx unknown
- 1973-02-23 US US05/335,255 patent/US3933838A/en not_active Expired - Lifetime
- 1973-02-24 ES ES412052A patent/ES412052A1/es not_active Expired
- 1973-02-24 DE DE19732309251 patent/DE2309251A1/de active Pending
- 1973-02-24 DE DE2365526*A patent/DE2365526A1/de active Pending
- 1973-02-26 GB GB938273A patent/GB1425505A/en not_active Expired
- 1973-02-26 JP JP48022273A patent/JPS5112630B2/ja not_active Expired
- 1973-02-26 FR FR7306736A patent/FR2181764B1/fr not_active Expired
- 1973-02-26 CA CA164,590A patent/CA1006525A/en not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| AU5246773A (en) | 1974-08-22 |
| BE795907A (fr) | 1973-06-18 |
| DE2365526A1 (de) | 1975-07-31 |
| JPS4897868A (enExample) | 1973-12-13 |
| GB1425505A (en) | 1976-02-18 |
| CA1006525A (en) | 1977-03-08 |
| FR2181764B1 (enExample) | 1976-07-02 |
| US3933838A (en) | 1976-01-20 |
| DE2309251A1 (de) | 1973-09-06 |
| ES412052A1 (es) | 1976-05-01 |
| FR2181764A1 (enExample) | 1973-12-07 |
| NL7302528A (enExample) | 1973-08-28 |