JPH10130261A5 - - Google Patents
Info
- Publication number
- JPH10130261A5 JPH10130261A5 JP1997289612A JP28961297A JPH10130261A5 JP H10130261 A5 JPH10130261 A5 JP H10130261A5 JP 1997289612 A JP1997289612 A JP 1997289612A JP 28961297 A JP28961297 A JP 28961297A JP H10130261 A5 JPH10130261 A5 JP H10130261A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- formula
- piperidinyl
- pyrrolidinyl
- phenoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US2951996P | 1996-10-24 | 1996-10-24 | |
| US60/029519 | 1996-10-24 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPH10130261A JPH10130261A (ja) | 1998-05-19 |
| JPH10130261A5 true JPH10130261A5 (https=) | 2005-06-30 |
Family
ID=21849446
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP9289612A Withdrawn JPH10130261A (ja) | 1996-10-24 | 1997-10-22 | ベンゾチオフェン化合物、中間体、組成物および方法 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US5985897A (https=) |
| EP (1) | EP0838462B1 (https=) |
| JP (1) | JPH10130261A (https=) |
| AT (1) | ATE259361T1 (https=) |
| CA (1) | CA2216592C (https=) |
| DE (1) | DE69727529T2 (https=) |
| ES (1) | ES2213805T3 (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6136030A (en) * | 1999-01-12 | 2000-10-24 | Purzer Pharmaceutical Co., Ltd. | Process for preparing porous bioceramic materials |
| US6894175B1 (en) * | 1999-08-04 | 2005-05-17 | The Procter & Gamble Company | 2-Decarboxy-2-phosphinico prostaglandin derivatives and methods for their preparation and use |
| JP2004531559A (ja) * | 2001-05-22 | 2004-10-14 | イーライ・リリー・アンド・カンパニー | エストロゲン欠乏または内因性エストロゲンに対する異常な生理反応に関連する疾患を抑制するためのテトラヒドロキノリン誘導体 |
| EP1395563B1 (en) | 2001-05-22 | 2006-03-29 | Eli Lilly And Company | 2-substituted 1,2,3,4-tetrahydroquinolines and derivatives thereof, compositions and methods |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1300575B (de) * | 1965-05-21 | 1969-08-07 | Bristol Myers Co | Benzo[b]thiophene |
| US3394125A (en) * | 1965-10-23 | 1968-07-23 | Bristol Myers Co | 2-phenyl-3-tertiary-aminoalkoxy phenyl-and corresponding tertiaryaminoalkyl thio benzfurans substituted in the benzo nucleus with an alkoxy or tertiaryamino alkoxy or alkylthio group |
| US4230862A (en) * | 1975-10-28 | 1980-10-28 | Eli Lilly And Company | Antifertility compounds |
| US4133814A (en) * | 1975-10-28 | 1979-01-09 | Eli Lilly And Company | 2-Phenyl-3-aroylbenzothiophenes useful as antifertility agents |
| US4418068A (en) * | 1981-04-03 | 1983-11-29 | Eli Lilly And Company | Antiestrogenic and antiandrugenic benzothiophenes |
| US4358593A (en) * | 1981-04-03 | 1982-11-09 | Eli Lilly And Company | Process for preparing 3-(4-aminoethoxybenzoyl)benzo[b]thiophenes |
| US4380635A (en) * | 1981-04-03 | 1983-04-19 | Eli Lilly And Company | Synthesis of acylated benzothiophenes |
| GB2097788B (en) * | 1981-04-03 | 1985-04-24 | Lilly Co Eli | Benzothiophene compounds and process for preparing them |
| US4916126A (en) * | 1987-09-25 | 1990-04-10 | Ciba-Geigy Corporation | Diacyl derivatives of 4-(trialkylbenzyl)-piperazinyl compounds |
| WO1989002893A1 (en) * | 1987-09-30 | 1989-04-06 | The University Of Tennessee Research Corporation | Certain 3-substituted 2-alkyl benzothiophene derivatives |
| US5395842A (en) * | 1988-10-31 | 1995-03-07 | Endorecherche Inc. | Anti-estrogenic compounds and compositions |
| DE4117512A1 (de) * | 1991-05-25 | 1992-11-26 | Schering Ag | 2-phenylbenzo(b)furane und -thiophene, verfahren zu deren herstellung und diese enthaltende pharmazeutische praeparate |
| JP3157882B2 (ja) * | 1991-11-15 | 2001-04-16 | 帝国臓器製薬株式会社 | 新規なベンゾチオフエン誘導体 |
| US6756388B1 (en) * | 1993-10-12 | 2004-06-29 | Pfizer Inc. | Benzothiophenes and related compounds as estrogen agonists |
| CA2145614A1 (en) * | 1994-03-31 | 1995-10-01 | Jeffrey A. Dodge | Intermediates and processes for preparing benzothiophene compounds |
| US7501441B1 (en) * | 1994-09-20 | 2009-03-10 | Eli Lilly And Company | Naphthyl compounds, intermediates, processes, compositions, and methods |
| SG64896A1 (en) * | 1995-02-28 | 1999-05-25 | Lilly Co Eli | Benzothiophene compounds intermediates compositions and methods |
| US5510357A (en) * | 1995-02-28 | 1996-04-23 | Eli Lilly And Company | Benzothiophene compounds as anti-estrogenic agents |
| US6395755B1 (en) * | 1995-03-10 | 2002-05-28 | Eli Lilly And Company | Benzothiophene pharmaceutical compounds |
-
1997
- 1997-09-29 CA CA002216592A patent/CA2216592C/en not_active Expired - Fee Related
- 1997-10-22 JP JP9289612A patent/JPH10130261A/ja not_active Withdrawn
- 1997-10-22 ES ES97308414T patent/ES2213805T3/es not_active Expired - Lifetime
- 1997-10-22 AT AT97308414T patent/ATE259361T1/de not_active IP Right Cessation
- 1997-10-22 DE DE69727529T patent/DE69727529T2/de not_active Expired - Fee Related
- 1997-10-22 EP EP97308414A patent/EP0838462B1/en not_active Expired - Lifetime
- 1997-10-23 US US08/956,087 patent/US5985897A/en not_active Expired - Fee Related
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