JPH0450304B2 - - Google Patents

Info

Publication number
JPH0450304B2
JPH0450304B2 JP58062056A JP6205683A JPH0450304B2 JP H0450304 B2 JPH0450304 B2 JP H0450304B2 JP 58062056 A JP58062056 A JP 58062056A JP 6205683 A JP6205683 A JP 6205683A JP H0450304 B2 JPH0450304 B2 JP H0450304B2
Authority
JP
Japan
Prior art keywords
reaction
titibabin
amination
ammonia
amination method
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
JP58062056A
Other languages
English (en)
Japanese (ja)
Other versions
JPS58208266A (ja
Inventor
Kei Matsukugiru Chaaruzu
Jei Sutoo Jeemuzu
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
REIRII IND Inc
Original Assignee
REIRII IND Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by REIRII IND Inc filed Critical REIRII IND Inc
Publication of JPS58208266A publication Critical patent/JPS58208266A/ja
Publication of JPH0450304B2 publication Critical patent/JPH0450304B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/73—Unsubstituted amino or imino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79—Acids; Esters
    • C07D213/80—Acids; Esters in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/81—Amides; Imides
    • C07D213/82—Amides; Imides in position 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pyridine Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Quinoline Compounds (AREA)
JP58062056A 1982-04-08 1983-04-08 改良チチバビン反応 Granted JPS58208266A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US06/366,598 US4386209A (en) 1982-04-08 1982-04-08 Chichibabin reaction
US366598 1982-04-08
US478138 1983-03-23

Publications (2)

Publication Number Publication Date
JPS58208266A JPS58208266A (ja) 1983-12-03
JPH0450304B2 true JPH0450304B2 (enExample) 1992-08-13

Family

ID=23443677

Family Applications (1)

Application Number Title Priority Date Filing Date
JP58062056A Granted JPS58208266A (ja) 1982-04-08 1983-04-08 改良チチバビン反応

Country Status (2)

Country Link
US (1) US4386209A (enExample)
JP (1) JPS58208266A (enExample)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5003069A (en) * 1982-04-08 1991-03-26 Reilly Industries, Inc. Chichibabin reaction
DE3886467T2 (de) * 1987-08-01 1994-06-01 Takeda Chemical Industries Ltd Alpha-ungesättigte Amine, ihre Herstellung und Verwendung.
PL163080B1 (pl) * 1990-04-23 1994-02-28 Inst Chemii Organicznej Pan Sposób wytwarzania amin aromatycznych PL
DE4232175A1 (de) * 1992-04-15 1993-10-21 Bayer Ag Verfahren zur Herstellung von 2-Amino-5-methyl-pyridin
DE4234637A1 (de) * 1992-10-14 1994-04-21 Bayer Ag Verfahren zur Herstellung von 2-substituierten 5-Alkyl-pyridinen
RU2165414C2 (ru) * 1994-06-24 2001-04-20 Рейлли Индастриз, Инк. Усовершенствованный способ аминирования пиридиновых оснований по чичибабину
IL114314A (en) * 1994-06-24 2000-12-06 Reilly Ind Inc Amination of pyridine bases
US5808081A (en) * 1995-06-26 1998-09-15 Reilly Industries, Inc. Chichibabin aminations of pyridine bases
US5972975A (en) * 1995-12-08 1999-10-26 Merck & Co., Inc. Substituted 2-aminopyridines as inhibitors of nitric oxide synthase
AR019190A1 (es) * 1998-07-08 2001-12-26 Sod Conseils Rech Applic Derivados de 2-aminopiridinas, productos intermedios para su preparacion, medicamentos y composiciones farmaceuticas que los contienen y su uso para preparar medicamentos
KR20090091347A (ko) * 2006-12-21 2009-08-27 이 아이 듀폰 디 네모아 앤드 캄파니 글루타르이미딘으로부터의 2,6-다이아미노피리딘의 합성 방법
US7999057B2 (en) * 2008-07-08 2011-08-16 E. I. Du Pont De Nemours And Company Gas-phase process for the synthesis of diaminopyridines from glutaronitriles
CN102276526B (zh) * 2011-08-08 2013-04-17 中国科学院长春应用化学研究所 一种2-氨基吡啶类化合物合成方法
CN106496105B (zh) * 2016-08-31 2019-01-11 南京红太阳生物化学有限责任公司 一种3-甲基吡啶氨化制备2-氨基-5-甲基吡啶的方法
JP7808109B2 (ja) * 2021-06-29 2026-01-28 大塚化学株式会社 ゴム組成物及びタイヤ
CN114409593B (zh) * 2022-01-20 2024-02-23 上海泾维化工科技有限公司 一种2-氨基-5-甲基吡啶的制备方法

Also Published As

Publication number Publication date
JPS58208266A (ja) 1983-12-03
US4386209A (en) 1983-05-31

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