JPH0346467B2 - - Google Patents

Info

Publication number
JPH0346467B2
JPH0346467B2 JP56015114A JP1511481A JPH0346467B2 JP H0346467 B2 JPH0346467 B2 JP H0346467B2 JP 56015114 A JP56015114 A JP 56015114A JP 1511481 A JP1511481 A JP 1511481A JP H0346467 B2 JPH0346467 B2 JP H0346467B2
Authority
JP
Japan
Prior art keywords
group
alkyl
formula
hydrogen
halogen
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
JP56015114A
Other languages
English (en)
Japanese (ja)
Other versions
JPS56125374A (en
Inventor
Omodei Sare Amedeo
Toia Emirio
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Gruppo Lepetit SpA
Original Assignee
Lepetit SpA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit SpA filed Critical Lepetit SpA
Publication of JPS56125374A publication Critical patent/JPS56125374A/ja
Publication of JPH0346467B2 publication Critical patent/JPH0346467B2/ja
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
    • C07D263/60—Naphthoxazoles; Hydrogenated naphthoxazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP1511481A 1980-02-08 1981-02-05 Novel naphthoimidazole and naphthoxazole derivatives, their manufacture and their use as medicinal goods Granted JPS56125374A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8004311 1980-02-08
AU71881/81A AU537378B2 (en) 1980-02-08 1981-06-16 Naphthimidazole and naphthoxazoles

Publications (2)

Publication Number Publication Date
JPS56125374A JPS56125374A (en) 1981-10-01
JPH0346467B2 true JPH0346467B2 (en, 2012) 1991-07-16

Family

ID=25636747

Family Applications (1)

Application Number Title Priority Date Filing Date
JP1511481A Granted JPS56125374A (en) 1980-02-08 1981-02-05 Novel naphthoimidazole and naphthoxazole derivatives, their manufacture and their use as medicinal goods

Country Status (5)

Country Link
US (2) US4360674A (en, 2012)
EP (1) EP0034249B1 (en, 2012)
JP (1) JPS56125374A (en, 2012)
AU (1) AU537378B2 (en, 2012)
CA (1) CA1165762A (en, 2012)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0034249B1 (en) * 1980-02-08 1984-10-24 Gruppo Lepetit S.P.A. New naphthimidazole and naphthoxazole derivatives, their preparation, and their use in pharmaceuticals
US4368201A (en) * 1981-07-20 1983-01-11 Usv Pharmaceutical Corporation Tetrahydronaphthoxazoles
GB8403141D0 (en) * 1984-02-07 1984-03-14 Lepetit Spa Imidazole derivatives
IL97144A (en) * 1990-02-27 1994-11-28 Erba Carlo Spa Substituted 1-(alkoxy-iminoalkyl)imidazole derivatives, their preparation and pharmaceutical compositions containing them
US5750542A (en) 1993-09-28 1998-05-12 Pfizer Benzisoxazole and benzisothizole derivatives as cholinesterase inhibitors
AU4632893A (en) * 1992-07-29 1994-03-03 Agouron Pharmaceuticals, Inc. Antiproliferative tricyclic compounds
US5714498A (en) * 1993-03-18 1998-02-03 Merck, Sharp, & Dohme, Ltd. Benzimidazole derivatives
US5773616A (en) * 1995-02-15 1998-06-30 Neurogen Corporation Certain bridged 4-phenyl-2-aminomethylimidazoles; new dopamine receptor subtype specific ligands
EP0809641A1 (en) * 1995-02-15 1997-12-03 Neurogen Corporation Certain bridged 4-phenyl-2-aminomethylimidazoles; new dopamine receptor subtype specific ligands
WO2009125809A1 (ja) * 2008-04-11 2009-10-15 第一三共株式会社 ピペリジン誘導体

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2964567D1 (en) * 1978-12-21 1983-02-24 Lepetit Spa New 3h-naphtho(1,2-d)imidazoles, processes for preparing them, compounds for use as antiinflammatory and antimicrobial agents and compositions for that use containing them
US4173634A (en) * 1979-02-23 1979-11-06 E. R. Squibb & Sons, Inc. Basically-substituted tricyclic pyrazoles useful as antiinflammatory agents
EP0034249B1 (en) * 1980-02-08 1984-10-24 Gruppo Lepetit S.P.A. New naphthimidazole and naphthoxazole derivatives, their preparation, and their use in pharmaceuticals

Also Published As

Publication number Publication date
EP0034249B1 (en) 1984-10-24
US4461894A (en) 1984-07-24
AU7188181A (en) 1982-12-23
EP0034249A2 (en) 1981-08-26
JPS56125374A (en) 1981-10-01
CA1165762A (en) 1984-04-17
US4360674A (en) 1982-11-23
EP0034249A3 (en) 1982-02-24
AU537378B2 (en) 1984-06-21

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