JP7649290B2 - ３－ブロモ－４，５－ジヒドロ－１ｈ－ピラゾールのカルボン酸誘導体の調製方法 - Google Patents

３－ブロモ－４，５－ジヒドロ－１ｈ－ピラゾールのカルボン酸誘導体の調製方法 Download PDF

Info

Publication number
JP7649290B2
JP7649290B2 JP2022509011A JP2022509011A JP7649290B2 JP 7649290 B2 JP7649290 B2 JP 7649290B2 JP 2022509011 A JP2022509011 A JP 2022509011A JP 2022509011 A JP2022509011 A JP 2022509011A JP 7649290 B2 JP7649290 B2 JP 7649290B2
Authority
JP
Japan
Prior art keywords
formula
compound
alkyl
pyrazole
ethyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
JP2022509011A
Other languages
English (en)
Japanese (ja)
Other versions
JP2022545773A5 (enExample
JP2022545773A (ja
Inventor
ジャンファ・マオ
ジンイー・マー
ドゥンジィエ・パン
チュンヤン・フゥオ
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
FMC Corp
Original Assignee
FMC Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by FMC Corp filed Critical FMC Corp
Publication of JP2022545773A publication Critical patent/JP2022545773A/ja
Publication of JP2022545773A5 publication Critical patent/JP2022545773A5/ja
Application granted granted Critical
Publication of JP7649290B2 publication Critical patent/JP7649290B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2022509011A 2019-08-19 2020-08-19 ３－ブロモ－４，５－ジヒドロ－１ｈ－ピラゾールのカルボン酸誘導体の調製方法 Active JP7649290B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201962888667P 2019-08-19 2019-08-19
US62/888,667 2019-08-19
US201962890154P 2019-08-22 2019-08-22
US62/890,154 2019-08-22
PCT/US2020/046947 WO2021034904A1 (en) 2019-08-19 2020-08-19 Process for the preparation of carboxylic acid derivatives of 3-bromo-4,5-dihydro-1h-pyrazoles

Publications (3)

Publication Number Publication Date
JP2022545773A JP2022545773A (ja) 2022-10-31
JP2022545773A5 JP2022545773A5 (enExample) 2023-08-10
JP7649290B2 true JP7649290B2 (ja) 2025-03-19

Family

ID=72340418

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022509011A Active JP7649290B2 (ja) 2019-08-19 2020-08-19 ３－ブロモ－４，５－ジヒドロ－１ｈ－ピラゾールのカルボン酸誘導体の調製方法

Country Status (15)

Country Link
US (1) US20220289706A1 (enExample)
EP (1) EP4017847B1 (enExample)
JP (1) JP7649290B2 (enExample)
KR (1) KR20220047992A (enExample)
CN (1) CN114341126B (enExample)
AU (1) AU2020333761A1 (enExample)
BR (1) BR112022002990A2 (enExample)
ES (1) ES3057453T3 (enExample)
IL (1) IL290505B1 (enExample)
MX (1) MX2022002043A (enExample)
PL (1) PL4017847T3 (enExample)
RS (1) RS67525B1 (enExample)
TW (1) TWI878337B (enExample)
WO (1) WO2021034904A1 (enExample)
ZA (1) ZA202202129B (enExample)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202342443A (zh) * 2022-01-31 2023-11-01 美商富曼西公司 用於製備３－溴－１－（３－氯吡啶－２－基）－４，５－二氫－１ｈ－吡唑－５－甲酸乙酯之方法

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005502658A (ja) 2001-08-13 2005-01-27 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 置換ジヒドロ３−ハロ−１ｈ−ピラゾール−５−カルボキシレート、それらの製造および使用
CN102399211A (zh) 2011-07-29 2012-04-04 山东永农作物科学有限公司 3-溴-1-(3-氯-2-吡啶基)-4,5-二氢-1h-吡唑-5-甲酸酯的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5291862A (en) * 1976-01-30 1977-08-02 Fuji Photo Film Co Ltd Preparation of 3-n-monosubstituted-amino-4-substituted-pyrazolone
US4730062A (en) * 1985-04-19 1988-03-08 Fmc Corporation Process of preparation of tetrafluoro 2,3-dihydrobenzofurans
ES2325757B1 (es) * 2005-07-15 2010-04-19 Laboratorios Del Dr. Esteve, S.A. Compuestos de pirazolina tiocarbonilsustituidos, su preparacion y uso como moduladores de cb1.
CN100582096C (zh) * 2008-03-04 2010-01-20 太原理工大学 一种发黄绿光的吡唑啉衍生物的合成方法
CN101550134B (zh) * 2008-04-01 2011-04-27 中国中化股份有限公司 一种制备2-[1h-吡唑-5-基]-4h-3,1-苯并噁嗪-4-酮类化合物的方法
EP2955176B1 (de) * 2010-06-15 2017-12-06 Bayer Intellectual Property GmbH Zusammensetzung enthaltend kristalline modifikation b von (3-chloropyridin-2-yl)-n-[4-cyano-2-methyl-6-(methylcarbamoyl)phenyl]-3-([5-(trifluormethyl)-2h- tetrazol-2-yl]methyl)-1h-pyrazol-5-carboxamid und ihre verwendung
RS54643B1 (sr) * 2010-06-29 2016-08-31 Fmc Corporation Derivat 6-acil-1,2,4-triazin-3,5-diona i herbicidi
CN102603752A (zh) * 2012-03-01 2012-07-25 健雄职业技术学院 7-溴吡唑并[1,5-a]嘧啶-3-甲酸酯类化合物、合成方法及应用
HUE064783T2 (hu) * 2017-09-28 2024-04-28 Albemarle Corp Brómozott égésgátló és alkalmazása poliuretán habokban

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005502658A (ja) 2001-08-13 2005-01-27 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー 置換ジヒドロ３−ハロ−１ｈ−ピラゾール−５−カルボキシレート、それらの製造および使用
CN102399211A (zh) 2011-07-29 2012-04-04 山东永农作物科学有限公司 3-溴-1-(3-氯-2-吡啶基)-4,5-二氢-1h-吡唑-5-甲酸酯的制备方法

Also Published As

Publication number Publication date
TW202112762A (zh) 2021-04-01
PL4017847T3 (pl) 2026-02-23
EP4017847B1 (en) 2025-10-01
AU2020333761A1 (en) 2022-03-03
IL290505A (en) 2022-04-01
CN114341126A (zh) 2022-04-12
MX2022002043A (es) 2022-05-11
JP2022545773A (ja) 2022-10-31
US20220289706A1 (en) 2022-09-15
ZA202202129B (en) 2025-06-25
BR112022002990A2 (pt) 2022-07-19
EP4017847C0 (en) 2025-10-01
TWI878337B (zh) 2025-04-01
EP4017847A1 (en) 2022-06-29
KR20220047992A (ko) 2022-04-19
ES3057453T3 (en) 2026-03-02
CN114341126B (zh) 2025-04-25
WO2021034904A1 (en) 2021-02-25
RS67525B1 (sr) 2026-01-30
IL290505B1 (en) 2026-02-01

Similar Documents

Publication Publication Date Title
EP1417200B1 (en) Substituted 1h-dihydropyrazoles, their preparation and use
JP4564748B2 (ja) 置換ジヒドロ３−ハロ−１ｈ−ピラゾール−５−カルボキシレート、それらの製造および使用
JP4633462B2 (ja) ３−ハロ−４，５−ジヒドロ−１ｈ−ピラゾールの製造方法
AU2002355952A1 (en) Substituted dihydro 3-halo-1H-pyrazole-5-carboxylates their preparation and use
JP4750019B2 (ja) ２−置換−５−オキソ−３−ピラゾリジンカルボキシレートの製造および使用
JP7649290B2 (ja) ３－ブロモ－４，５－ジヒドロ－１ｈ－ピラゾールのカルボン酸誘導体の調製方法
EP1773783B1 (fr) Procede de preparation de derives n-piperidino-1,5-diphenylpyrazole-3-carboxamide
AU2017258665A1 (en) Process for the preparation of herbicidal compounds
EA051533B1 (ru) Способ получения производных карбоновых кислот 3-бром-4,5-дигидро-1h-пиразолов
AU2021205515A1 (en) Methods for the preparation of Ethyl 3-bromo-1-(3-chloropyridin-2-yl)-1H-pyrazole-5-carboxylate
JP2025503256A (ja) エチル３－ブロモ－１－（３－クロロピリジン－２－イル）－４，５－ジヒドロ－１ｈ－ピラゾール－５－カルボキシラートの調製の方法
EP1944304B1 (en) Substituted 1h-dihydropyrazoles, their preparation and use
KR101815001B1 (ko) 고 입체순도를 갖는 4-치환된-5-원고리-설파미데이트-5-포스포네이트 화합물 및 이의 제조방법
EP1113004A2 (en) Intermediates for producing 3-(substituted phenyl)-5-(thienyl or furyl)-1,2,4-triazole compounds

Legal Events

Date Code Title Description
A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20230802

A621 Written request for application examination

Free format text: JAPANESE INTERMEDIATE CODE: A621

Effective date: 20230802

A977 Report on retrieval

Free format text: JAPANESE INTERMEDIATE CODE: A971007

Effective date: 20240718

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20240723

A601 Written request for extension of time

Free format text: JAPANESE INTERMEDIATE CODE: A601

Effective date: 20241023

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20250121

TRDD Decision of grant or rejection written
A01 Written decision to grant a patent or to grant a registration (utility model)

Free format text: JAPANESE INTERMEDIATE CODE: A01

Effective date: 20250212

A61 First payment of annual fees (during grant procedure)

Free format text: JAPANESE INTERMEDIATE CODE: A61

Effective date: 20250307

R150 Certificate of patent or registration of utility model

Ref document number: 7649290

Country of ref document: JP

Free format text: JAPANESE INTERMEDIATE CODE: R150

S111 Request for change of ownership or part of ownership

Free format text: JAPANESE INTERMEDIATE CODE: R313117

R350 Written notification of registration of transfer

Free format text: JAPANESE INTERMEDIATE CODE: R350