JP7394059B2 - 抗寄生生物性ポアオン組成物 - Google Patents

抗寄生生物性ポアオン組成物 Download PDF

Info

Publication number
JP7394059B2
JP7394059B2 JP2020533625A JP2020533625A JP7394059B2 JP 7394059 B2 JP7394059 B2 JP 7394059B2 JP 2020533625 A JP2020533625 A JP 2020533625A JP 2020533625 A JP2020533625 A JP 2020533625A JP 7394059 B2 JP7394059 B2 JP 7394059B2
Authority
JP
Japan
Prior art keywords
composition
compositions
animal
pour
isoxazoline
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
JP2020533625A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021507891A (ja
Inventor
シーハン,ジョン・ジェラルド
フリーホーフ,キース
フロシュライ-シゴニヤルト,アニー
Original Assignee
インターベット インターナショナル ベー. フェー.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=64949294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=JP7394059(B2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by インターベット インターナショナル ベー. フェー. filed Critical インターベット インターナショナル ベー. フェー.
Publication of JP2021507891A publication Critical patent/JP2021507891A/ja
Priority to JP2023132324A priority Critical patent/JP7627312B2/ja
Application granted granted Critical
Publication of JP7394059B2 publication Critical patent/JP7394059B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Images

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/045Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A61K31/05Phenols
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/22Heterocyclic compounds, e.g. ascorbic acid, tocopherol or pyrrolidones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • A61K9/0017Non-human animal skin, e.g. pour-on, spot-on
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A40/00Adaptation technologies in agriculture, forestry, livestock or agroalimentary production
    • Y02A40/70Adaptation technologies in agriculture, forestry, livestock or agroalimentary production in livestock or poultry

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Zoology (AREA)
  • Dermatology (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Environmental Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
JP2020533625A 2017-12-21 2018-12-21 抗寄生生物性ポアオン組成物 Active JP7394059B2 (ja)

Priority Applications (1)

Application Number Priority Date Filing Date Title
JP2023132324A JP7627312B2 (ja) 2017-12-21 2023-08-15 抗寄生生物性ポアオン組成物

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201762608760P 2017-12-21 2017-12-21
US62/608,760 2017-12-21
PCT/EP2018/086558 WO2019122324A1 (en) 2017-12-21 2018-12-21 Antiparasitic pour-on compositions

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2023132324A Division JP7627312B2 (ja) 2017-12-21 2023-08-15 抗寄生生物性ポアオン組成物

Publications (2)

Publication Number Publication Date
JP2021507891A JP2021507891A (ja) 2021-02-25
JP7394059B2 true JP7394059B2 (ja) 2023-12-07

Family

ID=64949294

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2020533625A Active JP7394059B2 (ja) 2017-12-21 2018-12-21 抗寄生生物性ポアオン組成物
JP2023132324A Active JP7627312B2 (ja) 2017-12-21 2023-08-15 抗寄生生物性ポアオン組成物

Family Applications After (1)

Application Number Title Priority Date Filing Date
JP2023132324A Active JP7627312B2 (ja) 2017-12-21 2023-08-15 抗寄生生物性ポアオン組成物

Country Status (9)

Country Link
US (1) US12390450B2 (https=)
EP (2) EP4559482A3 (https=)
JP (2) JP7394059B2 (https=)
AR (1) AR113997A1 (https=)
AU (2) AU2018386568B2 (https=)
CA (1) CA3085896A1 (https=)
ES (1) ES3018480T3 (https=)
MX (2) MX2020006512A (https=)
WO (1) WO2019122324A1 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2021122515A1 (en) * 2019-12-16 2021-06-24 Intervet International B.V. Parasite control in ruminants
EP4075981A1 (en) * 2019-12-16 2022-10-26 Intervet International B.V. Composition for lice control
KR20230043904A (ko) 2020-07-24 2023-03-31 엘랑코 유에스 인코포레이티드 이속사졸린 화합물 및 이의 중간체의 제조 공정
CN116744917A (zh) 2020-09-04 2023-09-12 礼蓝美国公司 适口调配物
EP4430947A1 (en) * 2023-03-17 2024-09-18 Przedsiebiorstwo Wielobranzowe "Vet-Agro" Sp. Z O.O. Therapeutic use of isoxazoline compounds, composition of isoxazoline compounds and kit for therapeutic use
CN117617236A (zh) * 2023-11-17 2024-03-01 中国农业大学 三唑类杀菌剂绿色乳油及其制备方法
WO2025191150A2 (en) 2024-03-15 2025-09-18 Krka, D.D., Novo Mesto Stable isoxazoline formulation for topical application to the skin
CN120053434B (zh) * 2025-02-28 2025-12-23 湖南尚成生物科技有限公司 一种弗雷拉纳滴剂及其制备方法
CN120531675A (zh) * 2025-06-11 2025-08-26 湖南尚成生物科技有限公司 一种氟雷拉纳莫昔克丁滴剂及其制备方法

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009156369A1 (en) 2008-06-24 2009-12-30 Intervet International B.V. Pharmaceutical transdermal compositions and method for treating inflammation in cattle
JP2014504586A (ja) 2010-12-27 2014-02-24 インターベツト・インターナシヨナル・ベー・ベー 経表面局所イソオキサゾリン製剤

Family Cites Families (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN101768129B (zh) 2004-03-05 2012-05-23 日产化学工业株式会社 异*唑啉取代苯甲酰胺化合物的制备中间体
TWI412322B (zh) 2005-12-30 2013-10-21 Du Pont 控制無脊椎害蟲之異唑啉
MY146638A (en) 2007-04-10 2012-09-14 Bayer Cropscience Ag Insecticidal aryl isoxazoline derivatives
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
KR101769728B1 (ko) 2007-06-27 2017-08-18 이 아이 듀폰 디 네모아 앤드 캄파니 동물 해충 방제 방법
TWI556741B (zh) 2007-08-17 2016-11-11 英特威特國際股份有限公司 異唑啉組成物及其作為抗寄生蟲藥上的應用
WO2009070687A1 (en) * 2007-11-26 2009-06-04 Merial Limited Solvent systems for pour-on formulations for combating parasites
TWI411395B (zh) 2007-12-24 2013-10-11 Syngenta Participations Ag 殺蟲化合物
US8377942B2 (en) 2008-12-18 2013-02-19 Novartis Ag Isoxazolines derivatives and their use as pesticide
HUE015568T4 (en) 2008-12-19 2017-10-30 Elanco Tiergesundheit Ag Isoxazoline derivatives and their use as pesticides
RS54772B1 (sr) 2009-12-17 2016-10-31 Merial Sas Antiparazitska jedinjenja dihidroazola i kompozicije koje ih sadrže
EP2556060A1 (en) 2010-04-08 2013-02-13 Ah Usa 42 Llc Substituted 3,5- diphenyl-isoxazoline derivatives as insecticides and acaricides
NZ611474A (en) 2010-12-27 2015-08-28 Intervet Int Bv Topical localized isoxazoline formulation comprising glycofurol
WO2012155352A1 (en) 2011-05-19 2012-11-22 Eli Lilly And Company Dihydroisoxazole compounds, parasiticidal uses and formulations thereof
RS58417B1 (sr) 2011-09-12 2019-04-30 Merial Inc Paraziticidne kompozicije koje sadrže izoksazolinsko aktivno sredstvo, postupci i upotrebe povezane sa njima
WO2013150055A1 (en) 2012-04-04 2013-10-10 Intervet International B.V. Solid oral pharmaceutical compositions for isoxazoline compounds
DK2892347T3 (da) 2012-09-07 2019-09-30 Zoetis Services Llc Spirocykliske parasiticide isoxazolin-kombinationer
NZ630169A (en) * 2013-02-27 2017-07-28 Laurie Robert Batt Anhydrous transdermal formulations
WO2014189837A1 (en) 2013-05-20 2014-11-27 Zoetis Llc Long-acting spiro-isoxazoline antiparasitic compositions
AU2014324837B2 (en) 2013-09-30 2019-01-17 Zoetis Services Llc Long-acting spiro-isoxazoline formulations
US9371293B2 (en) 2013-10-25 2016-06-21 Sumitomo Chemical Company, Limited Isoxazoline compound composition
WO2015066277A1 (en) 2013-11-01 2015-05-07 Merial Limited Antiparisitic and pesticidal isoxazoline compounds

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2009156369A1 (en) 2008-06-24 2009-12-30 Intervet International B.V. Pharmaceutical transdermal compositions and method for treating inflammation in cattle
JP2014504586A (ja) 2010-12-27 2014-02-24 インターベツト・インターナシヨナル・ベー・ベー 経表面局所イソオキサゾリン製剤

Also Published As

Publication number Publication date
MX2023010368A (es) 2023-09-12
BR112020012465A2 (pt) 2020-11-24
AU2018386568A1 (en) 2020-06-11
AU2018386568B2 (en) 2024-02-22
AR113997A1 (es) 2020-07-08
WO2019122324A1 (en) 2019-06-27
AU2024203397A1 (en) 2024-06-06
EP4559482A2 (en) 2025-05-28
EP4559482A3 (en) 2025-07-30
EP3727375B1 (en) 2025-03-19
MX2020006512A (es) 2020-09-07
EP3727375A1 (en) 2020-10-28
US20200390748A1 (en) 2020-12-17
JP2023154054A (ja) 2023-10-18
JP2021507891A (ja) 2021-02-25
RU2020123896A (ru) 2022-01-21
ES3018480T3 (es) 2025-05-16
CA3085896A1 (en) 2019-06-27
US12390450B2 (en) 2025-08-19
JP7627312B2 (ja) 2025-02-05

Similar Documents

Publication Publication Date Title
JP7627312B2 (ja) 抗寄生生物性ポアオン組成物
RU2602189C2 (ru) Изоксазолиновый состав, содержащий гликофурол для наружного и местного применения
KR102606187B1 (ko) 주사가능한 이속사졸린 제약 조성물 및 그의 기생충 침입에 대한 용도
AU2020268618B2 (en) Injectable pharmaceutical compositions and uses thereof
JP7578752B2 (ja) 注射可能なイソオキサゾリン医薬組成物および寄生生物の寄生に対するそれらの使用
JP2006522154A (ja) 動物用駆虫局所製剤
JP7274479B2 (ja) 寄生虫の寄生を治療するためのモキシデクチンを含有する組成物
RU2802299C2 (ru) Противопаразитарные композиции для применения путем обливания
AU2006100661A4 (en) Topical formulation
RU2856883C2 (ru) Фармацевтические композиции для инъекций и использование таковых
BR112020012465B1 (pt) Composição pour-on veterinária líquida para uso na proteção e no tratamento de infestações por parasitas de animais compreendendo fluralaner e uso deste
RU2829447C2 (ru) Фармацевтические композиции для инъекций и использование таковых
RU2799591C2 (ru) Инъекционные изоксазолиновые фармацевтические композиции и их применение

Legal Events

Date Code Title Description
A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20211214

A621 Written request for application examination

Free format text: JAPANESE INTERMEDIATE CODE: A621

Effective date: 20211214

A131 Notification of reasons for refusal

Free format text: JAPANESE INTERMEDIATE CODE: A131

Effective date: 20221213

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20230309

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A821

Effective date: 20230309

A02 Decision of refusal

Free format text: JAPANESE INTERMEDIATE CODE: A02

Effective date: 20230418

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A523

Effective date: 20230815

A521 Request for written amendment filed

Free format text: JAPANESE INTERMEDIATE CODE: A821

Effective date: 20230926

A911 Transfer to examiner for re-examination before appeal (zenchi)

Free format text: JAPANESE INTERMEDIATE CODE: A911

Effective date: 20231016

TRDD Decision of grant or rejection written
A01 Written decision to grant a patent or to grant a registration (utility model)

Free format text: JAPANESE INTERMEDIATE CODE: A01

Effective date: 20231114

A61 First payment of annual fees (during grant procedure)

Free format text: JAPANESE INTERMEDIATE CODE: A61

Effective date: 20231127

R150 Certificate of patent or registration of utility model

Ref document number: 7394059

Country of ref document: JP

Free format text: JAPANESE INTERMEDIATE CODE: R150