JP7346439B2 - Ｏｘ２ｒ化合物 - Google Patents

Ｏｘ２ｒ化合物 Download PDF

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JP7346439B2
JP7346439B2 JP2020552805A JP2020552805A JP7346439B2 JP 7346439 B2 JP7346439 B2 JP 7346439B2 JP 2020552805 A JP2020552805 A JP 2020552805A JP 2020552805 A JP2020552805 A JP 2020552805A JP 7346439 B2 JP7346439 B2 JP 7346439B2
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alkylene
alkyl
optionally substituted
haloalkyl
alkoxy
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JPWO2019191327A5 (https=
JP2021519776A (ja
JP2021519776A5 (https=
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ブラバンダー，ジェフ デ
ローゼンバウム，ダニエル
リャン，キレン
ワン，ウェンティアン
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University of Texas System
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University of Texas System
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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • C07D487/10—Spiro-condensed systems

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US12006330B2 (en) 2020-12-21 2024-06-11 Alkermes, Inc. Substituted macrocyclic compounds and related methods of treatment
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