JP7090551B2 - 眼状態の治療方法 - Google Patents

眼状態の治療方法 Download PDF

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Publication number
JP7090551B2
JP7090551B2 JP2018553080A JP2018553080A JP7090551B2 JP 7090551 B2 JP7090551 B2 JP 7090551B2 JP 2018553080 A JP2018553080 A JP 2018553080A JP 2018553080 A JP2018553080 A JP 2018553080A JP 7090551 B2 JP7090551 B2 JP 7090551B2
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JP2019513759A (ja
JP2019513759A5 (OSRAM
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ダグラス マイケル ジュニア アッカーマン
ジェームズ ルーディン
ケネス ジェイ． マンデル
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オイスター ポイント ファーマ インコーポレイテッド
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Priority to JP2022095460A priority Critical patent/JP2022120125A/ja
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13—Cyclosporins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0043—Nose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/04—Artificial tears; Irrigation solutions

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Ophthalmology & Optometry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Otolaryngology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP2018553080A 2016-04-07 2017-04-06 眼状態の治療方法 Active JP7090551B2 (ja)

Priority Applications (2)

Application Number Priority Date Filing Date Title
JP2022095460A JP2022120125A (ja) 2016-04-07 2022-06-14 眼状態の治療方法
JP2024086805A JP2024103594A (ja) 2016-04-07 2024-05-29 眼状態の治療方法

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201662319648P 2016-04-07 2016-04-07
US62/319,648 2016-04-07
PCT/US2017/026385 WO2017177024A1 (en) 2016-04-07 2017-04-06 Methods of treating ocular conditions

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2022095460A Division JP2022120125A (ja) 2016-04-07 2022-06-14 眼状態の治療方法

Publications (3)

Publication Number Publication Date
JP2019513759A JP2019513759A (ja) 2019-05-30
JP2019513759A5 JP2019513759A5 (OSRAM) 2020-05-14
JP7090551B2 true JP7090551B2 (ja) 2022-06-24

Family

ID=58549326

Family Applications (3)

Application Number Title Priority Date Filing Date
JP2018553080A Active JP7090551B2 (ja) 2016-04-07 2017-04-06 眼状態の治療方法
JP2022095460A Pending JP2022120125A (ja) 2016-04-07 2022-06-14 眼状態の治療方法
JP2024086805A Pending JP2024103594A (ja) 2016-04-07 2024-05-29 眼状態の治療方法

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Application Number Title Priority Date Filing Date
JP2022095460A Pending JP2022120125A (ja) 2016-04-07 2022-06-14 眼状態の治療方法
JP2024086805A Pending JP2024103594A (ja) 2016-04-07 2024-05-29 眼状態の治療方法

Country Status (19)

Country Link
US (3) US10709707B2 (OSRAM)
EP (2) EP3970724A1 (OSRAM)
JP (3) JP7090551B2 (OSRAM)
KR (2) KR102512777B1 (OSRAM)
CN (3) CN114432313A (OSRAM)
AU (1) AU2017248276B2 (OSRAM)
DK (1) DK3439661T3 (OSRAM)
EA (1) EA201892265A1 (OSRAM)
ES (1) ES2893126T3 (OSRAM)
IL (3) IL299204A (OSRAM)
MX (2) MX385698B (OSRAM)
MY (1) MY199237A (OSRAM)
NZ (1) NZ746468A (OSRAM)
PH (1) PH12018502154A1 (OSRAM)
PT (1) PT3439661T (OSRAM)
SG (1) SG11201808650QA (OSRAM)
TW (2) TWI876258B (OSRAM)
WO (1) WO2017177024A1 (OSRAM)
ZA (1) ZA201807438B (OSRAM)

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US9145396B2 (en) 2008-12-01 2015-09-29 Targacept, Inc. Synthesis and novel salt forms of (R)-5-((E)-2-pyrrolidin-3ylvinyl)pyrimidine
EP3848028B9 (en) 2014-10-20 2024-10-16 Oyster Point Pharma, Inc. Methods of treating ocular conditions
DK3439661T3 (da) 2016-04-07 2021-10-18 Oyster Point Pharma Inc Fremgangsmåder til behandling af øjenlidelser
TW202019424A (zh) 2018-07-10 2020-06-01 美商奧伊斯特普安生物製藥公司 治療眼部症狀之方法
EP3820443A1 (en) 2018-07-10 2021-05-19 Oyster Point Pharma, Inc. Combinations of positive allosteric modulators and nicotinic acetylcholine receptor agonists for treating ocular conditions
ES3039903T3 (en) * 2020-04-28 2025-10-27 Oyster Point Pharma Inc Local administration of nicotinic acetylcholine receptor agonists for the inhibition of coronavirus infections
IL308372A (en) * 2021-05-07 2024-01-01 Oyster Point Pharma Inc Co-therapy using a vector and a nicotinic agonist
WO2026080563A1 (en) 2024-10-09 2026-04-16 Oyster Point Pharma, Inc. Simpinicline oral formations and use thereof

Citations (3)

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Publication number Priority date Publication date Assignee Title
JP2003531168A (ja) 2000-04-21 2003-10-21 インスパイアー ファーマシューティカルズ，インコーポレイティド ニコチン・アセチルコリン受容体アゴニストによるドライ・アイ疾患の治療方法
JP2012510471A (ja) 2008-12-01 2012-05-10 ターガセプト，インコーポレイテッド （ｒ）−５−（（ｅ）−２−（ピロリジン−３−イルビニル）ピリミジンの合成および新規の塩形態
JP2017531044A (ja) 2014-10-20 2017-10-19 オイスター ポイント ファーマ インコーポレイテッド 眼の病状の治療方法

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WO2004039366A1 (en) 2002-11-01 2004-05-13 Pharmacia & Upjohn Company Llc Nicotinic acetylcholine agonists in the treatment of glaucoma and retinal neuropathy
US7098331B2 (en) 2003-03-05 2006-08-29 Targacept, Inc. Arylvinylazacycloalkane compounds and methods of preparation and use thereof
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WO2006040680A1 (en) 2004-10-15 2006-04-20 Pfizer Products Inc. Compositions and methods for intranasal, buccal, sublingual and pulmonary delivery of varenicline
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Publication number Priority date Publication date Assignee Title
JP2003531168A (ja) 2000-04-21 2003-10-21 インスパイアー ファーマシューティカルズ，インコーポレイティド ニコチン・アセチルコリン受容体アゴニストによるドライ・アイ疾患の治療方法
JP2012510471A (ja) 2008-12-01 2012-05-10 ターガセプト，インコーポレイテッド （ｒ）−５−（（ｅ）−２−（ピロリジン−３−イルビニル）ピリミジンの合成および新規の塩形態
JP2017531044A (ja) 2014-10-20 2017-10-19 オイスター ポイント ファーマ インコーポレイテッド 眼の病状の治療方法

Also Published As

Publication number Publication date
ES2893126T3 (es) 2022-02-08
KR102512777B1 (ko) 2023-03-23
AU2017248276B2 (en) 2023-07-13
IL299204A (en) 2023-02-01
IL262102B (en) 2022-03-01
BR112018070497A2 (pt) 2019-01-29
CN109310692B (zh) 2022-01-25
TW201737917A (zh) 2017-11-01
SG11201808650QA (en) 2018-10-30
WO2017177024A8 (en) 2018-11-08
AU2017248276A1 (en) 2018-11-22
JP2019513759A (ja) 2019-05-30
MX385698B (es) 2025-03-18
IL262102A (en) 2018-11-29
TW202320785A (zh) 2023-06-01
CN114432313A (zh) 2022-05-06
KR20230010813A (ko) 2023-01-19
EP3439661B1 (en) 2021-08-04
JP2022120125A (ja) 2022-08-17
ZA201807438B (en) 2024-09-25
US20200345734A1 (en) 2020-11-05
DK3439661T3 (da) 2021-10-18
JP2024103594A (ja) 2024-08-01
PT3439661T (pt) 2021-09-30
PH12018502154A1 (en) 2019-07-08
US10709707B2 (en) 2020-07-14
EP3439661A1 (en) 2019-02-13
MX2018012230A (es) 2019-03-28
ES2893126T8 (es) 2022-05-23
US20250000861A1 (en) 2025-01-02
US20190201397A1 (en) 2019-07-04
WO2017177024A1 (en) 2017-10-12
KR20190005859A (ko) 2019-01-16
CN109310692A (zh) 2019-02-05
MY199237A (en) 2023-10-22
IL290069B2 (en) 2023-05-01
KR102485299B1 (ko) 2023-01-06
IL290069A (en) 2022-03-01
TWI876258B (zh) 2025-03-11
CN114533737B (zh) 2024-05-31
MX2021010399A (es) 2022-01-18
NZ746468A (en) 2023-06-30
IL290069B1 (en) 2023-01-01
TWI790997B (zh) 2023-02-01
CN114533737A (zh) 2022-05-27
EA201892265A1 (ru) 2019-04-30
NZ785093A (en) 2024-07-05
EP3970724A1 (en) 2022-03-23
CA3020170A1 (en) 2017-10-12

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