JP6900050B2 - 去勢抵抗性前立腺がんの処置のためのアンドロゲン受容体の核移行の低分子阻害剤 - Google Patents

去勢抵抗性前立腺がんの処置のためのアンドロゲン受容体の核移行の低分子阻害剤 Download PDF

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JP6900050B2
JP6900050B2 JP2018549435A JP2018549435A JP6900050B2 JP 6900050 B2 JP6900050 B2 JP 6900050B2 JP 2018549435 A JP2018549435 A JP 2018549435A JP 2018549435 A JP2018549435 A JP 2018549435A JP 6900050 B2 JP6900050 B2 JP 6900050B2
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mmol
substituted
phenyl
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JP2019512515A5 (enExample
JP2019512515A (ja
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ピーター ウィプフ，
ピーター ウィプフ，
ジェイムズ ケー． ジョンソン，
ジェイムズ ケー． ジョンソン，
エリン エム． スコダ，
エリン エム． スコダ，
ジェエル ビー． ネルソン，
ジェエル ビー． ネルソン，
ゾウ ワン，
ゾウ ワン，
セレン タイ，
セレン タイ，
ケイタ タクボ，
ケイタ タクボ，
ジョン ミリガン，
ジョン ミリガン，
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University of Pittsburgh
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University of Pittsburgh
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  • Plural Heterocyclic Compounds (AREA)
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JP2018549435A 2016-03-24 2017-03-24 去勢抵抗性前立腺がんの処置のためのアンドロゲン受容体の核移行の低分子阻害剤 Active JP6900050B2 (ja)

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US15/080,237 US20160257657A1 (en) 2013-09-20 2016-03-24 Small molecule inhibitors of the nuclear translocation of androgen receptor for the treatment of castration-resistant prostate cancer
PCT/US2017/024105 WO2017165822A1 (en) 2016-03-24 2017-03-24 Small molecule inhibitor of the nuclear translocation of androgen receptor for the treatment of castration-resistant prostate cancer

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CN111902401B (zh) * 2018-02-23 2023-06-13 北京泰德制药股份有限公司 受体抑制剂、包含其的药物组合物及其用途
CA3099739A1 (en) * 2018-05-14 2019-11-21 University Of Pittsburgh - Of The Commonwealth System Of Higher Education Small molecule inhibitors of the nuclear translocation of androgen receptor for the treatment of castration-resistant prostate cancer
CN109438297B (zh) * 2018-12-03 2021-05-14 昆明积大制药股份有限公司 雄激素受体拮抗剂、其制备方法及其应用
WO2020123670A1 (en) * 2018-12-11 2020-06-18 Arizona Board Of Regents On Behalf Of The University Of Arizona Small molecule inhibitors of the androgen receptor activity and/or expression and uses thereof
IL326597A (en) 2019-10-07 2026-04-01 Contineum Therapeutics Inc Muscarinic acetylcholine m1 receptor antagonists
US11752149B2 (en) 2019-12-02 2023-09-12 Pipeline Therapeutics, Inc. Muscarinic acetylcholine M1 receptor antagonists
US11945790B2 (en) * 2020-12-22 2024-04-02 Immunomolecular Therapeutics, Inc. Compounds and methods for treating autoimmune disorders by targeting HLA-DQ2

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US20160257657A1 (en) * 2013-09-20 2016-09-08 University Of Pittsburgh - Of The Commonwealth System Of Higher Education Small molecule inhibitors of the nuclear translocation of androgen receptor for the treatment of castration-resistant prostate cancer
CA2924527C (en) 2013-09-20 2022-07-12 University Of Pittsburgh - Of The Commonwealth System Of Higher Education Compounds for treating prostate cancer

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WO2017165822A8 (en) 2017-11-02
JP7125801B2 (ja) 2022-08-25
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