JP6063094B2 - 経皮送達を促進するためのペプチド - Google Patents
経皮送達を促進するためのペプチド Download PDFInfo
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- JP6063094B2 JP6063094B2 JP2016515955A JP2016515955A JP6063094B2 JP 6063094 B2 JP6063094 B2 JP 6063094B2 JP 2016515955 A JP2016515955 A JP 2016515955A JP 2016515955 A JP2016515955 A JP 2016515955A JP 6063094 B2 JP6063094 B2 JP 6063094B2
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Classifications
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- A61K38/00—Medicinal preparations containing peptides
- A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
- A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
- A61K38/22—Hormones
- A61K38/28—Insulins
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- A61K31/575—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of three or more carbon atoms, e.g. cholane, cholestane, ergosterol, sitosterol
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- A61K38/08—Peptides having 5 to 11 amino acids
- A61K38/09—Luteinising hormone-releasing hormone [LHRH], i.e. Gonadotropin-releasing hormone [GnRH]; Related peptides
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- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
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- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/42—Proteins; Polypeptides; Degradation products thereof; Derivatives thereof, e.g. albumin, gelatin or zein
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/64—Proteins; Peptides; Derivatives or degradation products thereof
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61L—METHODS OR APPARATUS FOR STERILISING MATERIALS OR OBJECTS IN GENERAL; DISINFECTION, STERILISATION OR DEODORISATION OF AIR; CHEMICAL ASPECTS OF BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES; MATERIALS FOR BANDAGES, DRESSINGS, ABSORBENT PADS OR SURGICAL ARTICLES
- A61L27/00—Materials for grafts or prostheses or for coating grafts or prostheses
- A61L27/14—Macromolecular materials
- A61L27/22—Polypeptides or derivatives thereof, e.g. degradation products
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- A—HUMAN NECESSITIES
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- A61P17/00—Drugs for dermatological disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/04—Immunostimulants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
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- A—HUMAN NECESSITIES
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- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/001—Preparations for care of the lips
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- A—HUMAN NECESSITIES
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- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q19/00—Preparations for care of the skin
- A61Q19/08—Anti-ageing preparations
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K2039/54—Medicinal preparations containing antigens or antibodies characterised by the route of administration
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- A—HUMAN NECESSITIES
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- A61K39/00—Medicinal preparations containing antigens or antibodies
- A61K2039/555—Medicinal preparations containing antigens or antibodies characterised by a specific combination antigen/adjuvant
- A61K2039/55511—Organic adjuvants
- A61K2039/55516—Proteins; Peptides
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K2039/60—Medicinal preparations containing antigens or antibodies characteristics by the carrier linked to the antigen
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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Landscapes
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- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Immunology (AREA)
- Dermatology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Gastroenterology & Hepatology (AREA)
- Endocrinology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
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- Oral & Maxillofacial Surgery (AREA)
- Transplantation (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Cosmetics (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
- Coloring Foods And Improving Nutritive Qualities (AREA)
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| US201361864964P | 2013-08-12 | 2013-08-12 | |
| US61/864,964 | 2013-08-12 | ||
| PCT/US2014/050683 WO2015023649A2 (en) | 2013-08-12 | 2014-08-12 | Peptides for enhancing transdermal delivery |
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| CA3087881A1 (en) | 2017-01-17 | 2018-07-26 | Michael David FORREST | Therapeutic inhibitors of the reverse mode of atp synthase |
| JP2020518653A (ja) * | 2017-02-07 | 2020-06-25 | マイオセプト インコーポレイティド | 局所製剤及び方法 |
| US12337000B2 (en) | 2017-07-13 | 2025-06-24 | Michael David FORREST | Therapeutic modulators of the reverse mode of ATP synthase |
| ES2998479T3 (en) | 2017-11-03 | 2025-02-20 | Skinqri Llc | Multi-factor hair growth formulation |
| CN108853720A (zh) * | 2018-05-16 | 2018-11-23 | 邱骅轩 | 一种用于美容领域的自适应透皮离子电渗法导入系统 |
| CN113286579A (zh) * | 2018-08-23 | 2021-08-20 | 埃里克·F·伯恩斯坦 | 应用抗vegf化合物和使用这类化合物治疗皮肤病的系统、装置和方法 |
| US20210000910A1 (en) | 2019-07-03 | 2021-01-07 | Jysk Skin Solutions Pte Ltd | Topical compositions |
| CN111166692A (zh) * | 2020-03-18 | 2020-05-19 | 深圳市百吉因生物科技有限公司 | 一种高保湿性组合物 |
| EP4281034A1 (en) | 2021-01-24 | 2023-11-29 | Forrest, Michael, David | Inhibitors of atp synthase - cosmetic and therapeutic uses |
| US11877848B2 (en) | 2021-11-08 | 2024-01-23 | Satio, Inc. | Dermal patch for collecting a physiological sample |
| US12053284B2 (en) | 2021-11-08 | 2024-08-06 | Satio, Inc. | Dermal patch for collecting a physiological sample |
| US12214346B2 (en) | 2021-10-13 | 2025-02-04 | Satio, Inc. | Dermal patch with a diagnostic test strip |
| US11964121B2 (en) | 2021-10-13 | 2024-04-23 | Satio, Inc. | Mono dose dermal patch for pharmaceutical delivery |
| US12023156B2 (en) | 2021-10-13 | 2024-07-02 | Satio, Inc. | Dermal patch for collecting a physiological sample |
| US12048543B2 (en) | 2021-11-08 | 2024-07-30 | Satio, Inc. | Dermal patch for collecting a physiological sample with removable vial |
| US12178979B2 (en) | 2021-10-13 | 2024-12-31 | Satio, Inc. | Dermal patch for delivering a pharmaceutical |
| US11452474B1 (en) | 2021-04-14 | 2022-09-27 | Satio, Inc. | Dual lever dermal patch system |
| US12303470B2 (en) | 2021-06-03 | 2025-05-20 | Skinqri, Llc | Method and composition for selective treatment of androgen receptors |
| US12083204B2 (en) | 2022-06-02 | 2024-09-10 | L'oreal | Topical composition for homeostatic delivery of nitric oxide and uses thereof |
| US12295372B1 (en) * | 2022-06-09 | 2025-05-13 | S. C. Johnson & Son, Inc. | Oil-based insect repellent composition |
| WO2024259323A2 (en) * | 2023-06-14 | 2024-12-19 | Scott Shapiro | Pharmaceutical compositions for targeted delivery of bioactive agents with improved bioavailability and methods of use |
| KR102666595B1 (ko) * | 2023-06-16 | 2024-05-16 | ㈜에스에이치랩 | 박테리오파지 유래 펩타이드를 포함하는 피부 주름 개선용 생분해성 고분자 필러 및 이의 제조방법 |
| CN116983223A (zh) * | 2023-09-01 | 2023-11-03 | 天津医科大学总医院 | 赖诺普利在促进皮肤弹力纤维再生中的应用 |
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| US4834979A (en) | 1981-06-29 | 1989-05-30 | Alza Corporation | Medical bandage for administering beneficial drug |
| US4472480A (en) | 1982-07-02 | 1984-09-18 | Minnesota Mining And Manufacturing Company | Low surface energy liner of perfluoropolyether |
| US4751087A (en) | 1985-04-19 | 1988-06-14 | Riker Laboratories, Inc. | Transdermal nitroglycerin delivery system |
| US5656286A (en) | 1988-03-04 | 1997-08-12 | Noven Pharmaceuticals, Inc. | Solubility parameter based drug delivery system and method for altering drug saturation concentration |
| US5252334A (en) | 1989-09-08 | 1993-10-12 | Cygnus Therapeutic Systems | Solid matrix system for transdermal drug delivery |
| US5688523A (en) | 1995-03-31 | 1997-11-18 | Minnesota Mining And Manufacturing Company | Method of making a pressure sensitive skin adhesive sheet material |
| US6365178B1 (en) | 1996-09-06 | 2002-04-02 | Watson Pharmaceuticals, Inc. | Method of making pressure sensitive adhesive matrix patches for transdermal drug delivery using hydrophilic salts of drugs and hydrophobic pressure sensitive adhesive dispersions |
| ATE229817T1 (de) | 1996-10-24 | 2003-01-15 | Alza Corp | Penetrationsfördernde substanzen für die transdermale verabreichung von wirkstoffen, vorrichtungen und verfahren zur herstellung |
| GB0017999D0 (en) | 2000-07-21 | 2000-09-13 | Smithkline Beecham Biolog | Novel device |
| GB0023008D0 (en) | 2000-09-20 | 2000-11-01 | Glaxo Group Ltd | Improvements in vaccination |
| US7176278B2 (en) | 2001-08-30 | 2007-02-13 | Biorexis Technology, Inc. | Modified transferrin fusion proteins |
| US20030054025A1 (en) | 2001-09-14 | 2003-03-20 | 3M Innovative Properties Company | Non-contact printing method for making a medical pressure sensitive adhesive article |
| WO2004020454A2 (en) * | 2002-08-30 | 2004-03-11 | Biorexis Pharmaceutical Corporation | Modified transferrin fusion proteins comprising duplicate transferrin amino or carboxy terminal domains |
| US20070060512A1 (en) * | 2003-03-04 | 2007-03-15 | Homayoun Sadeghi | Dipeptidyl-peptidase protected protein |
| US20040202708A1 (en) | 2003-04-14 | 2004-10-14 | 3M Innovative Properties Company | Transdermal drug delivery device with translucent inorganic barrier layer |
| US7659252B2 (en) | 2005-09-15 | 2010-02-09 | Novomed Technologies, Inc. (Shanghai) | Transdermal delivery peptides and method of use thereof |
| MX2008008548A (es) * | 2005-12-30 | 2008-09-10 | Evonik Roehm Gmbh | Peptidos utiles como petidos penetradores de celulas. |
| CN1879888B (zh) * | 2006-02-15 | 2011-04-13 | 中国科学技术大学 | 透皮给药增强剂及其使用方法 |
| WO2011066493A1 (en) | 2009-11-30 | 2011-06-03 | 3M Innovative Properties Company | Conformable barrier sheet, methods, and device |
| CA2811113A1 (en) * | 2010-11-09 | 2012-05-18 | The Regents Of The University Of California | Skin permeating and cell entering (space) peptides and methods of use thereof |
| KR101327555B1 (ko) * | 2011-03-11 | 2013-11-08 | 서울대학교산학협력단 | 모공을 통해 피부를 투과하는 경피 전달용 펩타이드 |
| WO2012167081A1 (en) | 2011-06-03 | 2012-12-06 | 3M Innovative Properties Company | Hydrazino 1h-imidazoquinolin-4-amines and conjugates made therefrom |
| CN102247603B (zh) * | 2011-06-13 | 2013-03-20 | 中国科学技术大学 | 一种具有透皮给药能力的融合蛋白 |
| CN102225206B (zh) * | 2011-06-17 | 2013-03-06 | 中国科学技术大学 | 一种增强透皮给药组合物及其应用 |
| WO2013112488A2 (en) | 2012-01-23 | 2013-08-01 | Kythera Biopharmaceuticals, Inc. | Dermal filling compositions and methods |
| CN103145799B (zh) * | 2013-02-18 | 2014-04-16 | 大连理工大学 | 一组具有促进经皮和跨膜渗透作用的多肽及其应用 |
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| WO2015023649A2 (en) | 2015-02-19 |
| EP3033056A4 (en) | 2017-03-22 |
| WO2015023649A3 (en) | 2015-04-09 |
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| US20160199498A1 (en) | 2016-07-14 |
| CN105491982A (zh) | 2016-04-13 |
| US9642895B2 (en) | 2017-05-09 |
| EP3033056B1 (en) | 2020-01-15 |
| JP2016527188A (ja) | 2016-09-08 |
| EP3033056A2 (en) | 2016-06-22 |
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