JP6059802B2 - 長時間作用型ｇｌｐ−１ペプチドの使用 - Google Patents

長時間作用型ｇｌｐ−１ペプチドの使用 Download PDF

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Publication number
JP6059802B2
JP6059802B2 JP2015519000A JP2015519000A JP6059802B2 JP 6059802 B2 JP6059802 B2 JP 6059802B2 JP 2015519000 A JP2015519000 A JP 2015519000A JP 2015519000 A JP2015519000 A JP 2015519000A JP 6059802 B2 JP6059802 B2 JP 6059802B2
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Prior art keywords
glp
agonist
xaa
peptide
glu
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Japanese (ja)
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JP2015522573A5 (https=
JP2015522573A (ja
Inventor
クリスティン・ビョルン・ジェンセン
マッズ・フレデリク・ラスムッセン
ミラン・ズドラヴコヴィッチ
ペーター・クリステンセン
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Novo Nordisk AS
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Novo Nordisk AS
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/26—Glucagons
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Immunology (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Endocrinology (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Obesity (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Child & Adolescent Psychology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
JP2015519000A 2012-07-01 2013-06-21 長時間作用型ｇｌｐ−１ペプチドの使用 Active JP6059802B2 (ja)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
EP12174535 2012-07-01
EP12174535.0 2012-07-01
US201261694837P 2012-08-30 2012-08-30
US61/694,837 2012-08-30
US201261708162P 2012-10-01 2012-10-01
US61/708,162 2012-10-01
EP12186781 2012-10-01
EP12186781.6 2012-10-01
PCT/EP2013/063004 WO2014005858A1 (en) 2012-07-01 2013-06-21 Use of long-acting glp-1 peptides

Publications (3)

Publication Number Publication Date
JP2015522573A JP2015522573A (ja) 2015-08-06
JP2015522573A5 JP2015522573A5 (https=) 2016-03-10
JP6059802B2 true JP6059802B2 (ja) 2017-01-11

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ID=65858459

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015519000A Active JP6059802B2 (ja) 2012-07-01 2013-06-21 長時間作用型ｇｌｐ−１ペプチドの使用

Country Status (17)

Country Link
US (2) US9764003B2 (https=)
EP (3) EP2866825B1 (https=)
JP (1) JP6059802B2 (https=)
AU (3) AU2013286177B2 (https=)
BR (1) BR112014032938A2 (https=)
CA (1) CA2877056A1 (https=)
DK (1) DK2866825T3 (https=)
ES (2) ES3041720T3 (https=)
HR (2) HRP20200889T1 (https=)
HU (2) HUE072859T2 (https=)
MX (3) MX366405B (https=)
PL (2) PL3689365T3 (https=)
PT (1) PT2866825T (https=)
RS (2) RS67258B1 (https=)
RU (2) RU2018117557A (https=)
SI (1) SI2866825T1 (https=)
WO (1) WO2014005858A1 (https=)

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PL2696687T3 (pl) 2011-04-12 2017-06-30 Novo Nordisk A/S Pochodne podwójnie acylowanej GLP-1
HRP20181447T1 (hr) 2012-03-22 2018-11-02 Novo Nordisk A/S Pripravci glp-1 peptida i njihova priprava
JP6517690B2 (ja) 2012-06-20 2019-05-22 ノヴォ ノルディスク アー／エス ペプチド及び送達剤を含む錠剤製剤
EP2866825B1 (en) 2012-07-01 2020-04-08 Novo Nordisk A/S Use of long-acting glp-1 peptides
KR102272671B1 (ko) 2013-05-02 2021-07-06 노보 노르디스크 에이/에스 Glp-1 화합물의 경구 투여
GB201621987D0 (en) * 2016-12-22 2017-02-08 Archer Virgil L See Archer Sheri A Arecor Ltd Novel composition
DE102017106216A1 (de) * 2017-03-22 2018-09-27 Amw Gmbh Extrudierte Depotform zur anhaltenden Wirkstofffreisetzung
KR102665710B1 (ko) 2017-08-24 2024-05-14 노보 노르디스크 에이/에스 Glp-1 조성물 및 그 용도
CA3078652A1 (en) * 2017-10-12 2019-04-18 Novo Nordisk A/S Semaglutide in medical therapy
GB201720187D0 (en) * 2017-12-04 2018-01-17 Imperial Innovations Ltd Novel Compounds
JP6898518B2 (ja) 2018-02-02 2021-07-07 ノヴォ ノルディスク アー／エス Ｇｌｐ−１アゴニスト、ｎ−（８−（２−ヒドロキシベンゾイル）アミノ）カプリル酸の塩及び滑沢剤を含む固形組成物
TWI705820B (zh) 2018-06-22 2020-10-01 美商美國禮來大藥廠 Gip/glp1促效劑組合物
US20210162013A1 (en) * 2018-08-03 2021-06-03 Brown University Compositions and methods for improving the bioavailability of glp1 and analogues thereof
CN113766930B (zh) * 2019-02-26 2025-07-22 特韦斯特生物科学公司 Glp1受体的变异核酸文库
WO2020180534A1 (en) 2019-03-01 2020-09-10 President And Fellows Of Harvard College Methods and compositions for protein delivery
IL291876A (en) 2019-11-06 2022-06-01 Novo Nordisk As Receptor agonists in glp-1 type dementia
EP4086277A4 (en) * 2019-12-30 2024-02-14 Gan & Lee Pharmaceuticals Co., Ltd. Long-acting glp-1 compound
TW202140058A (zh) 2020-01-30 2021-11-01 美商美國禮來大藥廠 提派肽（ｔｉｒｚｅｐａｔｉｄｅ）之治療用途
CN115484935A (zh) 2020-02-14 2022-12-16 G2G生物公司 包括含有glp-1类似物或其药学上可接受的盐的缓释微球的药物组合物
JP7761567B2 (ja) 2020-02-18 2025-10-28 ノヴォ ノルディスク アー／エス 医薬製剤
CN112768087A (zh) * 2020-12-23 2021-05-07 吉林大学 利用孟德尔随机化方法验证索马鲁肽口服制剂预防二型糖尿病的用途
JP2024527528A (ja) * 2021-06-24 2024-07-25 ギラ セラピューティクス インコーポレイテッド 満腹感を誘導する、及び代謝障害を治療するための方法及びキット
US12514908B2 (en) 2021-07-05 2026-01-06 Mapi Pharma Ltd. Semaglutide depot systems and use thereof
US11865213B2 (en) * 2021-07-05 2024-01-09 Mapi Pharma Ltd. Semaglutide depot systems and use thereof
PT4408840T (pt) 2021-09-27 2025-10-07 Terns Pharmaceuticals Inc Ácidos benzimidazolocarboxílicos como agonistas de glp-1r
CN118401519A (zh) 2021-10-25 2024-07-26 拓臻制药公司 作为glp-1r激动剂的化合物
AU2022386166A1 (en) 2021-11-10 2024-06-20 I2O Therapeutics, Inc. Ionic liquid compositions
CN114621339B (zh) * 2021-12-28 2022-09-23 北京惠之衡生物科技有限公司 一种长效glp-1衍生物
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CN121843690A (zh) 2023-07-24 2026-04-10 莱兰斯坦福初级大学评议会 用于递送治疗性肽的组合物和方法
WO2025165146A1 (ko) * 2024-01-29 2025-08-07 주식회사 티온랩테라퓨틱스 세마글루타이드 또는 티르제파타이드의 개선된 의료 요법 제공을 위한 비만 및 당뇨 치료용으로써, 소수성 이온 페어링 겔레이션을 통한 초기 방출이 제어된 데포 조성물 및 이의 제조방법
KR102930984B1 (ko) * 2024-01-29 2026-02-25 주식회사 티온랩테라퓨틱스 세마글루타이드의 개선된 의료 요법 제공을 위한 비만 및 당뇨 치료용로써, 소수성 이온 페어링 겔레이션을 통한 초기 방출이 제어된 데포 조성물 및 이의 제조방법
WO2026046328A1 (en) * 2024-08-30 2026-03-05 Beijing Ql Biopharmaceutical Co., Ltd. Dosing regimen of glp-1 conjugates
CN118845644B (zh) * 2024-09-27 2025-01-17 杭州信海医药科技有限公司 一种司美格鲁肽注射液的制备方法

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KR20200077621A (ko) * 2014-10-16 2020-06-30 얀마 파워 테크놀로지 가부시키가이샤 작업 차량
KR102321242B1 (ko) * 2014-10-16 2021-11-02 얀마 파워 테크놀로지 가부시키가이샤 작업 차량

Also Published As

Publication number Publication date
US20150190474A1 (en) 2015-07-09
US9764003B2 (en) 2017-09-19
HUE072859T2 (hu) 2025-12-28
DK2866825T3 (da) 2020-06-08
HUE049152T2 (hu) 2020-09-28
HRP20200889T1 (hr) 2020-09-04
WO2014005858A1 (en) 2014-01-09
MX2019008148A (es) 2019-09-05
AU2018202504A1 (en) 2018-05-10
RU2657573C2 (ru) 2018-06-14
AU2020202573A1 (en) 2020-05-07
JP2015522573A (ja) 2015-08-06
AU2013286177B2 (en) 2018-04-26
EP3689365C0 (en) 2025-08-06
EP3689365A1 (en) 2020-08-05
HRP20251088T1 (hr) 2025-11-07
AU2013286177A1 (en) 2015-01-15
EP2866825B1 (en) 2020-04-08
EP4406593A3 (en) 2024-10-23
US20180085435A1 (en) 2018-03-29
RS60432B1 (sr) 2020-07-31
SI2866825T1 (sl) 2020-07-31
CA2877056A1 (en) 2014-01-09
AU2020202573B2 (en) 2023-04-20
EP4406593A2 (en) 2024-07-31
US10335462B2 (en) 2019-07-02
ES3041720T3 (en) 2025-11-14
MX376058B (es) 2025-03-07
MX2014014946A (es) 2015-04-08
EP2866825A1 (en) 2015-05-06
PL2866825T3 (pl) 2021-02-22
BR112014032938A2 (pt) 2017-08-01
RS67258B1 (sr) 2025-10-31
MX2020010693A (es) 2020-11-06
MX366405B (es) 2019-07-08
PT2866825T (pt) 2020-07-15
AU2018202504B2 (en) 2020-05-07
PL3689365T3 (pl) 2025-11-12
RU2018117557A (ru) 2019-03-22
ES2796839T3 (es) 2020-11-30
RU2015101826A (ru) 2016-08-20
RU2018117557A3 (https=) 2021-08-20
EP3689365B1 (en) 2025-08-06

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